GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5960 products of "GPCR/G-Protein"
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Histrelin acetate
CAS:Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Piperoxan hydrochloride
CAS:Piperoxan hydrochloride (Benodaine hydrochloride) is an α2 adrenoceptor antagonist.Formula:C14H20ClNO2Purity:99.61%Color and Shape:SolidMolecular weight:269.77Ref: TM-T4526
2mg39.00€5mg62.00€10mg92.00€25mg128.00€50mg166.00€100mg200.00€200mg299.00€1mL*10mM (DMSO)55.00€Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formula:C22H26N2O4Purity:98% - 99.9%Color and Shape:SolidMolecular weight:382.45Ref: TM-T6S0654
1mg62.00€2mg89.00€5mg132.00€10mg226.00€25mg384.00€50mg557.00€100mg785.00€200mg1,054.00€1mL*10mM (DMSO)146.00€CAY10526
CAS:CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formula:C12H7BrO3SPurity:98.75%Color and Shape:SolidMolecular weight:311.15TG4-155
CAS:TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.
Formula:C23H26N2O4Purity:97.2%Color and Shape:SolidMolecular weight:394.46Neuropeptide S (Rat) acetate
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.Formula:C97H164N34O29Purity:95.36%Color and Shape:SolidMolecular weight:2270.59Ref: TM-TP1982L
1mg87.00€2mg124.00€5mg192.00€10mg284.00€25mg452.00€50mg645.00€100mg867.00€200mg1,159.00€BRL-15572 dihydrochloride
CAS:BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formula:C25H27ClN2O·2HClPurity:99.74%Color and Shape:SolidMolecular weight:479.87Clemizole hydrochloride
CAS:Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3CCG215022
CAS:CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formula:C26H22FN7O3Purity:97.63% - 99.69%Color and Shape:SolidMolecular weight:499.5Ref: TM-T3498
1mg56.00€5mg114.00€10mg178.00€25mg394.00€50mg655.00€100mg1,035.00€1mL*10mM (DMSO)127.00€Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Lanreotide acetate
CAS:Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndromeFormula:C56H73N11O12S2Purity:>99.99%Color and Shape:SolidMolecular weight:1156.39Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41BD1063 dhydrochloride
CAS:BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).Formula:C13H20Cl4N2Purity:99.52% - ≥95%Color and Shape:SolidMolecular weight:346.12Ref: TM-T7488
2mg46.00€5mg69.00€10mg95.00€25mg177.00€50mg321.00€100mg472.00€200mg665.00€500mg1,018.00€Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71Taladegib
CAS:Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.Formula:C26H24F4N6OPurity:98.75% - >99.99%Color and Shape:SolidMolecular weight:512.5C-021
CAS:C 021 dihydrochloride is a potent CCR4 antagonist.Formula:C27H41N5O2Purity:99.74% - 99.90%Color and Shape:SolidMolecular weight:467.65Ref: TM-T21870
1mg49.00€2mg67.00€5mg90.00€10mg144.00€25mg286.00€50mg444.00€100mg622.00€1mL*10mM (DMSO)90.00€Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormula:C43H77N17O12S2Purity:99.79%Color and Shape:SolidMolecular weight:1088.32Phenylephrine
CAS:Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formula:C11H9Cl2N3O3SPurity:99.80% - >99.99%Color and Shape:SolidMolecular weight:334.18Ref: TM-T4300
1mg34.00€5mg66.00€10mg105.00€25mg217.00€50mg334.00€100mg502.00€500mg1,063.00€1mL*10mM (DMSO)73.00€Canagliflozin
CAS:Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.Formula:C24H25FO5SPurity:98.01% - >99.99%Color and Shape:SolidMolecular weight:444.52Ref: TM-T1782
2mg35.00€5mg50.00€10mg66.00€25mg87.00€50mg96.00€100mg123.00€500mg274.00€1mL*10mM (DMSO)52.00€
