GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5696 products of "GPCR/G-Protein"

Purity (%)

100

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MK-0557
CAS:
- 328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
Formula:C₂₂H₁₉FN₄O₃
Purity:99.88%
Color and Shape:Solid
Molecular weight:406.41
Ref: TM-TQ0286
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GLP-1(7-36), amide
CAS:
- 107444-51-9
GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.
Formula:C₁₄₉H₂₂₆N₄₀O₄₅
Purity:99.85%
Color and Shape:White Powder
Molecular weight:3297.63
Ref: TM-T3984
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tcY-NH2 TFA(327177-34-4 free base)
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
Formula:C₄₂H₅₀F₃N₇O₉
Purity:>99.99%
Color and Shape:Solid
Molecular weight:853.9
Ref: TM-TP1925L
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Decloxizine
CAS:
- 3733-63-9
Decloxizine is a H1 receptor antagonist
Formula:C₂₁H₂₈N₂O₂
Purity:99.53%
Color and Shape:White Or Similar To White Powder
Molecular weight:340.46
Ref: TM-T22713
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PF-06882961 Tris
CAS:
- 2230198-03-3
PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:C₃₅H₄₁FN₆O₇
Purity:98.74% - 99.79%
Color and Shape:Solid
Molecular weight:676.7
Ref: TM-T8876
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Serotonin
CAS:
- 50-67-9
Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!
Formula:C₁₀H₁₂N₂O
Purity:97.47% - 99.92%
Color and Shape:Solid
Molecular weight:176.22
Ref: TM-TN2437
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Otenabant
CAS:
- 686344-29-6
Otenabant (CP-945598) has been investigated for the treatment of Obesity.
Formula:C₂₅H₂₅Cl₂N₇O
Purity:99.43%
Color and Shape:Solid
Molecular weight:510.42
Ref: TM-T3530
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CPI-444
CAS:
- 1202402-40-1
CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.
Formula:C₂₀H₂₁N₇O₃
Purity:98.78%
Color and Shape:Solid
Molecular weight:407.43
Ref: TM-T7183
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OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).
Formula:C₇₉H₁₂₅N₂₃O₂₂
Purity:98.52%
Color and Shape:Solid
Molecular weight:1748.98
Ref: TM-TP1973L
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Vericiguat
CAS:
- 1350653-20-1
Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.
Formula:C₁₉H₁₆F₂N₈O₂
Purity:98.86% - 99.93%
Color and Shape:Solid
Molecular weight:426.38
Ref: TM-T17226
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Rimegepant
CAS:
- 1289023-67-1
View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.
Formula:C₂₈H₂₈F₂N₆O₃
Purity:99.1% - 99.99%
Color and Shape:Solid
Molecular weight:534.56
Ref: TM-T4610
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Senktide
CAS:
- 106128-89-6
Senktide is an agonist of tachykinin NK3 receptor.
Formula:C₄₀H₅₅N₇O₁₁S
Purity:99.84% - >99.99%
Color and Shape:White Powder
Molecular weight:841.97
Ref: TM-T7633
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Sarpogrelate hydrochloride
CAS:
- 135159-51-2
Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Formula:C₂₄H₃₂ClNO₆
Purity:99.73%
Color and Shape:Colorless Liquid
Molecular weight:465.97
Ref: TM-T4978
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β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.
Formula:C₁₂₀H₁₇₈N₃₄O₃₇S
Purity:99.64%
Color and Shape:Solid
Molecular weight:2720.97
Ref: TM-TP1004L
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Tetrahydrozoline hydrochloride
CAS:
- 522-48-5
Tetrahydrozoline hydrochloride (Murine Plus) is an imidazoline derivative with alpha receptor agonist activity.
Formula:C₁₃H₁₆N₂·HCl
Purity:99.90%
Color and Shape:Off-White Solid
Molecular weight:236.74
Ref: TM-T6703
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Mesdopetam hemitartrate
CAS:
- 2562346-14-7
Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.
