GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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ML-18
CAS:ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.Formula:C32H35N5O5Purity:98.62% - >99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-T4540
1mg34.00€5mg60.00€10mg96.00€25mg170.00€50mg264.00€100mg425.00€200mg587.00€1mL*10mM (DMSO)75.00€AdipoRon hydrochloride
CAS:AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).Formula:C27H29ClN2O3Color and Shape:SolidMolecular weight:464.99Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Formula:C20H24N2OSColor and Shape:SolidMolecular weight:340.48Apraclonidine
CAS:Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.Formula:C9H10Cl2N4Color and Shape:SolidMolecular weight:245.11Napitane Mesylate
CAS:Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.Formula:C23H29NO5SPurity:98%Color and Shape:SolidMolecular weight:431.55Xamoterol
CAS:Xamoterol is a cardiac stimulant.Formula:C16H25N3O5Color and Shape:SolidMolecular weight:339.39Tiapride
CAS:Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.Formula:C15H24N2O4SColor and Shape:SolidMolecular weight:328.43Melitracen hydrochloride
CAS:Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.Formula:C21H26ClNPurity:99.99%Color and Shape:Crystalline SolidMolecular weight:327.90Ref: TM-T4274
10mg44.00€25mg64.00€50mg93.00€100mg110.00€200mg161.00€500mg264.00€1mL*10mM (DMSO)48.00€Ajmalicine hydrochloride
CAS:Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.Formula:C21H25ClN2O3Color and Shape:SolidMolecular weight:388.89THIQ
CAS:THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).Formula:C33H41ClN6O2Purity:98.93%Color and Shape:SolidMolecular weight:589.17Guanabenz hydrochloride
CAS:Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.Formula:C8H9Cl3N4Purity:99.45%Color and Shape:SolidMolecular weight:267.54Siponimod
CAS:Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; >1000x selectivity over S1P2-4.Formula:C29H35F3N2O3Purity:99.13% - 99.8%Color and Shape:SolidMolecular weight:516.59Secretin (33-59), rat
CAS:Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35Dolasetron
CAS:Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.Formula:C19H20N2O3Purity:99.84% - 99.86%Color and Shape:White PowderMolecular weight:324.37Netupitant
CAS:Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).Formula:C30H32F6N4OPurity:99.43%Color and Shape:SolidMolecular weight:578.59RG7713
CAS:RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.Formula:C25H28ClN3O2Purity:99.74%Color and Shape:SolidMolecular weight:437.96AnaMorelin hydrochloride
CAS:AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).Formula:C31H43ClN6O3Purity:99.18% - ≥98%Color and Shape:SolidMolecular weight:583.16Ref: TM-T7225
1mg35.00€2mg50.00€5mg73.00€10mg96.00€25mg145.00€50mg177.00€100mg235.00€1mL*10mM (DMSO)95.00€1-Ethyl-6-aminouracil
CAS:1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have highFormula:C6H9N3O2Purity:99.29%Color and Shape:SolidMolecular weight:155.15RS-127445
CAS:RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.
Formula:C17H16FN3Purity:99.32%Color and Shape:SolidMolecular weight:281.33Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Formula:C24H25FN4O2Purity:99.33%Color and Shape:SolidMolecular weight:420.48
