GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(58 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5982 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852RS 100329
CAS:RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).Formula:C20H25F3N4O3Color and Shape:SolidMolecular weight:426.43ARC-239
CAS:ARC-239 is an agonist of α2-adrenergic receptor.Formula:C24H29N3O3Color and Shape:SolidMolecular weight:407.51Siponimod
CAS:Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.Formula:C29H35F3N2O3Purity:99.13% - 99.8%Color and Shape:SolidMolecular weight:516.59Ganirelix Acetate
CAS:Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormula:C82H117ClN18O15Purity:96.05%Color and Shape:SolidMolecular weight:1630.4Tesmilifene fumarate
CAS:Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。Formula:C23H29NO5Purity:99.86%Color and Shape:SolidMolecular weight:399.48Ref: TM-T22746
5mg44.00€10mg60.00€25mg110.00€50mg164.00€100mg235.00€200mg349.00€1mL*10mM (DMSO)49.00€Neurotensin
CAS:Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.Formula:C78H121N21O20Purity:>99.99%Color and Shape:SolidMolecular weight:1672.92CCG-50014
CAS:CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.Formula:C16H13FN2O2SPurity:98.53%Color and Shape:SolidMolecular weight:316.35AnaMorelin hydrochloride
CAS:AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formula:C31H43ClN6O3Purity:99.18% - ≥98%Color and Shape:SolidMolecular weight:583.16Ref: TM-T7225
1mg35.00€2mg50.00€5mg73.00€10mg96.00€25mg145.00€50mg177.00€100mg235.00€1mL*10mM (DMSO)95.00€Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formula:C24H25FN4O2Purity:99.33%Color and Shape:SolidMolecular weight:420.48Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formula:C32H39NO2Purity:99.65% - 99.99%Color and Shape:White To Off-White PowderMolecular weight:469.66Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formula:C17H27Cl2NOPurity:99.72% - 99.91%Color and Shape:SolidMolecular weight:332.31Ref: TM-T7176
5mg50.00€10mg74.00€25mg124.00€50mg197.00€100mg311.00€200mg467.00€500mg747.00€1mL*10mM (DMSO)52.00€ELA-14(human) acetate
ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.Formula:C77H123N25O19S2Purity:97.2%Color and Shape:SolidMolecular weight:1767.09Dapiprazole Hydrochloride
CAS:Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.Formula:C19H28ClN5Purity:99.75% - 99.93%Color and Shape:SolidMolecular weight:361.92Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66Taminadenant
CAS:Taminadenant is an adenosine receptor antagonist.Formula:C10H8BrN7Purity:99.11%Color and Shape:SolidMolecular weight:306.12Ref: TM-T16980
2mg35.00€5mg51.00€10mg88.00€25mg120.00€50mg170.00€100mg250.00€200mg373.00€1mL*10mM (DMSO)57.00€Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Ref: TM-TQ0227
1mg52.00€5mg111.00€10mg180.00€25mg243.00€50mg305.00€100mg424.00€1mL*10mM (DMSO)113.00€Pimavanserin
CAS:Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.Formula:C25H34FN3O2Purity:97.84% - 99.69%Color and Shape:Pale Yellow To Pale Orange SolidMolecular weight:427.55β-MSH (1-22) (human) acetate
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) , is an endogenous melanocortin-4 receptor (MC4-R) agonist.Formula:C120H178N34O37SPurity:99.64%Color and Shape:SolidMolecular weight:2720.97Rimegepant
CAS:View and buy Rimegepant from TargetMol.BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.Cited in 1 publications.Formula:C28H28F2N6O3Purity:99.1% - 99.99%Color and Shape:SolidMolecular weight:534.56
