
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(54 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5981 products of "GPCR/G-Protein"
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Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formula:C18H22ClNOPurity:99.44% - 99.85%Color and Shape:SolidMolecular weight:303.83Ref: TM-T7564
2mg35.00€5mg51.00€10mg81.00€25mg106.00€50mg147.00€100mg207.00€200mg306.00€1mL*10mM (DMSO)63.00€Tecalcet Free Base
CAS:Tecalcet Free Base is an oral calcium receptor agonistFormula:C18H22ClNOColor and Shape:SolidMolecular weight:303.83Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34Ref: TM-T2373
2mg35.00€5mg51.00€10mg80.00€25mg131.00€50mg210.00€100mg313.00€200mg445.00€1mL*10mM (DMSO)215.00€Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5Gadolinium chloride
CAS:Gadolinium chloride is a calcium-sensing receptor (CaSR) agonistFormula:Cl3GdPurity:98%Color and Shape:White Crystalline SolidMolecular weight:263.61Dexmedetomidine hydrochloride
CAS:Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C13H16N2·HClPurity:99.94% - 99.94%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:236.74Ref: TM-T6466
5mg42.00€10mg55.00€25mg88.00€50mg159.00€100mg226.00€200mg340.00€500mg563.00€1mL*10mM (DMSO)50.00€Vorapaxar sulfate
CAS:Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.Formula:C29H35FN2O8SPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:590.66Ref: TM-T3098
1mg38.00€2mg49.00€5mg79.00€10mg119.00€25mg210.00€50mg354.00€100mg528.00€500mg1,159.00€1mL*10mM (DMSO)99.00€AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formula:C17H21N5O2SPurity:99.81%Color and Shape:SolidMolecular weight:359.45Ref: TM-T5179
1mg39.00€2mg49.00€5mg81.00€10mg120.00€25mg236.00€50mg354.00€100mg510.00€1mL*10mM (DMSO)89.00€Zafirlukast
CAS:Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and anti-inflammatory effects. Cost-effective and quality-assured.Formula:C31H33N3O6SPurity:99% - 99.83%Color and Shape:SolidMolecular weight:575.68Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formula:C24H29ClN2O3Purity:99.5%Color and Shape:SolidMolecular weight:428.95Ref: TM-T9220
1mg44.00€5mg87.00€10mg117.00€25mg202.00€50mg304.00€100mg437.00€200mg612.00€1mL*10mM (DMSO)97.00€CPI-444
CAS:CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.Formula:C20H21N7O3Purity:98.78%Color and Shape:SolidMolecular weight:407.43Ref: TM-T7183
2mg34.00€5mg52.00€10mg73.00€25mg128.00€50mg197.00€100mg295.00€200mg442.00€1mL*10mM (DMSO)52.00€Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purity:98% - 99.494%Color and Shape:SolidMolecular weight:1706.9PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Formula:C23H25Cl2N3OSPurity:99.62%Color and Shape:SolidMolecular weight:462.44Ref: TM-T21667
1mg52.00€5mg111.00€10mg169.00€25mg323.00€50mg512.00€100mg740.00€500mg1,539.00€1mL*10mM (DMSO)123.00€RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Ref: TM-T9466
2mg37.00€5mg50.00€10mg88.00€25mg170.00€50mg264.00€100mg389.00€200mg550.00€1mL*10mM (DMSO)71.00€Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purity:>99.99%Color and Shape:SolidMolecular weight:1024.18Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purity:99.12%Color and Shape:SolidMolecular weight:184.067AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formula:C23H31ClN2O2Purity:99.71%Color and Shape:SolidMolecular weight:402.96Prasugrel Hydrochloride
CAS:<p>Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.</p>Formula:C20H20FNO3S·HClPurity:99.39% - 99.79%Color and Shape:SolidMolecular weight:409.9Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purity:99.33%Color and Shape:SolidMolecular weight:430.97Ref: TM-T9833
1mg96.00€5mg227.00€10mg359.00€25mg652.00€50mg929.00€100mg1,293.00€500mg2,593.00€1mL*10mM (DMSO)250.00€