Formula:C₂₈H₄₂F₂N₂O₁₂S₂
Purity:99.98%
Color and Shape:Solid
Molecular weight:700.77
Ref: TM-T9409
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Desmopressin acetate (16679-58-6 free base)
CAS:
- 62288-83-9
Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.
Formula:C₄₈H₆₈N₁₄O₁₄S₂
Purity:98.84% - >99.99%
Color and Shape:Solid
Molecular weight:1129.26
Ref: TM-T5144
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JNJ-5207852 dihydrochloride
CAS:
- 1782228-76-5
JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor
Formula:C₂₀H₃₄Cl₂N₂O
Purity:99.51%
Color and Shape:Solid
Molecular weight:389.4
Ref: TM-T8822
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Brexpiprazole
CAS:
- 913611-97-9
Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
Formula:C₂₅H₂₇N₃O₂S
Purity:99.06% - 99.96%
Color and Shape:Solid
Molecular weight:433.57
Ref: TM-T2306
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Guanfacine hydrochloride
CAS:
- 29110-48-3
Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
Formula:C₉H₁₀Cl₃N₃O
Purity:99.89% - 99.91%
Color and Shape:Solid
Molecular weight:282.55
Ref: TM-T2150
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Lerisetron
CAS:
- 143257-98-1
Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.
Formula:C₁₈H₂₀N₄
Purity:99.15% - 99.82%
Color and Shape:Solid
Molecular weight:292.38
Ref: TM-T8441
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Histrelin acetate
CAS:
- 220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.
Formula:C₆₈H₉₀N₁₈O₁₄
Purity:99.92%
Color and Shape:Solid
Molecular weight:1383.55
Ref: TM-TP2107L
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Regadenoson hydrate
CAS:
- 875148-45-1
Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.
Formula:C₁₅H₂₀N₈O₆
Purity:98%
Color and Shape:Solid
Molecular weight:408.37
Ref: TM-T26054
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SCH442416
CAS:
- 316173-57-6
SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).
Formula:C₂₀H₁₉N₇O₂
Purity:99.58%
Color and Shape:Solid
Molecular weight:389.41
Ref: TM-T23336
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Montelukast dicyclohexylamine
CAS:
- 577953-88-9
Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.
Formula:C₄₇H₅₉ClN₂O₃S
Color and Shape:Solid
Molecular weight:767.5
Ref: TM-T72145
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Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
Purity:98.27%
Color and Shape:Liquid
Molecular weight:N/A
Ref: TM-TP2071L
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Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.
Purity:95.44% - 99.73%
Color and Shape:Solid
Molecular weight:N/A
Ref: TM-TP1199L
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Xaliproden hydrochloride
CAS:
- 90494-79-4
Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.
Formula:C₂₄H₂₃ClF₃N
Purity:99.99%
Color and Shape:Solid
Molecular weight:417.89
Ref: TM-T9272
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Antalarmin
CAS:
- 157284-96-3
Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.
Formula:C₂₄H₃₄N₄
Color and Shape:Solid
Molecular weight:378.55
Ref: TM-T70433
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Neuropeptide S (Rat) acetate
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.
Formula:C₉₇H₁₆₄N₃₄O₂₉
Purity:95.36%
Color and Shape:Solid
Molecular weight:2270.59
Ref: TM-TP1982L
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BRL-15572 dihydrochloride
CAS:
- 193611-72-2
BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.
Formula:C₂₅H₂₇ClN₂O·2HCl
Purity:99.74%
Color and Shape:Solid
Molecular weight:479.87
Ref: TM-T6423
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PD 168568
CAS:
- 210688-56-5
PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.
Formula:C₂₂H₂₇N₃O
Color and Shape:Solid
Molecular weight:349.47
Ref: TM-T73215
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PACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), not VIP1.
Purity:98.16%
Color and Shape:Liquid
Molecular weight:N/A
Ref: TM-TP1878L
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Mecamylamine
CAS:
- 60-40-2
Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.
