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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5981 products of "GPCR/G-Protein"

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  • Tixanox sodium

    CAS:
    Tixanox sodium effectively blocks histamine release in the lungs triggered by anti-IgE. It has also been demonstrated that when administered orally, Tixanox sodium can successfully counteract exercise-induced asthma.
    Formula:C15H9NaO5S
    Color and Shape:Solid
    Molecular weight:324.28

    Ref: TM-T201247

    25mg
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    50mg
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    100mg
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  • Substituted piperidines-1

    CAS:
    Substituted piperidines-1 can promote the release of growth hormone in humans and animals.
    Formula:C29H39N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:517.67

    Ref: TM-T19567

    25mg
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    50mg
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    100mg
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  • CS-0777

    CAS:
    CS-0777 is a potent, selective, and orally active S1P1 agonist (sphingosine 1-phosphate receptor modulator).
    Formula:C21H31N2O5P
    Color and Shape:Solid
    Molecular weight:422.45

    Ref: TM-T31107

    25mg
    3,155.00€
    50mg
    4,161.00€
    100mg
    5,795.00€
  • MRS4865

    CAS:
    MRS4865 (compound 7a) serves as a chimeric antagonist for the P2Y14 receptor and an agonist for UDP-glucose, offering protection against neuropathic pain.
    Formula:C39H39F3N4O7
    Color and Shape:Solid
    Molecular weight:732.74

    Ref: TM-T200587

    25mg
    2,186.00€
    50mg
    2,950.00€
    100mg
    3,852.00€
  • Beloxepin

    CAS:
    Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.
    Formula:C19H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T26765

    25mg
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    50mg
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    100mg
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  • RU 52583

    CAS:
    RU 52583 is an alpha 2-adrenergic receptor antagonist.
    Formula:C18H20N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.36

    Ref: TM-T26155

    25mg
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  • AMG-369

    CAS:
    AMG-369 (AMG 247) is an S1P1/S1P5 dual agonist that delays the development of experimental autoimmune encephalomyelitis in rats.
    Formula:C26H22FN3O2S
    Purity:98.04% - 98.92%
    Color and Shape:Solid
    Molecular weight:459.54

    Ref: TM-T29971

    1mg
    393.00€
    5mg
    930.00€
    10mg
    1,254.00€
    25mg
    1,863.00€
  • TM38837

    CAS:
    <p>CB1 antagonist 4 is an inverse agonist of cannabinoid receptor 1 (CB1) with an IC50 of 0.4 nM. It can reduce body weight, improve plasma inflammatory markers, and enhance glucose homeostasis [1].</p>
    Formula:C27H20Cl2F3N7O
    Color and Shape:Solid
    Molecular weight:586.40

    Ref: TM-T86011

    10mg
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    50mg
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  • NBI 35965 hydrochloride

    CAS:
    NBI 35965 hydrochloride is a selective CRF1 (corticotropin-releasing factor receptor 1) antagonist that is both orally active and capable of penetrating the brain. It possesses a K i value of 4 nM and a pK i of 8.5, and does not affect CRF2. This compound effectively diminishes CRF or stress-triggered ACTH (adrenocorticotropic hormone) production in vivo, demonstrating pIC 50 values of 7.1 and 6.9. Additionally, NBI 35965 hydrochloride exhibits anxiolytic properties [1] [2].
    Formula:C21H23Cl3N4
    Color and Shape:Solid
    Molecular weight:437.79

    Ref: TM-T86978

    10mg
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    50mg
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  • SSTR5 antagonist 6

    CAS:
    SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].
    Formula:C22H28ClN3O4
    Color and Shape:Solid
    Molecular weight:433.93

    Ref: TM-T87442

    10mg
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    50mg
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  • PF-9404C

    CAS:
    PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.
    Formula:C16H25N3O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.38

    Ref: TM-T28391

    25mg
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  • Tebideutorexant

    CAS:
    Tebideutorexant, an orexin-1 receptor antagonist, shows anti-panic effects in rodents and humans, providing a tool for stress response and psychiatric research.
    Formula:C23H16D2F4N4O2
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:460.42

    Ref: TM-T70332

    1mg
    232.00€
    5mg
    503.00€
    10mg
    755.00€
    25mg
    1,286.00€
    50mg
    1,863.00€
    100mg
    2,793.00€
  • A1AR antagonist 1


    Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).
    Formula:C18H14N4O
    Color and Shape:Solid
    Molecular weight:302.33

    Ref: TM-T60687

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Taranabant

    CAS:
    Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.
    Formula:C27H25ClF3N3O2
    Purity:99.06% - 99.06%
    Color and Shape:Solid
    Molecular weight:515.96

    Ref: TM-T13080L

    1mg
    98.00€
  • Terguride

    CAS:
    Terguride: treats hyperprolactinemia, blocks 5-HT2A/B, activates dopamine receptors, studied for PAH.
    Formula:C20H28N4O
    Color and Shape:Solid
    Molecular weight:340.46

    Ref: TM-T71847

    25mg
    5,576.00€
    50mg
    7,392.00€
    100mg
    10,640.00€
  • SphK1-IN-1


    SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.
    Formula:C22H22N6O2
    Color and Shape:Solid
    Molecular weight:402.45

    Ref: TM-T61965

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Setomagpran

    CAS:
    Setomagpran is an antagonist of the mas-related G protein-coupled receptor (MRGPR) and possesses anti-inflammatory properties.
    Formula:C22H19Cl2F6N5O
    Color and Shape:Solid
    Molecular weight:554.316

    Ref: TM-T206418

    10mg
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    50mg
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  • LX2761

    CAS:
    LX2761 is a stable inhibitor for SGLT1/2 with IC50s of 2.2/2.7 nM; it targets SGLT1 in the GI tract.
    Formula:C32H47N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:601.80

    Ref: TM-T15797

    25mg
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    100mg
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  • H3R antagonist 2


    Compound 23: H3R antagonist with 170 nM Ki; inhibits AChE, BChE, hMAO B; IC50s: 180, 880, 775 nM; anti-pain, memory boost; crosses BBB. [1]
    Formula:C24H29NO3
    Color and Shape:Solid
    Molecular weight:379.49

    Ref: TM-T61603

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • GLP-1 receptor agonist 16

    CAS:
    GLP-1 receptoragonist 16 (Example 53) is a GLP-1 agonist applicable for research in diabetes, obesity, or diseases related to non-alcoholic steatohepatitis.
    Formula:C33H31ClFN3O4
    Color and Shape:Solid
    Molecular weight:588.068

    Ref: TM-T204526

    10mg
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    50mg
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  • DSP-1053 benzenesulfonate

    CAS:
    DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.
    Formula:C32H38BrNO7S
    Color and Shape:Solid
    Molecular weight:660.62

    Ref: TM-T72220

    25mg
    2,300.00€
    50mg
    3,022.00€
    100mg
    4,085.00€
  • Rocavorexant

    CAS:
    Rocavorexant is an antagonist of the orexin-1 receptor (orexin-1 receptor), exhibiting a pIC50 value of 9.1 for human OX1 and a pIC50 of 6.0 for human OX2.
    Formula:C18H19F3N8O
    Color and Shape:Solid
    Molecular weight:420.392

    Ref: TM-T206374

    10mg
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    50mg
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  • BIIE-0246 HCl

    CAS:
    BIIE-0246: A potent, non-peptide Y2 receptor antagonist; >650-fold more selective than Y1, Y4, Y5.
    Formula:C49H59Cl2N11O6
    Color and Shape:Solid
    Molecular weight:968.97

    Ref: TM-T69621

    1mg
    720.00€
    10mg
    1,510.00€
  • BAY-3153

    CAS:
    BAY-3153 is a selective CCR1 ( C-C motif chemokine receptor 1 ) antagonist (human IC 50 =3 nM ; rat IC 50 =11 nM ; mice IC 50 =81 nM) .
    Formula:C25H29Cl2N3O4
    Color and Shape:Solid
    Molecular weight:506.42

