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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5981 products of "GPCR/G-Protein"

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  • Chlorphenoxamine

    CAS:
    Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
    Formula:C18H22ClNO
    Purity:99.44% - 99.85%
    Color and Shape:Solid
    Molecular weight:303.83

    Ref: TM-T7564

    2mg
    35.00€
    5mg
    51.00€
    10mg
    81.00€
    25mg
    106.00€
    50mg
    147.00€
    100mg
    207.00€
    200mg
    306.00€
    1mL*10mM (DMSO)
    63.00€
  • Tecalcet Free Base

    CAS:
    Tecalcet Free Base is an oral calcium receptor agonist
    Formula:C18H22ClNO
    Color and Shape:Solid
    Molecular weight:303.83

    Ref: TM-T70555

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Vipadenant

    CAS:
    Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).
    Formula:C16H15N7O
    Purity:97.25% - 97.36%
    Color and Shape:Solid
    Molecular weight:321.34

    Ref: TM-T2373

    2mg
    35.00€
    5mg
    51.00€
    10mg
    80.00€
    25mg
    131.00€
    50mg
    210.00€
    100mg
    313.00€
    200mg
    445.00€
    1mL*10mM (DMSO)
    215.00€
  • Tozadenant

    CAS:
    Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
    Formula:C19H26N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.5

    Ref: TM-T7320

    5mg
    44.00€
    10mg
    67.00€
    25mg
    113.00€
    50mg
    190.00€
    100mg
    274.00€
    200mg
    394.00€
    1mL*10mM (DMSO)
    48.00€
  • Gadolinium chloride

    CAS:
    Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
    Formula:Cl3Gd
    Purity:98%
    Color and Shape:White Crystalline Solid
    Molecular weight:263.61

    Ref: TM-T22795

    25mg
    48.00€
    50mg
    58.00€
    100mg
    89.00€
    200mg
    126.00€
  • Dexmedetomidine hydrochloride

    CAS:
    Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.
    Formula:C13H16N2·HCl
    Purity:99.94% - 99.94%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:236.74

    Ref: TM-T6466

    5mg
    42.00€
    10mg
    55.00€
    25mg
    88.00€
    50mg
    159.00€
    100mg
    226.00€
    200mg
    340.00€
    500mg
    563.00€
    1mL*10mM (DMSO)
    50.00€
  • Vorapaxar sulfate

    CAS:
    Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.
    Formula:C29H35FN2O8S
    Purity:99.9% - >99.99%
    Color and Shape:Solid
    Molecular weight:590.66

    Ref: TM-T3098

    1mg
    38.00€
    2mg
    49.00€
    5mg
    79.00€
    10mg
    119.00€
    25mg
    210.00€
    50mg
    354.00€
    100mg
    528.00€
    500mg
    1,159.00€
    1mL*10mM (DMSO)
    99.00€
  • AVN-492

    CAS:
    AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
    Formula:C17H21N5O2S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:359.45

    Ref: TM-T5179

    1mg
    39.00€
    2mg
    49.00€
    5mg
    81.00€
    10mg
    120.00€
    25mg
    236.00€
    50mg
    354.00€
    100mg
    510.00€
    1mL*10mM (DMSO)
    89.00€
  • Zafirlukast

    CAS:
    Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and anti-inflammatory effects. Cost-effective and quality-assured.
    Formula:C31H33N3O6S
    Purity:99% - 99.83%
    Color and Shape:Solid
    Molecular weight:575.68

    Ref: TM-T6736

    10mg
    35.00€
    25mg
    49.00€
    50mg
    70.00€
    100mg
    92.00€
    500mg
    264.00€
    1mL*10mM (DMSO)
    62.00€
  • Naftopidil hydrochloride

    CAS:
    Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.
    Formula:C24H29ClN2O3
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:428.95

    Ref: TM-T9220

    1mg
    44.00€
    5mg
    87.00€
    10mg
    117.00€
    25mg
    202.00€
    50mg
    304.00€
    100mg
    437.00€
    200mg
    612.00€
    1mL*10mM (DMSO)
    97.00€
  • CPI-444

