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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5965 products of "GPCR/G-Protein"

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  • Sigma-LIGAND-1 hydrochloride

    CAS:
    Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.
    Formula:C27H34ClNO4
    Color and Shape:Solid
    Molecular weight:472.02
  • Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Formula:C22H28FNO3
    Purity:98.94% - 99.95%
    Color and Shape:Solid
    Molecular weight:373.46
  • Enprofylline

    CAS:
    Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.
    Formula:C8H10N4O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:194.19
  • Niaprazine

    CAS:
    <p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>
    Formula:C20H25FN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:356.44
  • Rimcazole dihydrochloride

    CAS:
    Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.
    Formula:C21H28ClN3
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:357.92
  • γ-L-Glutamyl-L-alanine

    CAS:
    γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).
    Formula:C8H14N2O5
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:218.21
  • Tavapadon

    CAS:
    Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.
    Formula:C19H16F3N3O3
    Purity:99.33% - 99.8%
    Color and Shape:Solid
    Molecular weight:391.34
  • Piboserod hydrochloride

    CAS:
    Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.
    Formula:C22H32ClN3O2
    Color and Shape:Solid
    Molecular weight:405.96
  • YIL781 hydrochloride

    CAS:
    YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).
    Formula:C24H29ClFN3O2
    Color and Shape:Solid
    Molecular weight:445.96
  • Cyclopiazonic acid

    CAS:
    Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.
    Formula:C20H20N2O3
    Purity:99.27% - 99.80%
    Color and Shape:Solid
    Molecular weight:336.38
  • SB756050

    CAS:
    SB756050 is a specific TGR5 agonist.
    Formula:C21H28N2O8S2
    Purity:98.78% - >99.99%
    Color and Shape:Solid
    Molecular weight:500.59
  • ML-193

    CAS:
    ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
    Formula:C28H25N5O4S
    Purity:97.74%
    Color and Shape:Solid
    Molecular weight:527.59
  • Dolasetron Mesylate hydrate

    CAS:
    Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
    Formula:C20H26N2O7S
    Purity:99.86% - 99.99%
    Color and Shape:Solid
    Molecular weight:438.49
  • BMY-25368

    CAS:
    BMY-25368 is a long-acting antagonist of the H2-receptor.
    Formula:C19H25N3O3
    Color and Shape:Solid
    Molecular weight:343.42
  • Fertirelin

    CAS:
    Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).
    Formula:C55H76N16O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1153.29
  • Bretylium tosylate

    CAS:
    <p>Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.</p>
    Formula:C18H24BrNO3S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:414.36
  • Guanethidine monosulfate

    CAS:
    Guanethidine monosulfate is an antihypertensive drug that reduces the release of catecholamines.
    Formula:C10H24N4O4S
    Purity:99.61% - 99.74%
    Color and Shape:Solid
    Molecular weight:296.39
  • SAX-187 hydrochloride

    CAS:
    WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.
    Formula:C15H14Cl2N4O2S2
    Color and Shape:Solid
    Molecular weight:417.33
  • Seltorexant hydrochloride

    CAS:
    Seltorexant hydrochloride is a selective, orally active and high-affinity antagonist of OX2R with pKi values of 8.0 and 8.1 for human and rat OX2R.
    Formula:C21H23ClFN7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.91
  • Ritanserin

    CAS:
    Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.
    Formula:C27H25F2N3OS
    Purity:99.77% - 99.89%
    Color and Shape:Solid
    Molecular weight:477.57