    Ref: TM-T73371

    1mg
    517.00€
    5mg
    1,130.00€
    10mg
    1,549.00€
    25mg
    2,300.00€
    50mg
    3,022.00€
  • L-97-1

    CAS:
    L-97-1 is an antagonist of the adenosine A1 receptor.
    Formula:C29H38N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.65

    Ref: TM-T24384

    25mg
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    50mg
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    100mg
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  • MRGPRX1 agonist 4


    Potent, oral MRGPRX1 agonist 4 modulates receptor positively (EC50: 0.1 μM) and reduces mice's thermal allergy response.
    Formula:C23H17Cl2F3N2O2S
    Color and Shape:Solid
    Molecular weight:513.36

    Ref: TM-T63549

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Nipradolol

    CAS:
    Nipradolol blocks alpha-1-adrenergic receptors, lowers IOP in rabbits, and reduces NA-induced muscle contraction and dog artery vasodilation.
    Formula:C15H22N2O6
    Color and Shape:Solid
    Molecular weight:326.35

    Ref: TM-T73083

    25mg
    2,300.00€
    50mg
    3,022.00€
    100mg
    4,085.00€
  • CBR Agonist-1


    CBR Agonist-1 targets CB1R and CB2R with Ki of 0.18 μM and 1.22 μM, useful for studying cannabinoid-related diseases.
    Formula:C27H27FN4O
    Color and Shape:Solid
    Molecular weight:442.53

    Ref: TM-T62583

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • SSTR4 agonist 4

    CAS:
    SSTR4 agonist 4, potent in pain research, shows promise in rodent pain models, with potential for Alzheimer's due to hippocampus activity.
    Formula:C19H26N4O
    Color and Shape:Solid
    Molecular weight:326.44

    Ref: TM-T60911

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Dopamine D3 receptor ligand-1


    Dopamine D 3 receptor ligand is a potent, selective, high-affinity dopamine D3 receptor ligand that is 89 times more selective for D3 (Ki: 8 nM) than D2 (Ki:
    Formula:C27H29N5O
    Color and Shape:Solid
    Molecular weight:439.55

    Ref: TM-T62528

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Thielavin B

    CAS:
    Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.
    Formula:C31H34O10
    Color and Shape:Solid
    Molecular weight:566.6

    Ref: TM-T73066

    2500µg
    2,585.00€
  • YNT-3708

    CAS:
    YNT-3708 is an orexin receptor (OXR) agonist, exhibiting EC50 values of 14.6 nM for OX1R and 277 nM for OX2R.
    Formula:C35H36N4O6S
    Color and Shape:Solid
    Molecular weight:640.749

    Ref: TM-T206764

    10mg
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    50mg
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  • SB 258741 hydrochloride


    SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].
    Formula:C19H31ClN2O2S
    Color and Shape:Solid
    Molecular weight:386.98

    Ref: TM-T61724

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Monlunabant

    CAS:
    Monlunabant ((S)-MRI-1891), a solid dispersion compound, functions as an inhibitor of the cannabinoid CB1 receptor [1].
    Formula:C26H22ClF3N6O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:591.00

    Ref: TM-T79137

    5mg
    138.00€
    10mg
    208.00€
    25mg
    To inquire
    50mg
    627.00€
  • SGLT1/2-IN-1

    CAS:
    SGLT1/2-IN-1 is a dual SGLT1/SGLT2 inhibitor.
    Formula:C25H28O8
    Color and Shape:Solid
    Molecular weight:456.48

    Ref: TM-T62830

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Merigolix

    CAS:
    Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .
    Formula:C36H35F7N4O6
    Color and Shape:Solid
    Molecular weight:752.68

    Ref: TM-T73327

    25mg
    2,157.00€
    50mg
    2,832.00€
    100mg
    3,800.00€
  • MrgprX2 antagonist-6


    MrgprX2 antagonist-6 is a potent antiallergic agent with inhibitory effects on mast cell degranulation.
    Formula:C24H23F3N6O3
    Color and Shape:Solid
    Molecular weight:500.47

    Ref: TM-T63394

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • (S)-YNT-3708

    CAS:
    <p>(S)-YNT-3708 is the S-isomer of YNT-3708, demonstrating relatively low activity against OX1R and OX2R receptors, with EC50 values of 3595 nM and 1661 nM, respectively.</p>
    Formula:C35H36N4O6S
    Color and Shape:Solid
    Molecular weight:640.749

    Ref: TM-T206866

    10mg
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    50mg
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  • AChE/BChE-IN-21

    CAS:
    AChE/BChE-IN-21 is an antagonist of the histamine H3 receptor, a calcium channel blocker, and an acetylcholinesterase inhibitor. It exhibits neuroprotective activities against H2O2 and Aβ1-40, and can restore cognitive functions in AD mice.
    Formula:C38H54N4O4
    Color and Shape:Solid
    Molecular weight:630.86

    Ref: TM-T200193

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • SAR-150640

    CAS:
    SAR-150640, a selective β3-adrenergic receptor agonist, prevents an increase in MMP activity and production observed after LPS stimulation or in cases of chorioamnionitis.
    Formula:C25H35ClN2O7S
    Color and Shape:Solid
    Molecular weight:543.07

    Ref: TM-T200896

    25mg
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    50mg
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    100mg
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  • Carazolol hydrochloride

    CAS:
    Carazolol (BM 51052) hydrochloride is a potent antagonist of β1/β2-adrenoceptors and also serves as a powerful and selective agonist of β3-adrenoceptors. It is utilized in research focusing on hypertension.
    Formula:C18H23ClN2O2
    Molecular weight:334.84

    Ref: TM-T206098

    10mg
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    50mg
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  • S1PR1 agonist 1

    CAS:
    <p>S1PR1 agonist 1 is a potent agonist of S1PR1. S1PR1 agonist 1 has potential in autoimmune diseases.</p>
    Formula:C29H30N4O4
    Color and Shape:Solid
    Molecular weight:498.57

    Ref: TM-T63378

    25mg
    2,033.00€
    50mg
    2,645.00€
    100mg
    3,345.00€
  • 5-HT2A receptor agonist-7

    CAS:
    5-HT2A receptor agonist-7 (517) functions as a modulator of the 5-HT2A receptor, with an EC50 value of less than 100 nM.
    Formula:C12H11F2N3
    Molecular weight:235.233

    Ref: TM-T206848

    10mg
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    50mg
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  • Tofogliflozin

    CAS:
    Tofogliflozin specifically inhibits SGLT2; IC50s are 2.9 nM (human), 14.9 nM (rat), 6.4 nM (mouse).
    Formula:C22H26O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.44

    Ref: TM-T13179

    25mg
    1,730.00€
    50mg
    2,262.00€
    100mg
    2,945.00€
  • GPBAR1-IN-3

    CAS:
    GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].
    Formula:C21H23NO2
    Color and Shape:Solid
    Molecular weight:321.41

    Ref: TM-T60863

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Methacycline

    CAS:
    <p>Methacycline, a tetracycline antibiotic, inhibits bacterial protein synthesis and effectively suppresses epithelial-mesenchymal transition (EMT). It blocks EMT in vitro and inhibits fibrogenesis in vivo without directly affecting the TGF-β1Smad signaling pathway. As an antimicrobial agent, Methacycline holds potential for research in pulmonary fibrosis.</p>
    Formula:C22H22N2O8
    Color and Shape:Solid
    Molecular weight:442.42

    Ref: TM-T201726

    10mg
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    50mg
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  • RGS10 modulator-1

    CAS:
    RGS10 modulator-1 (compound 15) is an effective regulator of RGS10. It significantly reverses IFNγ-induced expression of both RGS10 protein and mRNA, as well as COX-2 mRNA and iNOS expression triggered by IFNγ.
    Formula:C16H15BrN2O3S2
    Color and Shape:Solid
    Molecular weight:427.336