    CAS:
    CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.
    Formula:C20H21N7O3
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:407.43

    Ref: TM-T7183

    2mg
    34.00€
    5mg
    52.00€
    10mg
    73.00€
    25mg
    128.00€
    50mg
    197.00€
    100mg
    295.00€
    200mg
    442.00€
    1mL*10mM (DMSO)
    52.00€
  • Afamelanotide acetate

    CAS:
    <p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>
    Formula:C80H115N21O21
    Purity:98% - 99.494%
    Color and Shape:Solid
    Molecular weight:1706.9

    Ref: TM-T7589

    1mg
    73.00€
    5mg
    160.00€
    10mg
    230.00€
    25mg
    378.00€
    50mg
    565.00€
    100mg
    805.00€
  • PF-06882961 Tris

    CAS:
    PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C35H41FN6O7
    Purity:98.74% - 99.79%
    Color and Shape:Solid
    Molecular weight:676.7

    Ref: TM-T8876

    1mg
    131.00€
    5mg
    286.00€
    10mg
    430.00€
    25mg
    710.00€
    50mg
    998.00€
    100mg
    1,349.00€
    500mg
    2,688.00€
  • FAUC-365

    CAS:
    FAUC-365 is a D3 dopamine receptor agonist.
    Formula:C23H25Cl2N3OS
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:462.44

    Ref: TM-T21667

    1mg
    52.00€
    5mg
    111.00€
    10mg
    169.00€
    25mg
    323.00€
    50mg
    512.00€
    100mg
    740.00€
    500mg
    1,539.00€
    1mL*10mM (DMSO)
    123.00€
  • RTICBM-189

    CAS:
    RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.
    Formula:C15H14Cl2N2O
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:309.19

    Ref: TM-T9466

    2mg
    37.00€
    5mg
    50.00€
    10mg
    88.00€
    25mg
    170.00€
    50mg
    264.00€
    100mg
    389.00€
    200mg
    550.00€
    1mL*10mM (DMSO)
    71.00€
  • Melanotan (MT)-II

    CAS:
    Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
    Formula:C50H69N15O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1024.18

    Ref: TM-TP1324

    1mg
    35.00€
    2mg
    48.00€
    5mg
    70.00€
    10mg
    94.00€
    25mg
    160.00€
    50mg
    250.00€
    100mg
    406.00€
    200mg
    592.00€
  • Betazole dihydrochloride

    CAS:
    <p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>
    Formula:C5H11Cl2N3
    Purity:99.12%
    Color and Shape:Solid
    Molecular weight:184.067

    Ref: TM-T8599

    1mg
    35.00€
    5mg
    60.00€
    10mg
    96.00€
    25mg
    170.00€
    50mg
    306.00€
    100mg
    399.00€
    200mg
    568.00€
  • AC-90179 HCl

    CAS:
    AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.
    Formula:C23H31ClN2O2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:402.96

    Ref: TM-T26543

    1mg
    35.00€
    5mg
    64.00€
    10mg
    90.00€
    25mg
    134.00€
    50mg
    235.00€
    100mg
    349.00€
    1mL*10mM (DMSO)
    85.00€
  • Prasugrel Hydrochloride

    CAS:
    <p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>
    Formula:C20H20FNO3S·HCl
    Purity:99.39% - 99.79%
    Color and Shape:Solid
    Molecular weight:409.9

    Ref: TM-T6952

    1g
    183.00€
    50mg
    44.00€
    100mg
    57.00€
    500mg
    127.00€
  • Opiranserin hydrochloride

    CAS:
    Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM
    Formula:C21H35ClN2O5
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:430.97

    Ref: TM-T9833

    1mg
    96.00€
    5mg
    227.00€
    10mg
    359.00€
    25mg
    652.00€
    50mg
    929.00€
    100mg
    1,293.00€
    500mg
    2,593.00€
    1mL*10mM (DMSO)
    250.00€