CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5963 products of "GPCR/G-Protein"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • OXA(17-33)

    CAS:
    Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.
    Formula:C79H125N23O22
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1749

    Ref: TM-TP1973

    1mg
    1,423.00€
  • PAMP-12(human, porcine)

    CAS:
    Potent endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 57.2 nM). Corresponds to amino acids 9 to 20 of proadrenomedullin.
    Formula:C77H119N25O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1618.95

    Ref: TM-TP1880

    1mg
    605.00€
  • Crustacean Cardioactive Peptide (CCAP)

    CAS:
    Crustacean Cardioactive Peptide (CCAP) is a conserved modified cyclic nonapeptide primary structure of PFCNAFTGC-NH2, a disulfide bridge between Cys3 and Cys9.
    Formula:C42H58N10O12S2
    Purity:95.40%
    Color and Shape:Solid
    Molecular weight:959.1

    Ref: TM-TP1413

    1mg
    49.00€
    5mg
    99.00€
    10mg
    153.00€
    25mg
    246.00€
    50mg
    370.00€
    100mg
    534.00€
    200mg
    760.00€
  • Isoprenaline

    CAS:
    Isoprenaline is a non-selective and orally active β-adrenoceptor agonist.Isoproterenol is a potent peripheral vasodilator and bronchodilator.
    Formula:C11H17NO3
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:211.26

    Ref: TM-T21411

    10mg
    56.00€
    25mg
    97.00€
    50mg
    163.00€
    100mg
    255.00€
  • Losulazine

    CAS:

    Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.

    Formula:C27H22F4N4O3S
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:558.55

    Ref: TM-T68095

    1mg
    43.00€
    5mg
    96.00€
    10mg
    128.00€
    25mg
    234.00€
    50mg
    311.00€
    100mg
    454.00€
    200mg
    648.00€
  • CCR6 inhibitor 1

    CAS:

    CCR6 inhibitor 1 selectively blocks CCR6 (0.45 nM in monkeys, 6 nM in humans), aiding in vitro/vivo disease studies.

    Formula:C24H23F3N4O3S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:504.52

    Ref: TM-T10715

    1mg
    116.00€
    5mg
    283.00€
    10mg
    424.00€
    25mg
    682.00€
    50mg
    934.00€
    100mg
    1,301.00€
    500mg
    2,612.00€
  • LY-426965 hydrochloride

    CAS:
    LY-426965 hydrochloride is a bioactive chemical.
    Formula:C28H39ClN2O2
    Color and Shape:Solid
    Molecular weight:471.07

    Ref: TM-T33017

    25mg
    1,369.00€
  • Cenicriviroc Mesylate

    CAS:
    Cenicriviroc Mesylate (TBR-652 Mesylate) is an oral dual CCR2/CCR5 antagonist exhibiting anti-inflammatory and anti-fibrotic effects for liver fibrosis.
    Formula:C42H56N4O7S2
    Purity:98.819%
    Color and Shape:Solid
    Molecular weight:793.05

    Ref: TM-T10756

    1mg
    80.00€
    5mg
    127.00€
    10mg
    202.00€
    25mg
    406.00€
    50mg
    692.00€
    100mg
    924.00€
    1mL*10mM (DMSO)
    177.00€
  • γ-2-MSH (41-58), amide

    CAS:
    Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.
    Formula:C74H100N22O15S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1569.79

    Ref: TM-TP1532

    100mg
    To inquire
    500mg
    To inquire
  • T-10430


    T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.
    Formula:C17H22N6O
    Color and Shape:Solid
    Molecular weight:326.396

    Ref: TM-T204318

    10mg
    To inquire
    50mg
    To inquire
  • Danshenol B


    Danshenol B is a natural product that can be used as a reference standard.
    Formula:C22H26O4
    Color and Shape:Solid
    Molecular weight:354.446

    Ref: TM-T125490

    1mg
    To inquire
    5mg
    To inquire
  • Sulamserod

    CAS:
    Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related
    Formula:C19H28ClN3O5S
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:445.96

    Ref: TM-T13021

    1mg
    517.00€
    5mg
    1,130.00€
  • AL 34662

    CAS:
    AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a
    Formula:C10H13N3O
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:191.23

    Ref: TM-T22029

    1mg
    42.00€
    5mg
    88.00€
    10mg
    127.00€
    25mg
    216.00€
  • MLN-3897 TFA


    MLN-3897 TFA is a potent CCR1 antagonist that inhibits the binding of 125I-MIP-1α to THP-1 cell membranes.
    Formula:C32H32ClF3N2O6
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:633.05

    Ref: TM-T28072L

    1mg
    115.00€
    5mg
    245.00€
    10mg
    363.00€
    25mg
    562.00€
    50mg
    775.00€
    100mg
    1,035.00€
    200mg
    1,406.00€
    1mL*10mM (DMSO)
    To inquire
  • L803

    CAS:
    L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.
    Formula:C50H80N13O19P
    Color and Shape:Solid
    Molecular weight:1198.22

    Ref: TM-TP3907

    10mg
    To inquire
    50mg
    To inquire
  • CTP-amiodarone


    CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.
    Formula:C97H131F3I2N20O25S2
    Color and Shape:Solid
    Molecular weight:2352.13

    Ref: TM-TP2921

    10mg
    To inquire
    50mg
    To inquire
  • PF-9184

    CAS:
    PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.
    Formula:C21H14Cl2N2O4S
    Purity:97.43%
    Color and Shape:Solid
    Molecular weight:461.32

    Ref: TM-T21738

    1mg
    34.00€
    5mg
    72.00€
    10mg
    98.00€
    25mg
    To inquire
    50mg
    To inquire
  • 15-keto-17-phenyl trinor Prostaglandin F2α

    CAS:
    Bimatoprost is an F-series prostaglandin (PG) analog which has been approved for use as an ocular hypotensive drug.
    Formula:C23H30O5
    Color and Shape:Solid
    Molecular weight:386.488

    Ref: TM-T37934

    1mg
    220.00€
    5mg
    944.00€
    10mg
    1,700.00€
  • [Gln8]-C517 (LH-RH), chicken

    CAS:
    [Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.
    Formula:C54H71N15O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1154.23

    Ref: TM-TP1648

    100mg
    To inquire
    500mg
    To inquire
  • SDV-Exendin-3/4


    SDV-Exendin-3/4 is a 32-amino acid peptide.
    Formula:NA
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3443.87

    Ref: TM-TP1461

    1mg
    329.00€
    5mg
    1,044.00€