    Ref: TM-T204267

    10mg
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    50mg
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  • MK-0812

    CAS:
    MK-0812 is a dual antagonist of the CCR2 and CCR5 receptors that can alleviate adipose inflammation in ob/ob mice.
    Formula:C24H34F3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.54

    Ref: TM-TQ0182

    1mg
    107.00€
    5mg
    250.00€
    10mg
    449.00€
  • Toladryl

    CAS:
    Toladryl is a derivative of Diphenhydramine that can cross the blood-brain barrier and exhibits oral activity, with antihistamine and anticholinergic properties. Its anticholinergic effects are approximately a tenth of those seen with Diphenhydramine, yet it offers 2-4 times the protection against lethal doses of histamine in guinea pigs. The side effects of Toladryl are fewer and milder compared to Diphenhydramine; however, at higher doses, it may cause symptoms such as insomnia, agitation, and disorientation related to the central nervous system. Toladryl is utilized in the research of allergic diseases.
    Formula:C18H23NO
    Color and Shape:Solid
    Molecular weight:269.38

    Ref: TM-T200797

    25mg
    1,630.00€
    50mg
    2,107.00€
    100mg
    2,617.00€
  • Cicaprost

    CAS:
    Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.
    Formula:C22H30O5
    Color and Shape:Solid
    Molecular weight:374.47

    Ref: TM-T61526

    25mg
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    50mg
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    100mg
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  • SR 142948-C3-NHMe

    CAS:
    <p>SR 142948-C3-NHMe is the methylated form of SR 142948.</p>
    Formula:C42H58N6O6
    Color and Shape:Solid
    Molecular weight:742.946

    Ref: TM-T204738

    10mg
    To inquire
    50mg
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  • BI 639667

    CAS:
    BI 639667, an azaindazole-class compound, potently inhibits CCR1 (IC50=1.8 nM in calcium flux assays).
    Formula:C22H18FN5O3S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:451.47

    Ref: TM-T14899

    1mg
    115.00€
    5mg
    274.00€
    10mg
    472.00€
    25mg
    885.00€
    50mg
    1,311.00€
    1mL*10mM (DMSO)
    303.00€
  • CCR5 antagonist 1

    CAS:
    CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.
    Formula:C39H46ClF2N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:738.33

    Ref: TM-T10714

    25mg
    3,820.00€
    50mg
    4,826.00€
    100mg
    6,460.00€
  • Aplaviroc

    CAS:
    Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.
    Formula:C33H43N3O6
    Purity:97.98% - 98.26%
    Color and Shape:Solid
    Molecular weight:577.71

    Ref: TM-T14307

    1mg
    517.00€
    5mg
    1,130.00€
    10mg
    1,549.00€
    25mg
    2,300.00€
    50mg
    3,097.00€
    100mg
    4,161.00€
  • APJ receptor agonist 8

    CAS:
    <p>APJ receptor agonist 8 is a small molecule agonist of the APJ receptor, enhancing load-independent cardiac contractility in isolated perfused rat hearts.</p>
    Formula:C24H27N7O5S
    Purity:98.31% - 99.60%
    Color and Shape:Solid
    Molecular weight:525.58

    Ref: TM-T85710

    1mg
    201.00€
    5mg
    497.00€
    10mg
    701.00€
    25mg
    1,094.00€
  • A2A receptor antagonist 2


    A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).
    Formula:C25H28FN7O3
    Color and Shape:Solid
    Molecular weight:493.53

    Ref: TM-T63326

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • ONO-8809

    CAS:
    ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.
    Formula:C30H46BrNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:596.66

    Ref: TM-T28251

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • 9-Methyl-β-carboline

    CAS:
    9-Methyl-β-carboline is a cognitive enhancer with neuroprotective, neurorestorative, and anti-inflammatory properties. Its behavioral effects may be linked to hippocampal dopamine levels and the stimulation of dendritic and synaptic proliferation.
    Formula:C12H10N2
    Color and Shape:Solid
    Molecular weight:182.221

    Ref: TM-T204669

    10mg
    To inquire
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  • MRS4833

    CAS:
    MRS4833 (compound 15) is an orally active, potent, competitive antagonist of P2Y14R, exhibiting IC50 values of 5.92 nM for hP2Y14R and 4.8 nM for mP2Y14R. It reduces airway eosinophilia in protease-mediated asthma models and reverses chronic neuropathic pain in mouse CCI models.
    Formula:C30H24F3NO3
    Color and Shape:Solid
    Molecular weight:503.51

    Ref: TM-T200837

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  • Fosrolapitant

    CAS:
    Fosrolapitant is an antagonist of the neurokinin 1 (NK1) receptor.
    Formula:C27H29F6N2O8P
    Color and Shape:Solid
    Molecular weight:654.49

    Ref: TM-T201161

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  • BMS-986104

    CAS:
    BMS-986104 is an effective selective modulator of the S1P1 receptor. It demonstrates efficacy in the mouse EAE model, comparable to that of FTY720. Furthermore, BMS-986104 shows promising remyelination properties in three-dimensional brain cell cultures subjected to lysophosphatidylcholine (LPC)-induced demyelination.
    Formula:C22H35NO
    Color and Shape:Solid
    Molecular weight:329.52

    Ref: TM-T200882

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  • MRT-92

    CAS:
    MRT-92 is an antagonist of Smoothened (Smo) with anti-cancer activity, featuring a binding affinity (Ki) of 0.7 nM. It inhibits the Hedgehog signaling pathway by obstructing the overlapping binding sites within the transmembrane domain of the Smoothened receptor and suppresses the proliferation of cerebellar granule cells in rodents (IC50=0.4 nM). MRT-92 is utilized for research into cerebellar gliomas.
    Formula:C33H34N4O5
    Color and Shape:Solid
    Molecular weight:566.65

    Ref: TM-T200033

    25mg
    2,225.00€
    50mg
    2,921.00€
    100mg
    3,921.00€
  • Befiradol hydrochloride

    CAS:
    <p>Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.</p>
    Formula:C20H23Cl2F2N3O
    Purity:99.1%
    Color and Shape:Solid
    Molecular weight:430.32

    Ref: TM-T62385

    1mg
    104.00€
    5mg
    251.00€
    10mg
    368.00€
    25mg
    592.00€
    50mg
    817.00€
    100mg
    1,093.00€
    200mg
    1,473.00€
  • Nedemelteon

    CAS:
    Nedemelteon is an agonist of the melatonin receptor (melatonin receptor).
    Formula:C15H18N2O2
    Color and Shape:Solid
    Molecular weight:258.32

    Ref: TM-T201036

    25mg
    1,931.00€
    50mg
    2,529.00€
    100mg
    3,333.00€
  • Opipramol dihydrochloride

    CAS:
    Opipramol (Ensidon) is an atypical tricyclic antidepressant (TCA) primarily functioning as a sigma (σ) receptor agonist. It interacts effectively with sigma recognition sites, having a Ki value of 50 nM. Opipramol is applicable in the study of generalized anxiety disorder (GAD).
    Formula:C23H31Cl2N3O
    Color and Shape:Solid
    Molecular weight:436.418

    Ref: TM-T204660

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  • Aeruginosin 98-B

    CAS:
    Aeruginosin 98-B, a protease inhibitor, effectively inhibits trypsin, plasmin, and thrombin with IC50 values of 0.6, 7.0, and 10.0 μg/mL, respectively.
    Formula:C29H46N6O9S
    Color and Shape:Solid
    Molecular weight:654.78

    Ref: TM-T72736

    25mg
    4,436.00€
    50mg
    5,871.00€
    100mg
    8,360.00€
  • RWJ-68022

    CAS:
    RWJ-68022 (Example 9) is a cyclopentene derivative that serves as a motilin receptor antagonist. It competes with motilin and erythromycin at motilin receptor sites and is applicable in research on gastrointestinal disorders.
    Formula:C34H37Cl3N4O4
    Color and Shape:Solid
    Molecular weight:672.04

