GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5959 products of "GPCR/G-Protein"
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Avexitide
CAS:Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formula:C149H234N40O47SPurity:98% - 99.65%Color and Shape:SolidMolecular weight:3369.76BD1063 dhydrochloride
CAS:BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).Formula:C13H20Cl4N2Purity:99.52% - ≥95%Color and Shape:SolidMolecular weight:346.12Ref: TM-T7488
2mg46.00€5mg69.00€10mg95.00€25mg177.00€50mg321.00€100mg472.00€200mg665.00€500mg1,018.00€Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormula:C43H77N17O12S2Purity:99.79%Color and Shape:SolidMolecular weight:1088.32HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formula:C35H51N9O14Purity:>99.99%Color and Shape:SolidMolecular weight:821.84Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formula:C13H16ClN3O3Purity:98.15%Color and Shape:SolidMolecular weight:297.74Ref: TM-T9193
1mg50.00€5mg110.00€10mg172.00€25mg304.00€50mg424.00€100mg583.00€200mg785.00€1mL*10mM (DMSO)122.00€Betaxolol
CAS:Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Formula:C52H77N15O13Purity:>99.99%Color and Shape:SolidMolecular weight:1120.26Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurity:99.78% - >99.99%Color and Shape:SolidMolecular weight:463.871-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.
Formula:C9H15N3OPurity:95%Color and Shape:SolidMolecular weight:181.23VKGILS-NH2 Acetate
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor 2 (PAR2) agonist.Formula:C30H58N8O9Purity:98.83%Color and Shape:SolidMolecular weight:674.83Ref: TM-T21699L
1mg33.00€2mg49.00€5mg62.00€10mg92.00€25mg155.00€50mg224.00€100mg331.00€200mg470.00€1mL*10mM (DMSO)92.00€DORA-22
CAS:DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormula:C23H22F2N4O2Purity:97.67%Color and Shape:SolidMolecular weight:424.44Ref: TM-T5500
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)331.00€Diquafosol tetrasodium
CAS:Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormula:C18H22N4Na4O23P4Purity:98.25% - 99.97%Color and Shape:SolidMolecular weight:878.23Velneperit
CAS:Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.Formula:C17H24F3N3O3SPurity:99.70%Color and Shape:SolidMolecular weight:407.45Ref: TM-T17222
1mg34.00€2mg49.00€5mg74.00€10mg113.00€25mg245.00€50mg416.00€100mg613.00€1mL*10mM (DMSO)82.00€Elinzanetant
CAS:Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
Formula:C33H35F7N4O3Purity:98% - 99.13%Color and Shape:SolidMolecular weight:668.64Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85Carazolol
CAS:Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formula:C18H22N2O2Purity:99% - 99.53%Color and Shape:Yellowish SolidMolecular weight:298.38RS-67333
CAS:RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Formula:C19H29ClN2O2Purity:99.24%Color and Shape:SolidMolecular weight:352.9
![1-[(5-methylisoxazol-3-yl)methyl]piperazine](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT8582.webp&w=3840&q=75)
