
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Palonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurity:99.84% - 99.92%Color and Shape:White SolidMolecular weight:332.87Ro 10-5824 dihydrochloride
CAS:Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formula:C17H22Cl2N4Purity:99.79%Color and Shape:SolidMolecular weight:353.29Moxisylyte hydrochloride
CAS:Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.Formula:C16H26ClNO3Purity:99.94% - ≥95%Color and Shape:SolidMolecular weight:315.84Ziprasidone hydrochloride
CAS:<p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>Formula:C21H22CL2N4OSPurity:97.97% - 99.82%Color and Shape:SolidMolecular weight:449.4Vilazodone
CAS:<p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>Formula:C26H27N5O2Purity:99.61%Color and Shape:Light Yellow SolidMolecular weight:441.52Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Formula:C22H34Cl2N2O2Purity:98.55%Color and Shape:SolidMolecular weight:429.42Dimenhydrinate
CAS:Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.Formula:C24H28ClN5O3Purity:99.57% - 99.77%Color and Shape:Crystals Physical Description Crystalline White Powder (Ntp 1992)Molecular weight:469.96Adrenalone hydrochloride
CAS:Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.Formula:C9H11NO3·HClPurity:99.94%Color and Shape:SolidMolecular weight:217.65Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurity:99.64%Color and Shape:Light Yellow To Yellow SolidMolecular weight:396.51Promazine hydrochloride
CAS:Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formula:C17H21ClN2SPurity:99.90%Color and Shape:SolidMolecular weight:320.88Acebutolol hydrochloride
CAS:<p>Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.</p>Formula:C18H29ClN2O4Purity:99.92% - >99.99%Color and Shape:White Or Slightly Off-White Crystalline Powder SolidMolecular weight:372.89Pizotifen
CAS:<p>Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.</p>Formula:C19H21NSPurity:99.93%Color and Shape:SolidMolecular weight:295.44Linaclotide
CAS:<p>Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.</p>Formula:C59H79N15O21S6Purity:97.93% - 98.71%Color and Shape:SolidMolecular weight:1526.74MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Formula:C27H25N3O4S2Purity:97.44%Color and Shape:SolidMolecular weight:519.64Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formula:C15H20N2O2·HClPurity:99.64% - 99.92%Color and Shape:SolidMolecular weight:296.79Clozapine
CAS:<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formula:C18H19ClN4Purity:99.91% - 99.93%Color and Shape:Yellow Crystals From Acetone-Petroleum Ether SolidMolecular weight:326.82Cetirizine dihydrochloride
CAS:Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.Formula:C21H27Cl3N2O3Purity:99.4% - 99.97%Color and Shape:SolidMolecular weight:461.81Olinciguat
CAS:<p>Olinciguat (IW-1701) is an oral guanylate cyclase (sGC) stimulator.</p>Formula:C21H16F5N7O3Purity:99.33% - 99.71%Color and Shape:SolidMolecular weight:509.39Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Formula:C19H29ClN2O4Purity:99.49%Color and Shape:SolidMolecular weight:384.9Tipepidine hydrochloride
CAS:Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.Formula:C15H18ClNS2Purity:99.97%Color and Shape:SolidMolecular weight:311.89