    Ref: TM-T211737

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  • CCR3 antagonist 2

    CAS:
    CCR3 antagonist2 (example 66) is a CCR3 antagonist useful for researching inflammatory or allergic diseases, particularly those affecting the respiratory tract, such as inflammatory or obstructive airway conditions.
    Formula:C21H28ClN5O3
    Color and Shape:Solid
    Molecular weight:433.93

    Ref: TM-T212174

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  • NPRA agonist-11

    CAS:
    NPRA agonist-11 (Example 161) is an NPRA (NPR1) agonist with AC50 values of 1.681 μM and 0.989 μM for human and monkey, respectively. It is applicable in research on cardiovascular and other diseases.
    Formula:C37H52FN7O2
    Color and Shape:Solid
    Molecular weight:645.85

    Ref: TM-T211535

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  • Avitriptan

    CAS:
    Avitriptan is a 5-HT1B/1D receptor agonist with pKi values of 7.44 for 5-HT1Brat, 7.68 for 5-HT1Bhuman, and 8.36 for 5-HT1Dhuman. It can induce contraction in isolated coronary arteries and is used for the treatment of migraines.
    Formula:C22H30N6O3S
    Molecular weight:458.577

    Ref: TM-T206109

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  • D1R antagonist 1

    CAS:
    Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].
    Formula:C22H26BrNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.35

    Ref: TM-T78735

    5mg
    3,392.00€
  • GLP-1 receptor agonist 11

    CAS:
    GLP-1 Receptor Agonist 11 (compound 3) acts as an effective agonist for the GLP Receptor, finding use in research related to conditions like diabetes and non-alc. fatty liver disease [1].
    Formula:C31H31ClFN3O4
    Color and Shape:Solid
    Molecular weight:564.05

    Ref: TM-T86503

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  • Sigma-1 receptor antagonist 6

    CAS:
    Sigma-1 receptor antagonist 6 (Compound 12), a σ1R antagonist, demonstrates significant antiallodynic effects by targeting the Sigma-1 receptor (σ1R). This compound is effective in animal models for neuropathic pain, particularly for reducing mechanical allodynia caused by paclitaxel.
    Formula:C32H34N6
    Color and Shape:Solid
    Molecular weight:502.65

    Ref: TM-T89901

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  • HU 433

    CAS:
    <p>HU 433, a synthetic cannabinoid, acts as a CB2 receptor agonist and is an enantiomer of HU 308. It provides anti-inflammatory and neuroprotective effects by binding to the CB2 receptor, primarily found on immune cells, thereby modulating immune responses and inflammation. Additionally, HU 433 influences microglial signaling pathways, particularly LPS and IFNγ-mediated routes, affecting the phosphorylation of MAPKs, including ERK1/2, JNK, p38, and Akt. This compound is valuable in researching neuroinflammation and retinal diseases.</p>
    Formula:C27H42O3
    Color and Shape:Solid
    Molecular weight:414.62

    Ref: TM-T88373

    25mg
    1,784.00€
    50mg
    2,333.00€
    100mg
    3,039.00€
  • Anti-MRSA agent 19

    CAS:
    Anti-MRSA agent 19 (Compound 1) is an antibiotic that exhibits activity against Staphylococcus aureus. It is active against 40 clinical isolates from the CDC, representing diverse bacterial species with various resistance factors, including resistance to vancomycin, aminoglycoside/tetracycline, and oxazolidinone (median MIC=4 μg/mL).
    Formula:C15H10Cl3NO4
    Color and Shape:Solid
    Molecular weight:374.6

    Ref: TM-T201507

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  • Leukotriene B4 dimethyl amide

    CAS:
    LTB4 dimethyl amide: inhibits human neutrophil degranulation and rat lysozyme release; antagonizes LTB4 receptor on guinea pig lung membranes (Ki = 130 nM).
    Formula:C22H37NO3
    Color and Shape:Solid
    Molecular weight:363.53

    Ref: TM-T37618

    25µg
    598.00€
    50µg
    1,121.00€
    100µg
    2,118.00€
  • UNC10099984A

    CAS:
    UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a Ki value of 4.6 nM and an EC50 of 6.2 nM for β-arrestin. This compound is useful for research into central nervous system diseases related to the D2 receptor.
    Formula:C24H29Cl2N3O2
    Color and Shape:Solid
    Molecular weight:462.41

    Ref: TM-T201623

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  • ASP-2205

    CAS:
    ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), enhances the urethral closure reflex mediated by the genital nerve, thereby preventing urinary incontinence.
    Formula:C19H28N2O
    Color and Shape:Solid
    Molecular weight:300.44

    Ref: TM-T201450

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  • Quinagolide Free Base

    CAS:
    Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.
    Formula:C20H33N3O3S
    Color and Shape:Solid
    Molecular weight:395.56

    Ref: TM-T68483

    25mg
    2,442.00€
    50mg
    3,212.00€
    100mg
    4,370.00€
  • Rodatristat ethyl

    CAS:
    Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low doses.
    Formula:C29H31ClF3N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.04

    Ref: TM-T16779

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  • BAY-899

    CAS:
    BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.
    Formula:C25H19F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.45

    Ref: TM-T10476

    25mg
    2,680.00€
    50mg
    3,307.00€
    100mg
    4,180.00€
  • Udifitimod

    CAS:
    Udifitimod (BMS-986166) is a potent, selective, and orally active modulator of the S1P1R receptor, showing potential for research in autoimmune diseases.
    Formula:C25H33NO2
    Color and Shape:Solid
    Molecular weight:379.54

    Ref: TM-T73092

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  • Nolpitantium besilate

    CAS:
    Nolpitantium besilate is a neurokinin-1 receptor antagonist.
    Formula:C43H50Cl2N2O5S
    Color and Shape:Solid
    Molecular weight:777.84

    Ref: TM-T70455

    25mg
    2,870.00€
    50mg
    3,781.00€
    100mg
    5,225.00€
  • RBM10-8

    CAS:
    RBM10-8 irreversibly inhibits human sphingosine-1- phosphate lyase (hS1PL) while behaving also as an enzyme substrate.
    Formula:C17H36NO5P
    Color and Shape:Solid
    Molecular weight:365.45

    Ref: TM-T61406

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • 8-iso Prostaglandin F3α

    CAS:
    8-iso PGF3α is an isoprostane produced from the free-radical peroxidation of EPA.
    Formula:C20H32O5
    Color and Shape:Solid
    Molecular weight:352.47

    Ref: TM-T36164

    25µg
    948.00€
    50µg
    1,691.00€
    100µg
    3,002.00€
  • MF-592

    CAS:
    MF-592: EP4 receptor antagonist, hEP4 IC50 3 nM, hWB IC50 78 nM, great oral PK, rat arthritis ED50 0.1 mg/kg/day, promising for development.
    Formula:C34H33Cl2N3O6S
    Color and Shape:Solid
    Molecular weight:682.61

    Ref: TM-T71510

    25mg
    2,727.00€
    50mg
    3,591.00€
    100mg
    4,940.00€
  • L-654284

    CAS:
    L-654284 is an α2-adrenergic receptor antagonist characterized by its notable selectivity. It competes with 3H-clonidine and 3H-rauwolscine for binding in vitro, exhibiting Ki values of 0.8 nM and 1.1 nM, respectively. L-654284 effectively blocks the pre-ejaculatory effects of clonidine in isolated rat vas deferens, with a pA2 value of 9.1. The compound demonstrates significant selectivity for α2 over α1 adrenergic receptors, with a Ki value of 110 nM against 3H-prazosin binding. In vivo, L-654284 significantly increases the turnover of norepinephrine in the rat cerebral cortex, indicating its activity in blocking α2-adrenergic receptors within the central nervous system.
    Formula:C18H24N2O4S
    Color and Shape:Solid
    Molecular weight:364.46

