CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Tianeptine sodium salt
    Targetmol
    + Info

    Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>
    Formula:C21H24ClN2NaO4S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:458.93

    Ref: TM-T2402

  • SAG hydrochloride (912545-86-9(free base))
    Targetmol
    + Info

    SAG hydrochloride (912545-86-9(free base))

    CAS:
    <p>SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.</p>
    Formula:C28H29Cl2N3OS
    Purity:99.19% - 99.77%
    Color and Shape:Solid
    Molecular weight:526.52

    Ref: TM-T4211

  • R243
    Targetmol
    + Info

    R243

    CAS:
    <p>R243 is CCR8 signaling and chemotaxis inhibitor.</p>
    Formula:C21H27NO4
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:357.44

    Ref: TM-T24700

  • Brimonidine
    Targetmol
    + Info

    Brimonidine

    CAS:
    <p>Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and Alphagan-P.</p>
    Formula:C11H10BrN5
    Purity:99.626%
    Color and Shape:Yellow Solid
    Molecular weight:292.13

    Ref: TM-T20157

  • Temanogrel
    Targetmol
    + Info

    Temanogrel

    CAS:
    <p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>
    Formula:C24H28N4O4
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:436.5

    Ref: TM-T17033

  • Sonidegib
    Targetmol
    + Info

    Sonidegib

    CAS:
    <p>Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.</p>
    Formula:C26H26F3N3O3
    Purity:98% - 99.97%
    Color and Shape:Solid
    Molecular weight:485.5

    Ref: TM-T1926

  • Salmeterol Xinafoate
    Targetmol
    + Info

    Salmeterol Xinafoate

    CAS:
    <p>Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.</p>
    Formula:C36H45NO7
    Purity:98% - 98.24%
    Color and Shape:White Solid
    Molecular weight:603.75

    Ref: TM-T6653

  • MRT-81
    Targetmol
    + Info

    MRT-81

    CAS:
    <p>MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.</p>
    Formula:C31H29N3O5S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:555.64

    Ref: TM-T9532

  • ARN272
    Targetmol
    + Info

    ARN272

    CAS:
    <p>ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).</p>
    Formula:C27H20N4O2
    Purity:98.23%
    Color and Shape:Solid
    Molecular weight:432.47

    Ref: TM-T5357

  • BA 1 acetate(183241-31-8 free base)
    Targetmol
    + Info

    BA 1 acetate(183241-31-8 free base)

    <p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>
    Formula:C59H80N14O13
    Purity:95.3%
    Color and Shape:Solid
    Molecular weight:1193.35

    Ref: TM-TP1913L1

  • Pranlukast hemihydrate
    Targetmol
    + Info

    Pranlukast hemihydrate

    CAS:
    <p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>
    Formula:C27H23N5O40·5H2O
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:490.52

    Ref: TM-T63291

  • 5'-N-Ethylcarboxamidoadenosine
    Targetmol
    + Info

    5'-N-Ethylcarboxamidoadenosine

    CAS:
    <p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>
    Formula:C12H16N6O4
    Purity:98.95% - ≥95%
    Color and Shape:Powder
    Molecular weight:308.29

    Ref: TM-T7340

  • 9-FLUORENOL
    Targetmol
    + Info

    9-FLUORENOL

    CAS:
    <p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>
    Formula:C13H10O
    Purity:99.98%
    Color and Shape:Off-White Crystalline Powder
    Molecular weight:182.22

    Ref: TM-T8633

  • Ebastine
    Targetmol
    + Info

    Ebastine

    CAS:
    <p>Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.</p>
    Formula:C32H39NO2
    Purity:99.65% - 99.93%
    Color and Shape:White To Off-White Powder
    Molecular weight:469.66

    Ref: TM-T2335

  • Ocaperidone
    Targetmol
    + Info

    Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Formula:C24H25FN4O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T3497

  • Chlorcyclizine
    Targetmol
    + Info

    Chlorcyclizine

    CAS:
    <p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>
    Formula:C18H21ClN2
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:300.83

    Ref: TM-T9717

  • Regadenoson
    Targetmol
    + Info

    Regadenoson

    CAS:
    <p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>
    Formula:C15H18N8O5
    Purity:99.57% - 99.81%
    Color and Shape:Off-White Solid
    Molecular weight:390.35

    Ref: TM-T2671

  • Orexin B, rat, mouse Acetate
    Targetmol
    + Info

    Orexin B, rat, mouse Acetate

    Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.
    Formula:C128H219N45O36S
    Purity:94.61%
    Color and Shape:Solid
    Molecular weight:2996.45

    Ref: TM-TP1045L

  • S1RA hydrochloride
    Targetmol
    + Info

    S1RA hydrochloride

    CAS:
    <p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki &gt;</p>
    Formula:C20H24ClN3O2
    Purity:98% - 99.84%
    Color and Shape:Solid
    Molecular weight:373.87

    Ref: TM-T4229

  • AM095
    Targetmol
    + Info

    AM095

    CAS:
    AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.
    Formula:C27H23N2NaO5
    Purity:98.87%
    Color and Shape:Solid
    Molecular weight:478.47

    Ref: TM-T2000