GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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3-Hydroxy agomelatine D3
CAS:3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).Formula:C15H17NO3Purity:98%Color and Shape:SolidMolecular weight:262.32YNT-185 dihydrochloride
CAS:Potent OX2 agonist (EC50=28nM); 100x selective over OX1; prompts wakefulness, counters cataplexy in mice.Formula:C33H39Cl2N5O5SColor and Shape:SolidMolecular weight:688.67GSK682753A
CAS:GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2; IC50: 53.6 nM).Formula:C23H21Cl3N2O3Color and Shape:SolidMolecular weight:479.78Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formula:C19H23NO8Purity:99.79%Color and Shape:SolidMolecular weight:393.39LY223982
CAS:LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.Formula:C30H30O7Purity:99.86%Color and Shape:SolidMolecular weight:502.56SB-200646A
CAS:SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.Formula:C15H15ClN4OPurity:98%Color and Shape:SolidMolecular weight:302.76Sumanirole maleate
CAS:Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formula:C15H17N3O5Purity:98%Color and Shape:SolidMolecular weight:319.31Ozagrel Sodium
CAS:Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases.Formula:C13H12N2NaO2Purity:98%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:251.24Nefazodone
CAS:Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formula:C25H32ClN5O2Purity:99.85%Color and Shape:White To Off-White Crystalline PowderMolecular weight:470.01Ref: TM-T21451
2mg42.00€5mg60.00€10mg87.00€25mg177.00€50mg276.00€100mg422.00€200mg604.00€1mL*10mM (DMSO)95.00€S26131
CAS:S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormula:C31H34N2O4Purity:99.77%Color and Shape:SolidMolecular weight:498.61Terazosin
CAS:Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.Formula:C19H25N5O4Color and Shape:SolidMolecular weight:387.43MK-2894 sodium salt
CAS:MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.Formula:C25H22F3NNaO3SPurity:98%Color and Shape:SolidMolecular weight:496.5Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Formula:C61H93N19O15SPurity:99.68% - 99.90%Color and Shape:SolidMolecular weight:1364.57Ref: TM-T22344
1mg66.00€2mg92.00€5mg177.00€10mg281.00€25mg475.00€50mg677.00€100mg888.00€1mL*10mM (DMSO)355.00€[Sar9,Met(O2)11]-Substance P
CAS:[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.Formula:C64H100N18O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1393.66Veralipride
CAS:Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formula:C17H25N3O5SPurity:99.65%Color and Shape:SolidMolecular weight:383.46Zuclopenthixol dihydrochloride
CAS:Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Formula:C22H27Cl3N2OSPurity:98%Color and Shape:SolidMolecular weight:473.89Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formula:C32H51F3N8O9Purity:99.88%Color and Shape:SolidMolecular weight:748.79GLP-1 receptor agonist 9
CAS:1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.Formula:C32H31ClFN3O5Purity:98%Color and Shape:SolidMolecular weight:592.06Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFormula:C28H33ClN2·2HClPurity:98.05%Color and Shape:Off-White PowderMolecular weight:505.95Tiprenolol
CAS:Tiprenolol is a beta adrenergic receptor antagonist.[1]Formula:C13H21NO2SPurity:99.43%Color and Shape:SolidMolecular weight:255.38Ref: TM-T50081
1mg52.00€5mg98.00€10mg146.00€25mg235.00€50mg319.00€100mg447.00€200mg587.00€1mL*10mM (DMSO)89.00€
![[Sar9,Met(O2)11]-Substance P](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT7828.webp&w=3840&q=75)