    Ref: TM-T201031

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  • AB-FUBINACA 3-fluorobenzyl isomer

    CAS:
    AB-FUBINACA 3-fluorobenzyl isomer is a synthetic cannabinoid and an indazole derivative, exhibiting high affinity for central CB1 receptors (Ki= 0.9 nM) and possessing anticonvulsant activity.
    Formula:C20H21FN4O2
    Color and Shape:Solid
    Molecular weight:368.41

    Ref: TM-T201486

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  • O-1269

    CAS:
    O-1269 acts as a partial agonist for the cannabinoid receptor 1 (CB1R), with a binding affinity (Ki) of 32 nM. Additionally, it exhibits analgesic properties.
    Formula:C22H22Cl3N3O
    Color and Shape:Solid
    Molecular weight:450.79

    Ref: TM-T201557

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  • FDU-PB-22

    CAS:
    FDU-PB-22, a novel synthetic cannabinoid, undergoes rapid metabolism in human liver microsomes (HLM) with a half-life of 12.4 minutes.
    Formula:C26H18FNO2
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T201691

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  • GRK6-IN-4

    CAS:
    GRK6-IN-4 is an inhibitor of G protein-coupled receptor kinase 6 (GRK6) with an IC50 value of 1.56 μM. GRK6-IN-4 is applicable for research related to hematological malignancies, inflammatory diseases, and autoimmune disorders.
    Formula:C15H15N5
    Color and Shape:Solid
    Molecular weight:265.313

    Ref: TM-T204959

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  • Etoperidone

    CAS:
    Etoperidone is an antidepressant that acts as an orally active reuptake inhibitor for serotonin (serotonin) and noradrenaline (nor-adrenaline). It demonstrates specific binding affinities (Kd) for several receptors: 36 nM at the 5-HT2 receptor, 38 nM at the α1-adrenergic receptor (α1-adrenergic receptor), 85 nM at the 5-HT1A receptor, and 570 nM at the α2-adrenergic receptor (α2-adrenergic receptor).
    Formula:C19H28ClN5O
    Color and Shape:Solid
    Molecular weight:377.91

    Ref: TM-T201838

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  • CI-936

    CAS:
    CI-936 (MRS-3310) is an orally active A2 agonist with a binding affinity of 25 nM. In preclinical studies, it has demonstrated potent and selective effects, indicating potential antipsychotic efficacy. Additionally, CI-936 inhibits exploratory behavior in mice.
    Formula:C24H25N5O4
    Color and Shape:Solid
    Molecular weight:447.49

    Ref: TM-T211093

    10mg
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  • Meluadrine

    CAS:
    Meluadrine, a potent agonist of the β2 adrenergic receptor, is one of the metabolites of Tulobuterol [1].
    Formula:C12H18ClNO2
    Molecular weight:243.73

    Ref: TM-T86882

    10mg
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  • 8 Hydroxy PIPAT oxalate

    CAS:
    8 Hydroxy PIPAT oxalate is a selective 5-HT1A receptor agonist that enhances the spontaneous release of histamine by promoting the degranulation of mast cells in guinea pig and human intestinal preparations. By activating the serotonin signaling pathway, this compound demonstrates potential in regulating gastrointestinal functions and offers insight into the management and suppression of functional gastrointestinal disorders such as irritable bowel syndrome. Its effects in increasing histamine release could play a crucial role in gastrointestinal regulation.
    Formula:C18H24INO5
    Color and Shape:Solid
    Molecular weight:461.29

    Ref: TM-T201052

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  • 14,15-dehydro Leukotriene B4

    CAS:
    LTB4 is a leukocyte-activating fatty acid via 5-lipoxygenase. Two receptors, BLT1 and BLT2, bind it. 14,15-dehydro LTB4 is a stronger BLT1 antagonist.
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T37260

    25µg
    465.00€
    50µg
    898.00€
    100µg
    1,673.00€
  • Jimscaline

    CAS:
    Jimscaline (compound R-(-)2) is a 5-HT2A agonist and a mescaline analogue, used in neuroscience research.
    Formula:C13H19NO3
    Molecular weight:237.295

    Ref: TM-T204304

    10mg
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  • CTW0404

    CAS:
    CTW0404 is an effective positive allosteric modulator (PAM) of the 5-HT receptor, with promising implications for research into neuropsychiatric disorders.
    Formula:C21H33N3O2
    Molecular weight:359.51

    Ref: TM-T207589

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  • PD-147693

    CAS:
    PD-147693 (compound II) is an active metabolite of the presynaptic dopamine autoreceptor agonist CI-1007, and it exhibits antipsychotic activity similar to CI-1007.
    Formula:C24H27NO
    Molecular weight:345.477

    Ref: TM-T204694

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  • LAB687

    CAS:
    LAB687 (Compound 2a) is an inhibitor of microsomal triglyceride transfer protein (MTP) with an IC50 of 0.9 nM for inhibiting the secretion of apolipoprotein B (apoB) in HepG2 cells. Additionally, LAB687 acts as a Smoothened (Smo) antagonist, exhibiting IC50 values of 2.48 μM and 3.42 μM for mouse and human Smo receptors, respectively. This compound is effective in reducing triglyceride and low-density lipoprotein cholesterol (LDL-C) levels and in inhibiting the Hedgehog signaling pathway.
    Formula:C26H23F3N2O3
    Color and Shape:Solid
    Molecular weight:468.47

    Ref: TM-T212506

    10mg
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  • PSB-KK1415

    CAS:
    PSB-KK1415 is a selective agonist for the human orphan G protein-coupled receptor GPR18, with an EC50 of 19.1 nM.
    Formula:C24H23ClN6O2
    Molecular weight:462.93

    Ref: TM-T210393

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  • RXFP1 receptor agonist-10

    CAS:
    RXFP1 receptor agonist-10 (Compound 188) is an RXFP1 receptor agonist with an EC50 of 0.5 nM. It is useful for research into heart failure.
    Formula:C39H44F6N4O5
    Color and Shape:Solid
    Molecular weight:762.78

    Ref: TM-T210809

    10mg
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  • RS 61756-007

    CAS:
    RS 61756-007 is a selective thromboxane receptor (TP) agonist.
    Formula:C23H28O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.47

    Ref: TM-T26141

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  • MCTR1

    CAS:
    MCTR1, a pro-resolving mediator derived from DHA, promotes tissue repair and reduces inflammation by enhancing phagocytosis and decreasing eicosanoids.
    Formula:C32H47N3O9S
    Color and Shape:Solid
    Molecular weight:649.8

    Ref: TM-T37505

    10µg
    537.00€
    25µg
    1,264.00€
    50µg
    2,395.00€
    100µg
    3,990.00€
  • Disulergine

    CAS:
    Disulergine is a dopamine receptor agonist. It also prolactin release-inhibiting 8 alpha-amino-ergoline.
    Formula:C17H24N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.46

    Ref: TM-T24003

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  • Ro-24-4736

    CAS:
    Ro 24-4736 is an effective and selective platelet-activating factor antagonist.
    Formula:C31H20ClN5OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.04

    Ref: TM-T16768

    25mg
    2,147.00€
    50mg
    2,917.00€
    100mg
    3,790.00€
  • GLP-1 receptor agonist 15

    CAS:
    GLP-1 receptor agonist 15 (Example 4) is a GLP receptor agonist with an EC50 of 0.74 nM. It exhibits an IC50 of 10.1 μM against the hERG potassium ion channel. This compound is applicable for research in the diabetes field.
    Formula:C32H31ClFN3O5
    Color and Shape:Solid
    Molecular weight:592.057

    Ref: TM-T204742

    10mg
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  • Vibegron

    CAS:
    Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).
    Formula:C26H28N4O3
    Color and Shape:Solid
    Molecular weight:444.53

