GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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Substance P(1-7) TFA
CAS:Substance P(1-7) TFA is a fragment of neuropeptide P (SP), with anti-harmful effects, used in neurological disease research.Formula:C43H66F3N13O12Purity:98.23%Color and Shape:SolidMolecular weight:1014.061-(2-Methoxyphenyl)piperazine hydrochloride
CAS:Compound PDK0265, with CAS No. 5464-78-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0265 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C11H16N2OMolecular weight:192.253-Deoxyglucosone
CAS:3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with proteinFormula:C6H10O5Purity:95%Color and Shape:SolidMolecular weight:162.14Xenin-8
CAS:neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effectsFormula:C51H79N15O9Purity:98%Color and Shape:SolidMolecular weight:1046.27γ3-MSH
CAS:γ3-MSH, originating from the N-terminal segment of pro-opiomelanocortin (POMC), induces aldosterone secretion in cultured human adrenal tumor cells [1].Formula:C126H188N44O37SColor and Shape:SolidMolecular weight:2943.18Onzigolide
CAS:Onzigolide (BIM-23A760) is a dual agonist for D2R and SSTR2 with strong dopamine and somatostatin properties.Formula:C86H116N16O12S4Color and Shape:SolidMolecular weight:1694.21Femoxetine
CAS:Femoxetine: antidepressant, enhances morphine, inhibits MAO-A/B, boosts mice's exercise capacity.Formula:C20H25NO2Purity:99.1% - 99.35%Color and Shape:SolidMolecular weight:311.42Triamterene
CAS:Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formula:C12H11N7Purity:99.77%Color and Shape:Yellow Yellow SolidMolecular weight:253.26CCR6 antagonist 1
CAS:CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.
Formula:C17H12F3NO2Purity:99.83%Color and Shape:SoildMolecular weight:319.28CUR61414 hydrochloride
CUR61414 hydrochloride: potent cell-permeable Hedgehog pathway inhibitor, IC50=100-200 nM, selectively targets Smo (Ki=44 nM), induces cancer cell apoptosis.Formula:C31H43ClN4O5Purity:94.05%Color and Shape:SolidMolecular weight:587.15Cisapride hydrate
CAS:Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.Formula:C23H31ClFN3O5Purity:98%Color and Shape:SolidMolecular weight:483.96Oxatomide
CAS:Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).Formula:C27H30N4OPurity:99.28% - 99.72%Color and Shape:White PowderMolecular weight:426.55Ref: TM-T19839
1mg35.00€5mg75.00€10mg114.00€25mg222.00€50mg356.00€100mg557.00€500mg1,153.00€1mL*10mM (DMSO)84.00€Cortistatin-14
CAS:Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Formula:C81H114N20O18S2Purity:98.06% - 98.23%Color and Shape:SolidMolecular weight:1720.03Hemopressin(human, mouse) TFA
CAS:Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.Formula:C52H80F3N13O14Purity:98%Color and Shape:SolidMolecular weight:1168.27IRL-1038 TFA
IRL-1038 TFA is an ETB receptor antagonist used in the study of cardiovascular disease.Formula:C70H93F3N14O17S2Purity:98.79%Color and Shape:SolidMolecular weight:1523.7N-Desmethyl Pimavanserin
CAS:N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.Formula:C24H32FN3O2Purity:98.02%Color and Shape:SolidMolecular weight:413.53Tabernanthalog
CAS:TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.Formula:C14H18N2OPurity:99.82% - 99.89%Color and Shape:SoildMolecular weight:230.31Ref: TM-T60221
1mg175.00€2mg264.00€5mg404.00€10mg592.00€25mg888.00€50mg1,243.00€100mg1,701.00€500mg3,402.00€1mL*10mM (DMSO)344.00€BMS-193885
CAS:BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.Formula:C33H42N4O6Purity:99.73%Color and Shape:SolidMolecular weight:590.71GV-150013X
CAS:GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKiFormula:C33H34N4O3Purity:99.94%Color and Shape:SoildMolecular weight:534.65Ref: TM-T27503L
1mg90.00€5mg190.00€10mg259.00€25mg394.00€50mg532.00€100mg698.00€200mg924.00€1mL*10mM (DMSO)270.00€Boc-Phe-Leu-Phe-Leu-Phe
CAS:Boc-Phe-Leu-Phe-Leu-Phe is a chemotactic peptide antagonist that inhibits the release of peptide leukotrienes induced by FMLP.Formula:C44H59N5O8Color and Shape:SolidMolecular weight:785.97
