
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(441 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5965 products of "GPCR/G-Protein"
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Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53CCR2 antagonist 4 hydrochloride
CAS:CCR2 antagonist 4 hydrochloride is a specific CCR2 antagonist (IC50s: 180 nM for CCR2b). It potently inhibits MCP-1-induced chemotaxis (IC50: 24 nM).Formula:C21H22Cl2F3N3O2Color and Shape:SolidMolecular weight:476.32CAY10444
CAS:CAY10444 is an S1P3 specific antagonist.Formula:C15H29NO2SPurity:99.15% - 99.61%Color and Shape:SolidMolecular weight:287.46CYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79N-Cbz-DL-tryptophan
CAS:N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formula:C19H18N2O4Purity:99.97%Color and Shape:SolidMolecular weight:338.36Samelisant dihydrochloride
CAS:SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.Formula:C21H33Cl2N3O3Color and Shape:SolidMolecular weight:446.41Galnon TFA
CAS:Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).Formula:C42H47F3N4O8Purity:99.47%Color and Shape:SolidMolecular weight:792.84CRT0273750
CAS:CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formula:C25H22ClF3N4O2Purity:99.91%Color and Shape:SolidMolecular weight:502.92Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Bevantolol
CAS:Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purity:99.13% - 99.81%Color and Shape:SolidMolecular weight:311.63Benorilate
CAS:Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formula:C17H15NO5Purity:98.39% - 99.85%Color and Shape:SolidMolecular weight:313.3NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:431.55Carbazochrome
CAS:Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.Formula:C10H12N4O3Purity:98.36%Color and Shape:Nacarat Crystalline PowderMolecular weight:236.23Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formula:C17H19N3O4Color and Shape:SolidMolecular weight:329.356Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Sigma-LIGAND-1 hydrochloride
CAS:Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19
