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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5965 products of "GPCR/G-Protein"

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  • Alimemazine hemitartrate

    CAS:
    Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.
    Formula:C18H22N2SC4H6O6
    Purity:98.16% - 99.69%
    Color and Shape:Solid
    Molecular weight:448.53
  • CCR2 antagonist 4 hydrochloride

    CAS:
    CCR2 antagonist 4 hydrochloride is a specific CCR2 antagonist (IC50s: 180 nM for CCR2b). It potently inhibits MCP-1-induced chemotaxis (IC50: 24 nM).
    Formula:C21H22Cl2F3N3O2
    Color and Shape:Solid
    Molecular weight:476.32
  • CAY10444

    CAS:
    CAY10444 is an S1P3 specific antagonist.
    Formula:C15H29NO2S
    Purity:99.15% - 99.61%
    Color and Shape:Solid
    Molecular weight:287.46
  • CYM-5520

    CAS:
    CYM-5520 is a noncompetitive allosteric agonist of S1P2
    Formula:C21H19N3O2
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:345.39
  • ML 10302

    CAS:
    ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.
    Formula:C15H21ClN2O3
    Color and Shape:Solid
    Molecular weight:312.79
  • N-Cbz-DL-tryptophan

    CAS:
    N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
    Formula:C19H18N2O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:338.36
  • Samelisant dihydrochloride

    CAS:
    SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.
    Formula:C21H33Cl2N3O3
    Color and Shape:Solid
    Molecular weight:446.41
  • Galnon TFA

    CAS:
    Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).
    Formula:C42H47F3N4O8
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:792.84
  • CRT0273750

    CAS:
    CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.
    Formula:C25H22ClF3N4O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:502.92
  • Picotamide

    CAS:
    Picotamide has anticoagulant and fibrinolytic properties.
    Formula:C21H20N4O3
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:376.41
  • Bevantolol

    CAS:
    Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].
    Formula:C20H27NO4
    Color and Shape:Solid
    Molecular weight:345.43
  • Lodoxamide

    CAS:
    <p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>
    Formula:C11H6ClN3O6
    Purity:99.13% - 99.81%
    Color and Shape:Solid
    Molecular weight:311.63
  • Benorilate

    CAS:
    Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.
    Formula:C17H15NO5
    Purity:98.39% - 99.85%
    Color and Shape:Solid
    Molecular weight:313.3
  • NPS ALX Compound 4a

    CAS:
    NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)
    Formula:C25H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.55
  • Carbazochrome

    CAS:
    Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.
    Formula:C10H12N4O3
    Purity:98.36%
    Color and Shape:Nacarat Crystalline Powder
    Molecular weight:236.23
  • Quipazine maleate

    CAS:
    Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.
    Formula:C17H19N3O4
    Color and Shape:Solid
    Molecular weight:329.356
  • Olcegepant

    CAS:
    Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4
    Formula:C38H47Br2N9O5
    Purity:96.08% - 97.24%
    Color and Shape:Solid
    Molecular weight:869.65
  • Sigma-LIGAND-1 hydrochloride

    CAS:
    Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.
    Formula:C27H34ClNO4
    Color and Shape:Solid
    Molecular weight:472.02
  • Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Formula:C22H28FNO3
    Purity:98.94% - 99.95%
    Color and Shape:Solid
    Molecular weight:373.46
  • Enprofylline

    CAS:
    Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.
    Formula:C8H10N4O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:194.19