    Ref: TM-T35052

    25mg
    1,414.00€
    50mg
    1,995.00€
    100mg
    2,725.00€
  • SSTR5 antagonist 2 hydrochloride


    SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.
    Formula:C32H36ClFN2O5
    Color and Shape:Solid
    Molecular weight:583.09

    Ref: TM-T64119

    25mg
    1,454.00€
    50mg
    1,890.00€
    100mg
    3,068.00€
  • Oral antiplatelet agent 1

    CAS:
    Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.
    Formula:C23H24N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.53

    Ref: TM-T12316

    25mg
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  • PF-4693627

    CAS:
    PF-4693627 is an effective and selective microsomal prostaglandin E synthase-1 inhibitor (IC50=3 nM).
    Formula:C26H29Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:502.43

    Ref: TM-T16504

    1mg
    234.00€
    5mg
    1,093.00€
    10mg
    2,052.00€
    500µg
    131.00€
  • AGH-107

    CAS:
    AGH-107 is a highly selective 5-HT7 receptor agonist that can cross the blood-brain barrier, featuring a Ki value of 6 nM and an EC50 value of 19 nM. Demonstrating high selectivity for central nervous system targets, AGH-107 also exhibits high metabolic stability and low toxicity in HEK-293 and HepG2 cell cultures.
    Formula:C13H12IN3
    Color and Shape:Solid
    Molecular weight:337.16

    Ref: TM-T201735

    10mg
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  • Flucopride

    CAS:
    Flucopride (Compound 4a) acts as an acetylcholinesterase inhibitor (AChE) with an IC50 value of 24 nM and serves as a partial agonist for the human 5-HT4 receptor (5-HT4R) with a Ki of 9.6 nM for (h)5-HT4R. It promotes non-amyloidogenic processing of APP in COS-7 cells transiently expressing (h)5-HT4R with an EC50 of 23.0 nM. Flucopride is also likely to exhibit significant gastrointestinal tract (GIT) penetration and blood-brain barrier (BBB) permeability, as determined in PAMPA experiments.
    Formula:C22H33FN2O2
    Color and Shape:Solid
    Molecular weight:376.51

    Ref: TM-T201815

    10mg
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  • R-137696

    CAS:
    R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal stomach. It is utilized in research related to functional dyspepsia.
    Formula:C17H23N3O2
    Color and Shape:Solid
    Molecular weight:301.38

    Ref: TM-T201501

    10mg
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    50mg
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  • SB-423562

    CAS:
    SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
    Formula:C26H32N2O4
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:436.54

    Ref: TM-T12846

    1mg
    39.00€
    5mg
    85.00€
    10mg
    126.00€
    25mg
    221.00€
    50mg
    338.00€
    100mg
    467.00€
    200mg
    640.00€
    1mL*10mM (DMSO)
    94.00€
  • LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:480.39

    Ref: TM-T63166

    1mg
    202.00€
    5mg
    512.00€
    10mg
    738.00€
    25mg
    1,121.00€
    50mg
    1,510.00€
    100mg
    2,062.00€
  • BQ-788

    CAS:
    BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.
    Formula:C34H51N5O7
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:641.8

    Ref: TM-T10595

    1mg
    137.00€
    2mg
    188.00€
    5mg
    329.00€
    10mg
    472.00€
    25mg
    753.00€
    50mg
    1,017.00€
    100mg
    1,378.00€
    500mg
    2,737.00€
    1mL*10mM (DMSO)
    360.00€
  • AZD-5672

    CAS:
    AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.
    Formula:C32H38F2N2O5S2
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:632.78

    Ref: TM-T30260

    1mg
    202.00€
    5mg
    459.00€
    10mg
    643.00€
    25mg
    938.00€
    50mg
    1,311.00€
    100mg
    1,786.00€
    1mL*10mM (DMSO)
    560.00€
  • Vofopitant dihydrochloride

    CAS:
    Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.
    Formula:C21H25Cl2F3N6O
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:505.36

    Ref: TM-T13329L

    1mg
    99.00€
    5mg
    235.00€
    10mg
    376.00€
    25mg
    712.00€
    50mg
    1,064.00€
    100mg
    1,454.00€
    500mg
    2,822.00€
    1mL*10mM (DMSO)
    261.00€
  • SB-224289 hydrochloride

    CAS:
    SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
    Formula:C32H33ClN4O3
    Purity:98.99% - 99.96%
    Color and Shape:Solid
    Molecular weight:557.08

    Ref: TM-T12841

    1mg
    42.00€
    5mg
    88.00€
    10mg
    115.00€
    25mg
    To inquire
    50mg
    To inquire
    1mL*10mM (DMSO)
    101.00€
  • Vofopitant

    CAS:
    Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).
    Formula:C21H23F3N6O
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:432.44

    Ref: TM-T13329

    1mg
    99.00€
    5mg
    235.00€
    10mg
    349.00€
    25mg
    565.00€
    50mg
    818.00€
    100mg
    1,103.00€
    500mg
    2,205.00€
  • AZD5462

    CAS:
    AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.
    Formula:C30H41FN2O6
    Purity:98.32% - 99.63%
    Color and Shape:Solid
    Molecular weight:544.65

    Ref: TM-T63838

    1mg
    354.00€
    5mg
    850.00€
    10mg
    1,206.00€
    25mg
    1,882.00€
    50mg
    2,642.00€
    100mg
    3,345.00€
  • Dersimelagon

    CAS:
    Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.
    Formula:C36H45F4N3O5
    Purity:97.35% - 98.23%
    Color and Shape:Solid
    Molecular weight:675.75

    Ref: TM-T25310

    1mg
    79.00€
    5mg
    180.00€
    10mg
    264.00€
    25mg
    452.00€
    50mg
    647.00€
  • BMS-986141

    CAS:
    BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614
    Formula:C27H23N5O5S2
    Purity:98.43% - 99.26%
    Color and Shape:Solid
    Molecular weight:561.63

    Ref: TM-T63966

    1mg
    612.00€
    5mg
    1,216.00€
    10mg
    1,549.00€
    25mg
    2,213.00€
  • PF-07258669

    CAS:
    PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
    Formula:C25H27FN6O2
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:462.52

    Ref: TM-T69526

    1mg
    802.00€
    5mg
    1,605.00€
    10mg
    2,612.00€
    25mg
    5,159.00€
    50mg
    8,255.00€
  • Treprostinil diethanolamine

    CAS:
    Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,
    Formula:C27H45NO7
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:495.65

    Ref: TM-T63349

    1mg
    35.00€
    5mg
    80.00€
    10mg
    120.00€
    25mg
    235.00€
    50mg
    349.00€
    100mg
    515.00€
  • Rolapitant hydrochloride

    CAS:
    Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.
    Formula:C25H27ClF6N2O2
    Purity:98.35% - 99.79%
    Color and Shape:Solid
    Molecular weight:536.94

    Ref: TM-T3724

    1mg
    153.00€
    5mg
    365.00€
    10mg
    520.00€
    25mg
    780.00€
    50mg
    1,054.00€
    100mg
    1,425.00€
    200mg
    1,882.00€
    1mL*10mM (DMSO)
    439.00€
  • BIBP3226 TFA

    CAS:
    BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).
    Formula:C29H32F3N5O5
    Color and Shape:Solid
    Molecular weight:587.59

    Ref: TM-T10540

    1mg
    Discontinued
    Discontinued product
  • JMV 2959

    CAS:
    JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).
    Formula:C30H32N6O2
    Color and Shape:Solid
    Molecular weight:508.61

    Ref: TM-T11719L

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product
  • ML-00253764 hydrochloride

    CAS:
    ML-00253764 hydrochloride is an antagonist of nonpeptidic melanocortin receptor 4 (MC4R) (Ki and IC50 of 0.16 µM and 0.103 µM, respectively).
    Formula:C18H19BrClFN2O
    Color and Shape:Solid
    Molecular weight:413.71

