GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5971 products of "GPCR/G-Protein"
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Bucindolol
CAS:Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.Formula:C22H25N3O2Purity:99.9%Color and Shape:SolidMolecular weight:363.45BMS-986278
CAS:BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,
Formula:C22H31N5O5Purity:99.86%Color and Shape:SolidMolecular weight:445.51GRK6-IN-2
CAS:GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.
Formula:C21H21FN6Purity:98.94%Color and Shape:SolidMolecular weight:376.435-LOX inhibitor
CAS:5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) is an itraconazole impurity, a LOX-5 inhibitor.Formula:C22H27N5O2Purity:98.01%Color and Shape:SolidMolecular weight:393.48Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS:(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H14D5Cl2N3SColor and Shape:SolidMolecular weight:289.28Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formula:C21H21D8Cl3N2O2Color and Shape:SolidMolecular weight:455.88SR59230A hydrochloride
CAS:SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formula:C21H28ClNO2Purity:99.49%Color and Shape:SolidMolecular weight:361.91Ropinirole
CAS:Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formula:C16H24N2OPurity:99.68%Color and Shape:SolidMolecular weight:260.38L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formula:C18H19ClN4Purity:98%Color and Shape:SolidMolecular weight:326.82R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formula:C27H26FN3OSPurity:98.55%Color and Shape:SolidMolecular weight:459.58Ref: TM-T16709
1mg35.00€5mg74.00€10mg119.00€25mg269.00€50mg447.00€100mg733.00€200mg973.00€1mL*10mM (DMSO)75.00€PACAP (1-38), human, ovine, rat
CAS:PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formula:C203H331N63O53SPurity:96.93% - 98.16%Color and Shape:SolidMolecular weight:4534.26Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formula:C21H21N·HClPurity:99.88% - 99.97%Color and Shape:SolidMolecular weight:323.86Travoprost
CAS:Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formula:C26H35F3O6Purity:97.39% - 99.58%Color and Shape:Colorless OilMolecular weight:500.55Ref: TM-T5841
1mg46.00€5mg88.00€10mg120.00€25mg175.00€50mg255.00€100mg371.00€200mg507.00€1mL*10mM (DMSO)96.00€Triflupromazine
CAS:Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formula:C18H19F3N2SColor and Shape:SolidMolecular weight:352.42Blontuvetmab
CAS:Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].Color and Shape:LiquidN-Methyl amisulpride
CAS:N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formula:C18H29N3O4SColor and Shape:SolidMolecular weight:383.51Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurity:98%Color and Shape:SolidMolecular weight:506.59Meticillin
CAS:Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.Formula:C17H20N2O6SColor and Shape:SolidMolecular weight:380.42Rocatinlimab
CAS:Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Color and Shape:Liquid
