GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(441 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5965 products of "GPCR/G-Protein"
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Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Bevantolol
CAS:Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purity:99.13% - 99.81%Color and Shape:SolidMolecular weight:311.63Benorilate
CAS:Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formula:C17H15NO5Purity:98.39% - 99.85%Color and Shape:SolidMolecular weight:313.3NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:431.55Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formula:C17H19N3O4Color and Shape:SolidMolecular weight:329.356Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formula:C52H83N13O14Purity:99.86%Color and Shape:SolidMolecular weight:1114.29Sigma-LIGAND-1 hydrochloride
CAS:Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurity:99.56%Color and Shape:SolidMolecular weight:356.44Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Formula:C25H37NO4Purity:98% - >99.99%Color and Shape:Crystalline SolidMolecular weight:415.57Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formula:C25H27N3O2SPurity:99.06% - 99.96%Color and Shape:SolidMolecular weight:433.57γ-L-Glutamyl-L-alanine
CAS:γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).Formula:C8H14N2O5Purity:99.49%Color and Shape:SolidMolecular weight:218.21PF-04418948
CAS:<p>PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.</p>Formula:C23H20FNO5Purity:98.67% - 99.45%Color and Shape:SolidMolecular weight:409.41Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formula:C22H32ClN3O2Color and Shape:SolidMolecular weight:405.96Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formula:C18H22ClNOPurity:99.44% - 99.85%Color and Shape:SolidMolecular weight:303.83UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formula:C52H68N10O14S2Purity:99.78%Color and Shape:SolidMolecular weight:1121.29Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Formula:C29H33FN2O4Purity:98.77% - 99.93%Color and Shape:SolidMolecular weight:492.58Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formula:C51H70N10O12S2Purity:99.03% - 99.87%Color and Shape:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMolecular weight:1079.3Cyclopiazonic acid
CAS:Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Formula:C20H20N2O3Purity:99.27% - 99.80%Color and Shape:SolidMolecular weight:336.38