    Ref: TM-T12072

    1mg
    Discontinued
    Discontinued product
  • Beraprost sodium

    CAS:
    Beraprost sodium is a stable and orally active prodrug of PGI2.
    Formula:C24H29NaO5
    Color and Shape:Solid
    Molecular weight:420.481

    Ref: TM-T13859

    1mg
    Discontinued
    Discontinued product
  • HOKU-81

    CAS:
    HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.
    Formula:C12H18ClNO2
    Color and Shape:Solid
    Molecular weight:243.73

    Ref: TM-T15498

    1mg
    Discontinued
    Discontinued product
  • SB-399885 hydrochloride

    CAS:
    SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
    Formula:C18H22Cl3N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.81

    Ref: TM-T12843

    1mg
    Discontinued
    Discontinued product
  • SR 146131

    CAS:
    SR 146131 is a potent and selective agonist of the nonpeptide receptor.
    Formula:C32H36ClN3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:610.16

    Ref: TM-T16935

    1mg
    Discontinued
    Discontinued product
  • CYM 9484

    CAS:
    CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with an IC50 value of 19 nM.
    Formula:C27H31N3O3S2
    Color and Shape:Solid
    Molecular weight:509.68

    Ref: TM-T10921

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product
  • ML-290

    CAS:
    ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.
    Formula:C24H21F3N2O5S
    Color and Shape:Solid
    Molecular weight:506.49

    Ref: TM-T16101

    1mg
    Discontinued
    Discontinued product
  • 7-Desmethyl-agomelatine

    CAS:
    7-Desmethyl-agomelatine, a metabolite of Agomelatine, exhibits lower activity than Agomelatine, which functions as a melatonergic (MT1 and MT2) agonist and 5-HT2C antagonist.
    Formula:C14H15NO2
    Color and Shape:Solid
    Molecular weight:229.27

    Ref: TM-T10193

    1mg
    Discontinued
    Discontinued product
  • Pumosetrag Hydrochloride

    CAS:
    Pumosetrag Hydrochloride is an orally available 5-HT3 partial agonist. It is developed for the treatment of irritable bowel syndrome and gastroesophageal reflux disease.
    Formula:C15H18ClN3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.84

    Ref: TM-T16683

    1mg
    Discontinued
    Discontinued product
  • Arotinolol

    CAS:
    Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand [125I-ICYP] to [5HT1B-serotonergic] receptor sites. It is an antihypertensive agent.
    Formula:C15H21N3O2S3
    Color and Shape:White Solid
    Molecular weight:371.54

    Ref: TM-T10371

    1mg
    Discontinued
    Discontinued product
  • SHA 68

    CAS:
    SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with IC50 values of 22.0 nM for NPSR Asn107 and 23.8 nM for NPSR Ile107.
    Formula:C26H24FN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.49

    Ref: TM-T12895

    1mg
    Discontinued
    Discontinued product
  • Protease-Activated Receptor-4

    CAS:
    Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
    Formula:C33H46N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:666.77

    Ref: TM-T7380

    1mg
    Discontinued
    Discontinued product
  • Patecibart

    CAS:
    <p>Patecibart is a humanized immunoglobulin G4-kappa monoclonal antibody that functions as an antagonist to the endothelin receptor A (EDNRA).</p>
    Purity:98%
    Color and Shape:Liquid

    Ref: TM-T81538

    ne
    Discontinued
    1mg
    Discontinued
    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • Sarizotan

    CAS:
    Sarizotan (EMD 128130) is an orally active compound that acts as an agonist for serotonin 5-HT 1A receptors and dopamine receptors, with IC50 values of 6.5 nM for rat 5-HT 1A, 0.1 nM for human 5-HT 1A, 15.1 nM for rat D 2, 17 nM for human D 2, 6.8 nM for human D 3, and 2.4 nM for human D 4.2.
    Formula:C22H21FN2O
    Color and Shape:Solid
    Molecular weight:348.421

    Ref: TM-T40439

    ne
    Discontinued
    Discontinued product
  • 6-Chloro-5-(2-chloroethyl)indolin-2-one

    CAS:
    6-Chloro-5-(2-chloroethyl)indolin-2-one is a useful organic compound for research related to life sciences. The catalog number is T64862 and the CAS number is 118289-55-7.
    Formula:C10H9Cl2NO
    Color and Shape:Solid
    Molecular weight:230.09

    Ref: TM-T64862

    ne
    Discontinued
    Discontinued product
  • 3-Hydroxybenzylamine

    CAS:
    3-Hydroxybenzylamine is a useful organic compound for research related to life sciences. The catalog number is T124305 and the CAS number is 73604-31-6.
    Formula:C7H9NO
    Color and Shape:Solid
    Molecular weight:123.155

    Ref: TM-T124305

    ne
    Discontinued
    Discontinued product
  • 1-Oleoyl Lysophosphatidic Acid

    CAS:
    <p>1-Oleoyl Lysophosphatidic Acid (1-Oleoyl LPA) is a biologically active phospholipid that can be used to study cancer and atherosclerosis.</p>
    Formula:C21H41O7P
    Color and Shape:Solid
    Molecular weight:436.52

    Ref: TM-T36907

    22.91mM*1
    Discontinued
    22.91mM*100
    Discontinued
    22.91mM*2.5
    Discontinued
    22.91mM*500
    Discontinued
    Discontinued product
  • Propiram fumarate HCl

    CAS:
    <p>Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.</p>
    Formula:C16H25N3O·xClH
    Purity:99.25%
    Color and Shape:Soild

    Ref: TM-T28453L

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Amelubant

    CAS:
    Amelubant (BIIL 284) is a prodrug of active metabolites BIIL 260 and BIIL 315 with anti-inflammatory activity[1]. It is a potent, oral, long-acting LTB4 receptor antagonist that negligibly binds to the LTB4 receptor, exhibiting Kis of 221 nM and 230 nM in vital cells and membranes.
    Formula:C33H34N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:538.63

    Ref: TM-T14210

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • SKF 89748

    CAS:
    SKF 89748 is an agonists of alpha 1-adrenoceptor.
    Formula:C12H17NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:223.33

    Ref: TM-T28789

    25mg
    Discontinued
    Discontinued product
  • BRL 15572

    CAS:
    BRL 15572 is a useful organic compound for research related to life sciences. The catalog number is T64501 and the CAS number is 734517-40-9.
    Formula:C25H27ClN2O
    Color and Shape:Solid
    Molecular weight:406.95

    Ref: TM-T64501

    ne
    Discontinued
    Discontinued product
  • Goserelin acetate(65807-02-5 Free base)


    <p>Goserelin acetate (ICI-118630 acetate) is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>
    Purity:99.77%
    Color and Shape:Odour Solid

    Ref: TM-T36918L

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • GSK-3050002


    <p>GSK-3050002 (HGS-1035) is a humanized IgG1 antibody that targets and binds to CCL20. It holds potential for inflammation research. For isotype control, refer to Human IgG1 kappa, Isotype Control.</p>
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-766

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • 1-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol

    CAS:
    1-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-yl)ethanol is a useful organic compound for research related to life sciences. The catalog number is T65156 and the CAS number is 24155-42-8.
    Formula:C11H10Cl2N2O
    Color and Shape:Solid
    Molecular weight:257.11

    Ref: TM-T65156

    ne
    Discontinued
    Discontinued product
  • (R)-(-)-α-Methylhistamine dihydrochloride

    CAS:
    R(-)-alpha-Methylhistamine 2HCl is an effective and selective agonist of the H3 histamine receptor.
    Formula:C6H13Cl2N3
    Color and Shape:Solid
    Molecular weight:198.09

    Ref: TM-T24698

    ne
    Discontinued
    Discontinued product
  • BX471 hydrochloride

    CAS:
    BX471 hydrochloride (ZK-811752 hydrochloride) is a potent, selective non-peptide CCR1 antagonist with a Ki of 1 nM for human CCR1, exhibiting 250-fold selectivity over CCR2, CCR5, and CXCR4.
    Formula:C21H25Cl2FN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.35