Formula:C₁₁H₂₁N
Color and Shape:Solid
Molecular weight:167.29
Ref: TM-T69019
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NNC-0640
CAS:
- 307986-98-7
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
Formula:C₂₉H₃₁N₇O₄S
Purity:97.04%
Color and Shape:Solid
Molecular weight:573.67
Ref: TM-T7364
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Parmodulin 2
CAS:
- 423735-93-7
ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).
Formula:C₁₇H₁₇BrN₂O₂
Purity:97.35% - 99.95%
Color and Shape:Solid
Molecular weight:361.23
Ref: TM-T1893
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Exo1
CAS:
- 75541-83-2
Exo1 is an inhibitor of the exocytic pathway
Formula:C₁₅H₁₂FNO₃
Purity:98.75%
Color and Shape:Solid
Molecular weight:273.26
Ref: TM-T4609
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Solabegron HCl
CAS:
- 451470-34-1
Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.
Formula:C₂₃H₂₄Cl₂N₂O₃
Color and Shape:Solid
Molecular weight:447.35
Ref: TM-T12970L
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Napitane Mesylate
CAS:
- 149189-73-1
Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.
Formula:C₂₃H₂₉NO₅S
Purity:98%
Color and Shape:Solid
Molecular weight:431.55
Ref: TM-T26363
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AP1189 acetate
CAS:
- 959850-74-9
AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.
Formula:C₁₆H₁₈N₆O₄
Purity:99.95%
Color and Shape:Solid
Molecular weight:358.35
Ref: TM-T9596
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Apraclonidine
CAS:
- 66711-21-5
Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.
Formula:C₉H₁₀Cl₂N₄
Color and Shape:Solid
Molecular weight:245.11
Ref: TM-T60350
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Eltoprazine
CAS:
- 98224-03-4
Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.
Formula:C₁₂H₁₆N₂O₂
Color and Shape:Solid
Molecular weight:220.27
Ref: TM-T38145
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Riociguat
CAS:
- 625115-55-1
Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterial
Formula:C₂₀H₁₉FN₈O₂
Purity:99.28% - 99.95%
Color and Shape:Solid
Molecular weight:422.42
Ref: TM-T6968
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Hydroxyzine
CAS:
- 68-88-2
Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
Formula:C₂₁H₂₇ClN₂O₂
Purity:99.54% - ≥95%
Color and Shape:Oil Solid
Molecular weight:374.9
Ref: TM-T20884
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GUANABENZ
CAS:
- 5051-62-7
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
Formula:C₈H₈Cl₂N₄
Purity:98.31%
Color and Shape:White Solid From Acetonitrile Solid
Molecular weight:231.08
Ref: TM-T5471
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Pranlukast hemihydrate
CAS:
- 150821-03-7
Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.
Formula:C₂₇H₂₃N₅O₄₀·5H₂O
Purity:99.28%
Color and Shape:Solid
Molecular weight:490.52
Ref: TM-T63291
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Batefenterol
CAS:
- 743461-65-6
Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).
Formula:C₄₀H₄₂ClN₅O₇
Purity:97.94% - 98.4%
Color and Shape:Solid
Molecular weight:740.24
Ref: TM-T7079
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Carazolol
CAS:
- 57775-29-8
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
Formula:C₁₈H₂₂N₂O₂
Purity:99% - 99.53%
Color and Shape:Yellowish Solid
Molecular weight:298.38
Ref: TM-T3284
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ARC-239
CAS:
- 67339-62-2
ARC-239 is an agonist of α2-adrenergic receptor.
Formula:C₂₄H₂₉N₃O₃
Color and Shape:Solid
Molecular weight:407.51
Ref: TM-T26651
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Alizapride
CAS:
- 59338-93-1
Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].
Formula:C₁₆H₂₁N₅O₂
Color and Shape:Solid
Molecular weight:315.37
Ref: TM-T60813
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Prazosin
CAS:
- 19216-56-9
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Formula:C₁₉H₂₁N₅O₄
Purity:99.86%
Color and Shape:White To Tan Powder Solid
Molecular weight:383.4
Ref: TM-T22406
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MK-571 sodium
CAS:
- 115103-85-0
MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.
