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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • SSR240612
    Targetmol
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    SSR240612

    CAS:
    <p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>
    Formula:C42H53ClN4O7S
    Purity:98.59% - 99.16%
    Color and Shape:Solid
    Molecular weight:793.41

    Ref: TM-T5048

  • Cimetidine hydrochloride
    Targetmol
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    Cimetidine hydrochloride

    CAS:
    <p>Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.</p>
    Formula:C10H17ClN6S
    Color and Shape:Solid
    Molecular weight:288.8

    Ref: TM-T60584

  • AM966
    Targetmol
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    AM966

    CAS:
    <p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>
    Formula:C27H23ClN2O5
    Purity:98.06% - 99.79%
    Color and Shape:Solid
    Molecular weight:490.93

    Ref: TM-T4278

  • SB 242084 dihydrochloride
    Targetmol
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    SB 242084 dihydrochloride

    CAS:
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.
    Formula:C21H21Cl3N4O2
    Color and Shape:Solid
    Molecular weight:467.78

    Ref: TM-T37114

  • Veralipride
    Targetmol
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    Veralipride

    CAS:
    <p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>
    Formula:C17H25N3O5S
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:383.46

    Ref: TM-T7632

  • Canagliflozin
    Targetmol
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    Canagliflozin

    CAS:
    <p>Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.</p>
    Formula:C24H25FO5S
    Purity:98.01% - >99.99%
    Color and Shape:Solid
    Molecular weight:444.52

    Ref: TM-T1782

  • AVN-101
    Targetmol
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    AVN-101

    CAS:
    <p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>
    Formula:C21H25ClN2
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:340.89

    Ref: TM-T26690

  • ML-18
    Targetmol
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    ML-18

    CAS:
    <p>ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.</p>
    Formula:C32H35N5O5
    Purity:98.62% - >99.99%
    Color and Shape:Solid
    Molecular weight:569.65

    Ref: TM-T4540

  • Conopressin S acetate(111317-90-9 free base)
    Targetmol
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    Conopressin S acetate(111317-90-9 free base)

    <p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>
    Formula:C43H77N17O12S2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:1088.32

    Ref: TM-TP1192L

  • Methyldopa hydrate
    Targetmol
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    Methyldopa hydrate

    CAS:
    <p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>
    Formula:C10H13NO4H2O
    Purity:99.67%
    Color and Shape:White Solid
    Molecular weight:238.24

    Ref: TM-T5954

  • Avexitide
    Targetmol
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    Avexitide

    CAS:
    <p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>
    Formula:C149H234N40O47S
    Purity:98% - 99.65%
    Color and Shape:Solid
    Molecular weight:3369.76

    Ref: TM-TP2100

  • GSK189254A
    Targetmol
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    GSK189254A

    CAS:
    <p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>
    Formula:C21H25N3O2
    Purity:98.71% - 99.858%
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-TQ0066

  • [Sar9,Met(O2)11]-Substance P
    Targetmol
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    [Sar9,Met(O2)11]-Substance P

    CAS:
    [Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
    Formula:C64H100N18O15S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1393.66

    Ref: TM-T7828

  • CHEMBL241987
    Targetmol
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    CHEMBL241987

    CAS:
    <p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>
    Formula:C16H11N3O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:261.28

    Ref: TM-T8598

  • Eledoisin Related Peptide 2TFA
    Targetmol
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    Eledoisin Related Peptide 2TFA

    Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.
    Formula:C38H60F6N8O10S
    Purity:99%
    Color and Shape:Solid
    Molecular weight:934.99

    Ref: TM-T7631L

  • Cinacalcet
    Targetmol
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    Cinacalcet

    CAS:
    <p>Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .</p>
    Formula:C22H22F3N
    Purity:99.48%
    Color and Shape:Yellow Oil
    Molecular weight:357.41

    Ref: TM-T8403

  • 3-AQC
    Targetmol
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    3-AQC

    CAS:
    <p>3-AQC is a competitive antagonist of 5-HT3.</p>
    Formula:C20H21N5O4
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:395.41

    Ref: TM-T8475

  • IPSU
    Targetmol
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    IPSU

    CAS:
    <p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>
    Formula:C23H27N5O2
    Purity:97.05%
    Color and Shape:Solid
    Molecular weight:405.49

    Ref: TM-T5503

  • Men 10376 TFA(135306-85-3,free)
    Targetmol
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    Men 10376 TFA(135306-85-3,free)

    <p>Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4</p>
    Formula:C59H69F3N12O12
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:1195.25

    Ref: TM-TP1086

  • JNJ-37822681
    Targetmol
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    JNJ-37822681

    CAS:
    <p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>
    Formula:C17H17F5N4
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:372.34

    Ref: TM-T27677