    Ref: TM-T14845

    ne
    Discontinued
    Discontinued product
  • 4-Hydroxypropranolol hydrochloride

    CAS:
    4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic receptors (pA2s: 8.24 and 8.26).
    Formula:C16H22ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:311.8

    Ref: TM-T10150

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • (Rac)-Zevaquenabant

    CAS:
    (Rac)-Zevaquenabant ((Rac)-MRI-1867, compound 6b) is a potent and selective antagonist of cannabinoid receptor type 1 (CB1R) and inducible nitric oxide synthase (iNOS), with a binding affinity (Ki) of 5.7 nM for CB1R. It holds promise as an investigative tool in liver fibrosis research due to these characteristics.
    Formula:C25H21ClF3N5O2S
    Color and Shape:Solid
    Molecular weight:547.98

    Ref: TM-T39074

    ne
    Discontinued
    Discontinued product
  • N-methyl-2-AI (hydrochloride)

    CAS:
    N-methyl-2-AI (hydrochloride) is a useful organic compound for research related to life sciences. The catalog number is T66396 and the CAS number is 10408-85-2.
    Formula:C10H14ClN
    Color and Shape:Solid
    Molecular weight:183.68

    Ref: TM-T66396

    ne
    Discontinued
    Discontinued product
  • Vornorexant

    CAS:
    Vornorexant (ORN-0829; TS-142) is a potent dual OX1R and OX2R antagonist with IC50 values of 1.05 nM and 1.27 nM, respectively. It exhibits potent sleep-promoting effects in vivo and can be used for insomnia treatment research.
    Formula:C23H22FN7O2
    Color and Shape:Solid
    Molecular weight:447.474

    Ref: TM-T39004

    ne
    Discontinued
    Discontinued product
  • CRTh2 antagonist 3

    CAS:
    CRTh2 antagonist 3, a potent molecule, activates PDK1 (EC50=2μM, Kd=8.4μM) and may cause cardiovascular inflammation.
    Formula:C19H20N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.44

    Ref: TM-T10890

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • dapitant

    CAS:
    Dapitant, a non-peptide, selective antagonist of human NKI receptors, is representative of the 7,7,4-triarylperhydroisoindol-4-ols.
    Formula:C37H39NO4
    Color and Shape:Solid
    Molecular weight:561.71

    Ref: TM-T68049

    ne
    Discontinued
    Discontinued product
  • TAK-683

    CAS:
    TAK-683: a full KISS1R agonist, IC50=170 pM; a nonapeptide metastin analog with human EC50=0.96 nM, rat EC50=1.6 nM.
    Formula:C64H83N17O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1298.45

    Ref: TM-TP2156L

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Desmethyl cariprazine

    CAS:
    Desmethyl cariprazine is a Cariprazine active metabolite. Cariprazine, an antipsychotic drug candidate, shows a high affinity for the D3 (Ki: 0.085 nM) and D2 (Ki: 0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM).
    Formula:C20H30Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.38

    Ref: TM-T15100

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • 4-Hydroxyatomoxetine

    CAS:
    4-Hydroxyatomoxetine, an active metabolite of Atomoxetine, is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.
    Formula:C17H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:271.35

    Ref: TM-T10145

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Anti-GLP1R Antibody


    <p>Anti-GLP1R Antibody is a human antibody expressed in CHO cells, targeting GLP1R. For isotype controls, refer to Human IgG1 kappa, Isotype Control.</p>
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-804

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • Picumeterol

    CAS:
    Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in vivo trials, Picumeterol produced long-lasting airway smooth muscle relaxation. Picumeterol is a pure R enantiomer that can be used to improve lung function and reduce airway hyperreactivity in patients with asthma.
    Formula:C21H29Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.38

    Ref: TM-T68129

    ne
    Discontinued
    Discontinued product
  • TAK-448

    CAS:
    TAK-448 (MVT-602), a potent KISS1R agonist, IC50: 460 pM, EC50: 632 pM, trialed for Prostate Cancer and Hypogonadism.
    Formula:C58H80N16O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1225.36

    Ref: TM-TP1094

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • Canagliflozin-d4

    CAS:
    <p>Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.</p>
    Formula:C24H25FO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.54

    Ref: TM-T10669

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    Discontinued product
  • 2-Methyl-5-HT hydrochloride

    CAS:
    2-Methyl-5-HT hydrochloride (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.
    Formula:C11H15ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:226.7

    Ref: TM-T10075L2

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • RU 24969 succinate

    CAS:
    <p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>
    Formula:C18H22N2O5
    Color and Shape:Solid
    Molecular weight:346.38

    Ref: TM-T71502

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Pamoic acid

    CAS:
    <p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>
    Formula:C23H16O6
    Purity:99.99%
    Color and Shape:Fine Yellow Powder
    Molecular weight:388.37

    Ref: TM-T8353

    1g
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • Flumexadol

    CAS:
    Flumexadol is a selective 5-HT2C receptor agonist with an affinity (Ki) of 25 nM for the (+)-enantiomer and exhibits 40-fold selectivity over the 5-HT2A receptor. It is an orally active, non-narcotic analgesic.
    Formula:C11H12F3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:231.21

    Ref: TM-T11302

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • GR 218,231

    CAS:
    GR 218,231 is a selective antagonist of D3 dopamine receptor.
    Formula:C24H33NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.59

    Ref: TM-T27431

    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • Imetit dihydrobromide

    CAS:
    Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors (Ki: 0.3 and 2.7 nM). Imetit mimics the histamine effect in triggering a shape change in eosinophils (EC50: 25 nM).
    Formula:C6H12Br2N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.06

    Ref: TM-T15565

    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product
  • MEN11467

    CAS:
    MEN11467 is a novel, orally available, potent and selective peptidomimetic tachykinin NK 1 receptor antagonist for the study of acute colon cancer.
    Formula:C38H40N4O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:600.75

    Ref: TM-T12000

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • Neurokinin antagonist 1

    CAS:
    Neurokinin antagonist 1 is a potent is a neuropeptide antagonist that can be used to study neurological disorders.
    Formula:C38H40N4O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:600.75

    Ref: TM-T10056

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • SB251023

    CAS:
    SB251023 is an agonist of β3-adrenoceptor.
    Formula:C28H34NO6P
    Color and Shape:Solid
    Molecular weight:511.55

    Ref: TM-T28687

    25mg
    Discontinued
    Discontinued product
  • S1P1 agonist 6

    CAS:
    <p>Compound I (S1P1 agonist 6) is an S1P1 agonist that mitigates autoimmune activity by inhibiting lymphocyte trafficking and has potential as an immunosuppressive</p>
    Formula:C25H26F3NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.47

    Ref: TM-T79816

    ne
    Discontinued
    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • AEF0117

    CAS:
    <p>AEF0117 is a signaling inhibitor of CB1-SSi that inhibits cannabinoid self-administration and can be used to study cannabis withdrawal.</p>
    Formula:C29H40O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:436.63

    Ref: TM-T79909

    ne
    Discontinued
    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • 2-MNG

    CAS:
    <p>2-MNG (2-Mercaptonicotinoyl glycine) is a novel melanogenesis inhibitor. 2-MNG inhibits two mechanisms of UV-induced skin pigmentation in vivo.</p>
    Formula:C8H8N2O3S
    Color and Shape:Liquid
    Molecular weight:212.23

    Ref: TM-T89029

    1mg
    Discontinued
    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    1mL*10mM (DMSO)
    Discontinued
    Discontinued product
  • Dimethandrolone Undecanoate

    CAS:
    Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.
    Formula:C31H50O3
    Purity:99.65% - >99.99%
    Color and Shape:Solid
    Molecular weight:470.73

    Ref: TM-T27176

    1mg
    Discontinued
    5mg
    Discontinued
    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    Discontinued product