Formula:C₂₆H₂₇ClN₂O₃S₂·Na
Purity:97.86% - 99.58%
Color and Shape:Solid
Molecular weight:537.07
Ref: TM-T3148
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Cetirizine Impurity B dihydrochloride
CAS:
- 1000690-91-4
Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.
Formula:C₁₉H₂₃Cl₃N₂O₂
Purity:97.33%
Color and Shape:Solid
Molecular weight:417.76
Ref: TM-T9084
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E7046
CAS:
- 1369489-71-3
E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.
Formula:C₂₂H₁₈F₅N₃O₄
Purity:99.86%
Color and Shape:Solid
Molecular weight:483.4
Ref: TM-TQ0025
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Pimavanserin
CAS:
- 706779-91-1
Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.
Formula:C₂₅H₃₄FN₃O₂
Purity:97.84% - 99.69%
Color and Shape:Pale Yellow To Pale Orange Solid
Molecular weight:427.55
Ref: TM-T2076
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[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:
- 125580-28-1
[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 receptor with anxiolytic effects.
Formula:C₁₉₀H₂₈₆N₅₄O₅₆
Purity:99.39%
Color and Shape:Solid
Molecular weight:4223
Ref: TM-TP2206
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Amylin, amide, rat acetate(124447-81-0,free base)
Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.
Formula:C₁₆₉H₂₇₆N₅₂O₅₅S₂
Purity:98.93%
Color and Shape:Solid
Molecular weight:3980.45
Ref: TM-TP1232L
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β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor
Formula:C₁₆₄H₂₇₁N₅₁O₅₀S₃
Purity:99.35%
Color and Shape:Solid
Molecular weight:3853.46
Ref: TM-TP2167
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Eprazinone dihydrochloride
CAS:
- 10402-53-6
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
Formula:C₂₄H₃₂N₂O₂·2HCl
Purity:99.25%
Color and Shape:A White Or Almost White Crys
Molecular weight:453.44
Ref: TM-T3034
+ Info
Azaperone
CAS:
- 1649-18-9
Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.
Formula:C₁₉H₂₂FN₃O
Purity:98.73%
Color and Shape:White Or Off-White Crystalline
Molecular weight:327.4
Ref: TM-T6398
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Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.
Formula:C₉₁H₁₄₃N₂₇O₂₆S₄
Purity:99.41%
Color and Shape:Solid
Molecular weight:2157
Ref: TM-TP1104L
+ Info
[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2
Formula:C₄₀H₆₈N₈O₁₀
Purity:99.31%
Color and Shape:Solid
Molecular weight:821.02
Ref: TM-T38807L
+ Info
Selexipag
CAS:
- 475086-01-2
Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.
Formula:C₂₆H₃₂N₄O₄S
Purity:99.98% - >99.99%
Color and Shape:Solid
Molecular weight:496.62
Ref: TM-T3216
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Substance P (7-11)
CAS:
- 51165-05-0
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
Formula:C₃₁H₄₄N₆O₅S
Purity:98.39%
Color and Shape:Solid
Molecular weight:612.78
Ref: TM-T7554
+ Info
Xanthotoxol
CAS:
- 2009-24-7
Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.
Formula:C₁₁H₆O₄
Purity:99.97%
Color and Shape:Solid
Molecular weight:202.16
Ref: TM-T4S1659
+ Info
Methiothepin mesylate
CAS:
- 74611-28-2
Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
Formula:C₂₁H₂₈N₂O₃S₃
Purity:98% - 99.92%
Color and Shape:Solid
Molecular weight:452.65
Ref: TM-T2190
+ Info
Praliciguat
CAS:
- 1628730-49-3
Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.
Formula:C₂₁H₁₄F₈N₆O₂
Purity:98.82%
Color and Shape:Solid
Molecular weight:534.36
Ref: TM-T16569
+ Info
Facinicline (free base)
CAS:
- 677306-35-3
Facinicline (free base) is a partial agonist of the nicotinic alpha-7 (α7) receptor. It is used for the oral treatment of Alzheimer's.
