GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5958 products of "GPCR/G-Protein"
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Tamsolusin Hydrochloride
CAS:Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.Formula:C20H29ClN2O5SPurity:99.92%Color and Shape:SoildMolecular weight:444.97Brombuterol hydrochloride
CAS:Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formula:C12H19Br2ClN2OColor and Shape:SolidMolecular weight:402.56Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formula:C19H24Cl2N2Color and Shape:SolidMolecular weight:354.33Canagliflozin (Standard)
CAS:Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).Formula:C24H25FO5SColor and Shape:SolidMolecular weight:444.52Apraclonidine hydrochloride
CAS:Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.Formula:C9H11Cl3N4Purity:99.74%Color and Shape:SolidMolecular weight:281.57Doxazosin D8
CAS:Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Formula:C23H25N5O5Purity:98%Color and Shape:SolidMolecular weight:459.52Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63Rebamipide-d4
CAS:Rebamipide D4 is deuterium labeled Rebamipide.Formula:C19H15ClN2O4Purity:98%Color and Shape:SolidMolecular weight:374.81Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63Ceralifimod
CAS:Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).Formula:C27H33NO4Color and Shape:SolidMolecular weight:435.56NBI-27914
CAS:NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.Formula:C18H20Cl4N4Purity:99.47% - 99.64%Color and Shape:SolidMolecular weight:434.19Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purity:98%Color and Shape:White PowderMolecular weight:1084.23SB-277011 hydrochloride
CAS:SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.Formula:C28H31ClN4OPurity:98.54%Color and Shape:SolidMolecular weight:475.03V-0219
CAS:V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Formula:C20H25F3N4O2Purity:99.91%Color and Shape:SoildMolecular weight:410.43Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formula:C18H18ClN3SPurity:99.93%Color and Shape:SolidMolecular weight:343.87Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H18ClN3SPurity:98%Color and Shape:White Crystalline PowderMolecular weight:247.79Furprofen
CAS:Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Formula:C14H12O4Purity:98.62% - 99.25%Color and Shape:SolidMolecular weight:244.24L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Formula:C27H22BrNO4SPurity:98.97%Color and Shape:SolidMolecular weight:536.44Clozapine-d8
CAS:Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.Formula:C18H19ClN4Color and Shape:SolidMolecular weight:334.87Virodhamine
CAS:Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formula:C22H37NO2Purity:98%Color and Shape:SoildMolecular weight:347.53
