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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5968 products of "GPCR/G-Protein"

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  • Fluoroclebopride

    CAS:
    Fluoroclebopride is a dopamine (DA) D2 receptor ligand.
    Formula:C20H23ClFN3O2
    Purity:99.68% - 99.91%
    Color and Shape:Solid
    Molecular weight:391.87

    Ref: TM-T3187

    1mg
    35.00€
    5mg
    74.00€
    10mg
    96.00€
    25mg
    159.00€
    50mg
    235.00€
    100mg
    376.00€
    500mg
    867.00€
    1mL*10mM (DMSO)
    96.00€
  • Carbazochrome

    CAS:
    Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.
    Formula:C10H12N4O3
    Purity:98.36%
    Color and Shape:Nacarat Crystalline Powder
    Molecular weight:236.23

    Ref: TM-T3616

    250mg
    49.00€
    500mg
    59.00€
  • Idazoxan hydrochloride

    CAS:
    Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
    Formula:C11H12N2O2·HCl
    Purity:99.42% - 99.84%
    Color and Shape:Solid
    Molecular weight:240.69

    Ref: TM-T0115

    2mg
    35.00€
    5mg
    52.00€
    10mg
    78.00€
    25mg
    133.00€
    50mg
    187.00€
    100mg
    281.00€
    200mg
    416.00€
    1mL*10mM (DMSO)
    50.00€
  • JK184

    CAS:
    <p>JK184 is a potent Hedgehog (Hh) pathway inhibitor.</p>
    Formula:C19H18N4OS
    Purity:98.93% - 99.89%
    Color and Shape:Solid
    Molecular weight:350.44

    Ref: TM-T3588

    5mg
    35.00€
    10mg
    50.00€
    25mg
    93.00€
    50mg
    160.00€
    100mg
    250.00€
    200mg
    359.00€
  • BMS-813160

    CAS:
    BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.
    Formula:C25H40N8O2
    Purity:99.66% - 99.79%
    Color and Shape:Solid
    Molecular weight:484.64

    Ref: TM-T4584

    1mg
    63.00€
    5mg
    137.00€
    10mg
    187.00€
    25mg
    341.00€
    50mg
    567.00€
    100mg
    810.00€
    500mg
    1,644.00€
    1mL*10mM (DMSO)
    145.00€
  • ML221

    CAS:
    ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in
    Formula:C17H11N3O6S
    Purity:97.74%
    Color and Shape:Solid
    Molecular weight:385.35

    Ref: TM-T4390

    2mg
    To inquire
    5mg
    52.00€
    10mg
    85.00€
    25mg
    144.00€
    50mg
    227.00€
    100mg
    369.00€
    200mg
    To inquire
    1mL*10mM (DMSO)
    55.00€
  • Hydroxyzine

    CAS:
    Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.
    Formula:C21H27ClN2O2
    Purity:99.54% - ≥95%
    Color and Shape:Oil Solid
    Molecular weight:374.9

    Ref: TM-T20884

    50mg
    43.00€
    1mL*10mM (DMSO)
    47.00€
  • GUANABENZ

    CAS:
    GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
    Formula:C8H8Cl2N4
    Purity:98.31%
    Color and Shape:White Solid From Acetonitrile Solid
    Molecular weight:231.08

    Ref: TM-T5471

    5mg
    42.00€
    10mg
    57.00€
    25mg
    92.00€
    50mg
    127.00€
    100mg
    180.00€
    200mg
    264.00€
    1mL*10mM (DMSO)
    48.00€
  • NPS ALX Compound 4a

    CAS:
    NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)
    Formula:C25H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.55

    Ref: TM-T12262

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Benorilate

    CAS:
    Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.
    Formula:C17H15NO5
    Purity:98.39% - 99.85%
    Color and Shape:Solid
    Molecular weight:313.3

    Ref: TM-T3276

    1g
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • Decloxizine dihydrochloride

    CAS:
    <p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>
    Formula:C21H28N2O2·2ClH
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:413.39

    Ref: TM-T5495

    25mg
    50.00€
    50mg
    74.00€
    100mg
    97.00€
    200mg
    160.00€
  • Lodoxamide

    CAS:
    <p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>
    Formula:C11H6ClN3O6
    Purity:99.13% - 99.81%
    Color and Shape:Solid
    Molecular weight:311.63

    Ref: TM-T4566

    5mg
    47.00€
    10mg
    60.00€
    25mg
    94.00€
    50mg
    111.00€
    100mg
    187.00€
    200mg
    325.00€
  • Bevantolol

    CAS:
    Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].
    Formula:C20H27NO4
    Color and Shape:Solid
    Molecular weight:345.43

    Ref: TM-T61138

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • SB-200646

    CAS:
    SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
    Formula:C15H14N4O
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:266.3

    Ref: TM-T8357

    1mg
    65.00€
    5mg
    129.00€
    10mg
    187.00€
    25mg
    315.00€
    50mg
    454.00€
    100mg
    620.00€
    1mL*10mM (DMSO)
    135.00€
  • Bepotastine

    CAS:
    Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.
    Formula:C21H25ClN2O3
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:388.89

    Ref: TM-T7893

    2mg
    37.00€
    5mg
    52.00€
    10mg
    82.00€
    25mg
    149.00€
    50mg
    216.00€
    100mg
    329.00€
    200mg
    490.00€
    1mL*10mM (DMSO)
    59.00€
  • 5-HT1A modulator 2 hydrochloride

    CAS:
    5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.
    Formula:C11H16ClNO
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:213.7

    Ref: TM-T37197

    25mg
    44.00€
    50mg
    56.00€
    1mL*10mM (DMSO)
    48.00€
  • Picotamide

    CAS:
    Picotamide has anticoagulant and fibrinolytic properties.
    Formula:C21H20N4O3
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:376.41

    Ref: TM-T9153

    1mg
    40.00€
    5mg
    97.00€
    10mg
    156.00€
    25mg
    255.00€
    50mg
    368.00€
    100mg
    505.00€
    200mg
    692.00€
    1mL*10mM (DMSO)
    99.00€
  • Exo1

    CAS:
    Exo1 is an inhibitor of the exocytic pathway
    Formula:C15H12FNO3
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:273.26

    Ref: TM-T4609

    10mg
    46.00€
    25mg
    86.00€
    50mg
    137.00€
    100mg
    187.00€
    1mL*10mM (DMSO)
    34.00€
  • Fenspiride

    CAS:
    Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.
    Formula:C15H20N2O2
    Color and Shape:Solid
    Molecular weight:260.33

    Ref: TM-T60417

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CRT0273750

    CAS:
    CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.
    Formula:C25H22ClF3N4O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:502.92

    Ref: TM-T31101

    1mg
    35.00€
    5mg
    78.00€
    10mg
    114.00€
    25mg
    226.00€
    50mg
    339.00€
    100mg
    509.00€
    1mL*10mM (DMSO)
    85.00€