Formula:C₁₅H₁₈N₄O
Color and Shape:Solid
Molecular weight:270.33
Ref: TM-T31741
+ Info
BMY 7378 dihydrochloride
CAS:
- 21102-95-4
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
Formula:C₂₂H₃₃Cl₂N₃O₃
Purity:97.32% - 99.08%
Color and Shape:Solid
Molecular weight:458.42
Ref: TM-T3046
+ Info
Tirzepatide Acetate(2023788-19-2 free base)
Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.
Formula:C₂₂₇H₃₅₂N₄₈O₇₀
Purity:97.3% - 98.05%
Color and Shape:Solid
Molecular weight:4873.5
Ref: TM-TP1111L
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5-Benzyloxygramine
CAS:
- 1453-97-0
5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
Formula:C₁₈H₂₀N₂O
Purity:99.13%
Color and Shape:Solid
Molecular weight:280.36
Ref: TM-T35841
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Acitazanolast
CAS:
- 114607-46-4
Acitazanolast (WP-871) is an anti-allergic drug candidate.
Formula:C₉H₇N₅O₃
Purity:98.25%
Color and Shape:Solid
Molecular weight:233.18
Ref: TM-T7812
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Melitracen hydrochloride
CAS:
- 10563-70-9
Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.
Formula:C₂₁H₂₆ClN
Purity:99.99%
Color and Shape:Crystalline Solid
Molecular weight:327.90
Ref: TM-T4274
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Abaperidone Hydrochloride
CAS:
- 183849-45-8
Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.
Formula:C₂₅H₂₆ClFN₂O₅
Color and Shape:Solid
Molecular weight:488.94
Ref: TM-T26508
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[Pyr1]-Apelin-13
CAS:
- 217082-60-5
[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.
Formula:C₆₉H₁₀₈N₂₂O₁₆S
Purity:99.71%
Color and Shape:Solid
Molecular weight:1533.8
Ref: TM-TP1260
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VPC171
CAS:
- 1018830-99-3
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
Formula:C₁₈H₁₂F₃NOS
Purity:99.78%
Color and Shape:Solid
Molecular weight:347.35
Ref: TM-T29112
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Mequitazine
CAS:
- 29216-28-2
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
Formula:C₂₀H₂₂N₂S
Purity:99.98%
Color and Shape:Solid
Molecular weight:322.47
Ref: TM-T4499
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S 38093 HCl
CAS:
- 1222097-72-4
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
Formula:C₁₇H₂₅ClN₂O₂
Purity:97.91%
Color and Shape:Solid
Molecular weight:324.85
Ref: TM-T4087
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Fipamezole HCl
CAS:
- 150586-72-4
Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.
Formula:C₁₄H₁₆ClFN₂
Color and Shape:Solid
Molecular weight:266.74
Ref: TM-T27321
+ Info
MF-766
CAS:
- 1050656-06-8
MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.
Formula:C₂₇H₂₁F₃N₂O₃
Purity:99.54% - 99.59%
Color and Shape:Solid
Molecular weight:478.46
Ref: TM-T9622
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Vilazodone Hydrochloride
CAS:
- 163521-08-2
Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the
Formula:C₂₆H₂₇N₅O₂·HCl
Purity:99.56% - >99.99%
Color and Shape:Solid
Molecular weight:477.99
Ref: TM-T6232
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ESI-09
CAS:
- 263707-16-0
ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.
Formula:C₁₆H₁₅ClN₄O₂
Purity:97.24% - 99.57%
Color and Shape:Solid
Molecular weight:330.77
Ref: TM-T2244
+ Info
ML382
CAS:
- 1646499-97-9
ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
Formula:C₁₈H₂₀N₂O₄S
Purity:99.79%
Color and Shape:Solid
Molecular weight:360.43
Ref: TM-T8538
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Ciproxifan maleate
CAS:
- 184025-19-2
Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity
Formula:C₂₀H₂₂N₂O₆
Purity:99.39%
Color and Shape:Solid
Molecular weight:386.4
Ref: TM-T2004
+ Info
AM095
CAS:
- 1345614-59-6
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.
