GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(985 products)
- Adenosine Receptor(244 products)
- Adrenergic Receptor(2,991 products)
- Bombesin Receptor(32 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(209 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(181 products)
- Hedgehog/Smoothened(46 products)
- Histamine Receptor(380 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(309 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5696 products of "GPCR/G-Protein"
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Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formula:C22H21Cl3N4OPurity:98% - 99.91%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:463.79Metaproterenol hemisulfate
CAS:<p>Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.</p>Formula:C11H17NO3·5H2O4SPurity:98.53% - 99.74%Color and Shape:SolidMolecular weight:260.3Nylidrin hydrochloride
CAS:Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.Formula:C19H26ClNO2Purity:99.35%Color and Shape:SolidMolecular weight:335.87Clonidine hydrochloride
CAS:Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formula:C9H10Cl3N3Purity:99.16% - 99.86%Color and Shape:SolidMolecular weight:266.55Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Formula:C16H26ClNO3Purity:99.94% - ≥95%Color and Shape:SolidMolecular weight:315.84Silodosin
CAS:Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.Formula:C25H32F3N3O4Purity:99.282% - 99.76%Color and Shape:Colorless To Pink SolidMolecular weight:495.53Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Formula:C17H28ClNO2Purity:97.32% - 99.86%Color and Shape:White Crystalline PowderMolecular weight:313.86Roxatidine Acetate hydrochloride
CAS:Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Formula:C18H26ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:367.87Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Formula:C10H13NO4Purity:98.95% - 99.86%Color and Shape:Less Or Almost Colorless Crystals Or White To Yellowish-White FineMolecular weight:211.21AH 6809
CAS:<p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>Formula:C17H14O5Purity:97.59%Color and Shape:SolidMolecular weight:298.29(3aR,9aR)-Fluparoxan
CAS:<p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H10FNO2Purity:97.82%Color and Shape:SoildMolecular weight:195.19Fluvoxamine maleate
CAS:<p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>Formula:C19H25F3N2O6Purity:99.92% - 99.94%Color and Shape:White Crystalline PowderMolecular weight:434.41Talastine
CAS:Talastine is an antihistamine compound that can induce an allergic rash.Formula:C19H21N3OPurity:99.44% - 99.84%Color and Shape:SolidMolecular weight:307.39(R)-Elagolix
CAS:<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Formula:C32H30F5N3O5Purity:99.08%Color and Shape:SolidMolecular weight:631.59Aripiprazole
CAS:Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formula:C23H27Cl2N3O2Purity:99.43% - 99.62%Color and Shape:Colourless Flake Crystalline SolidMolecular weight:448.39Levosulpiride
CAS:<p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>Formula:C15H23N3O4SPurity:98.20% - 99.88%Color and Shape:White Crystalline PowderMolecular weight:341.43Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H11ClFNO2Purity:99.98%Color and Shape:SoildMolecular weight:231.65Lafutidine
CAS:<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Formula:C22H29N3O4SPurity:98.55%Color and Shape:Yellowish White Crystalline PowderMolecular weight:431.55Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Formula:C21H24ClNOPurity:99.77% - >99.99%Color and Shape:White To Slightly Yellowish Crystalline SolidMolecular weight:341.88
