GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Detomidine hydrochloride
CAS:Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.Formula:C12H14N2·HClPurity:99.97%Color and Shape:SolidMolecular weight:222.71BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21%Color and Shape:SolidMolecular weight:372.89Tetracosactide acetate
CAS:Cosyntropin (acetate) stimulates the release of corticosteroids such as cortisol from the adrenal gland.Formula:C138H214N40O33SPurity:99.76%Color and Shape:SolidMolecular weight:2993.54Tofogliflozin (hydrate)
CAS:Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).Formula:C22H28O7Purity:97.03% - 98.78%Color and Shape:SolidMolecular weight:404.45Ref: TM-T5016
1mg35.00€2mg49.00€5mg74.00€10mg109.00€25mg202.00€50mg324.00€100mg505.00€200mg717.00€1mL*10mM (DMSO)82.00€Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purity:99.59% - 99.90%Color and Shape:White PowderMolecular weight:1371.53Ref: TM-T21410
5mg52.00€10mg78.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€1mL*10mM (DMSO)116.00€Myristicin
CAS:Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formula:C11H12O3Purity:99.828%Color and Shape:LiquidMolecular weight:192.21Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43AZ3451
CAS:AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).Formula:C30H27BrN4O3Purity:98.12%Color and Shape:SolidMolecular weight:571.46Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS:Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-Formula:C24H35ClO9Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:502.98Rolapitant hydrochloride hydrate
CAS:Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.Formula:C25H29ClF6N2O3Color and Shape:SolidMolecular weight:554.95Hydroxyzine dihydrochloride
CAS:Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formula:C21H27ClN2O2·2HClPurity:99.46% - 99.79%Color and Shape:Oil PowderMolecular weight:447.83Darbufelone mesylate
CAS:Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).Formula:C19H28N2O5S2Purity:96.81% - 99.92%Color and Shape:SolidMolecular weight:428.57Ref: TM-T10960L
1mg50.00€5mg99.00€10mg167.00€25mg340.00€50mg557.00€100mg790.00€200mg1,063.00€1mL*10mM (DMSO)109.00€Adenosine amine congener
CAS:Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.Formula:C28H32N8O6Purity:97.86%Color and Shape:SolidMolecular weight:576.6Prasugrel Hydrochloride
CAS:Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
Formula:C20H20FNO3S·HClPurity:99.39% - 99.79%Color and Shape:SolidMolecular weight:409.9GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:C51H65N9O10Purity:97.86%Color and Shape:SolidMolecular weight:964.12Ibutamoren
CAS:Ibutamoren (MK-677) is a drug which acts as a potent, orally active growth hormone secretagogue, mimicking the GH stimulating action of the endogenous hormone ghrelin. It also alters the metabolism of body fat and so may have an application in the treatment of obesity.Formula:C27H36N4O5SPurity:97.59%Color and Shape:SolidMolecular weight:528.66BPTU
CAS:BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).Formula:C23H22F3N3O3Purity:99.37% - 99.89%Color and Shape:SolidMolecular weight:445.43Ref: TM-T4132
1mg35.00€2mg50.00€5mg69.00€10mg110.00€25mg225.00€50mg389.00€100mg577.00€1mL*10mM (DMSO)69.00€Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852RS 100329
CAS:RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formula:C20H25F3N4O3Color and Shape:SolidMolecular weight:426.43Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purity:97.41%Color and Shape:SolidMolecular weight:244.38