Formula:C₂₇H₂₃N₂NaO₅
Purity:98.87%
Color and Shape:Solid
Molecular weight:478.47
Ref: TM-T2000
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AHN 1-055 hydrochloride
CAS:
- 202646-03-5
AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).
Formula:C₂₁H₂₄ClF₂NO
Purity:99.89%
Color and Shape:Solid
Molecular weight:379.87
Ref: TM-T39429
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Raclopride
CAS:
- 84225-95-6
Raclopride is a selective antagonist of dopamine D2/D3 receptor.
Formula:C₁₅H₂₀Cl₂N₂O₃
Purity:99.17%
Color and Shape:Solid
Molecular weight:347.24
Ref: TM-T7635
+ Info
ACEPROMAZINE MALEATE
CAS:
- 3598-37-6
ACEPROMAZINE MALEATE is a dopamine receptor antagonist
Formula:C₂₃H₂₆N₂O₅S
Purity:98.87% - 99.51%
Color and Shape:Off White Or Yellow Crystalline Powder
Molecular weight:442.53
Ref: TM-T7728
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KB-5492 anhydrous
CAS:
- 129200-10-8
KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.
Formula:C₂₇H₃₄N₂O₁₀
Color and Shape:Solid
Molecular weight:546.57
Ref: TM-T24254
+ Info
Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.
Formula:C₃₅H₄₇FN₁₀O₈
Purity:97.97%
Color and Shape:Solid
Molecular weight:754.85
Ref: TM-TP1127L1
+ Info
Perospirone
CAS:
- 150915-41-6
Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
Formula:C₂₃H₃₀N₄O₂S
Purity:99.23%
Color and Shape:White Powder
Molecular weight:426.57
Ref: TM-T4576
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DAPTA
CAS:
- 106362-34-9
DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.
Formula:C₃₅H₅₆N₁₀O₁₅
Purity:>99.99%
Color and Shape:Solid
Molecular weight:856.88
Ref: TM-T7624
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Bevantolol hydrochloride
CAS:
- 42864-78-8
Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
Formula:C₂₀H₂₈ClNO₄
Purity:99.49%
Color and Shape:Solid
Molecular weight:381.9
Ref: TM-T8143
+ Info
Pimozide
CAS:
- 2062-78-4
Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.
Formula:C₂₈H₂₉F₂N₃O
Purity:99.63% - >99.99%
Color and Shape:Solid
Molecular weight:461.55
Ref: TM-T2546
+ Info
L-DOPA methyl ester (hydrochloride)
CAS:
- 1421-65-4
L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formula:C₁₀H₁₄ClNO₄
Purity:98.69% - 99.81%
Color and Shape:White Solid
Molecular weight:247.675
Ref: TM-T7654
+ Info
Fuscoside
CAS:
- 131631-89-5
Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.
Formula:C₂₆H₃₁N₃O₄
Purity:98.13% - 99.66%
Color and Shape:Solid
Molecular weight:449.54
Ref: TM-T4355
+ Info
Cinaciguat hydrochloride
CAS:
- 646995-35-9
Cinaciguat( BAY582667, BAY58-2667) is a soluble guanosine cyclase activator that can prevent cardiac dysfunction in rat models of type 1 diabetes.
Formula:C₃₆H₄₀ClNO₅
Color and Shape:Solid
Molecular weight:602.17
Ref: TM-T1984L
+ Info
Pitolisant hydrochloride
CAS:
- 903576-44-3
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).
Formula:C₁₇H₂₇Cl₂NO
Purity:99.72% - 99.91%
Color and Shape:Solid
Molecular weight:332.31
Ref: TM-T7176
+ Info
Chlorphenesin
CAS:
- 104-29-0
Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.
Formula:C₉H₁₁ClO₃
Purity:99.59%
Color and Shape:Solid
Molecular weight:202.63
Ref: TM-T4507
+ Info
Ocaperidone
CAS:
- 129029-23-8
Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.
Formula:C₂₄H₂₅FN₄O₂
Purity:99.33%
Color and Shape:Solid
Molecular weight:420.48
Ref: TM-T3497