GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83MRT-81
CAS:MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formula:C31H29N3O5SPurity:99.72%Color and Shape:SolidMolecular weight:555.64Ref: TM-T9532
1mg48.00€5mg97.00€10mg145.00€25mg255.00€50mg368.00€100mg505.00€200mg692.00€1mL*10mM (DMSO)116.00€BD-1047 dihydrobromide
CAS:BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormula:C13H22Br2Cl2N2Purity:98.13% - 99.39%Color and Shape:SolidMolecular weight:437.04Ref: TM-T1740
1mg37.00€2mg48.00€5mg73.00€10mg95.00€25mg168.00€50mg290.00€100mg490.00€1mL*10mM (DMSO)74.00€Spiperone hydrochloride
CAS:5-HT2A serotonin and selective D2-like dopamine receptor antagonistFormula:C23H27ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:431.93Brimonidine Tartrate
CAS:Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).Formula:C15H16BrN5O6Purity:99.95%Color and Shape:Off-White Crystalline SolidMolecular weight:442.22BRL-15572 dihydrochloride
CAS:BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formula:C25H27ClN2O·2HClPurity:99.74%Color and Shape:SolidMolecular weight:479.87Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.Formula:C63H93N15O20SPurity:98.11%Color and Shape:SolidMolecular weight:1412.57TY-52156
CAS:TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).Formula:C18H19Cl2N3OPurity:99.91% - 99.91%Color and Shape:SolidMolecular weight:364.27Ref: TM-T17183
2mg40.00€5mg60.00€10mg87.00€25mg166.00€50mg298.00€100mg510.00€200mg683.00€1mL*10mM (DMSO)66.00€HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purity:99.51%Color and Shape:SolidMolecular weight:614.57Fabomotizole
CAS:Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.Formula:C15H21N3O2SPurity:99.4%Color and Shape:SolidMolecular weight:307.41Sitaxsentan sodium
CAS:Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.Formula:C18H14ClN2O6S2·NaPurity:98.39% - 99.01%Color and Shape:SolidMolecular weight:476.89Treprostinil
CAS:<p>Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).</p>Formula:C23H34O5Purity:99.29%Color and Shape:SolidMolecular weight:390.51Riociguat
CAS:Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth muscle and is used to treat severe pulmonary arterialFormula:C20H19FN8O2Purity:99.28% - 99.95%Color and Shape:SolidMolecular weight:422.42Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Formula:C12H16ClN3O2Purity:98.95% - 99.13%Color and Shape:SolidMolecular weight:269.73Binodenoson
CAS:Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.Formula:C17H25N7O4Purity:99.74%Color and Shape:SolidMolecular weight:391.42Ref: TM-T9516
1mg99.00€5mg235.00€10mg354.00€25mg588.00€50mg787.00€100mg1,103.00€1mL*10mM (DMSO)259.00€Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Color and Shape:SolidMolecular weight:858.34Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purity:99.15% - 99.82%Color and Shape:SolidMolecular weight:292.38LIXIVAPTAN
CAS:Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formula:C27H21ClFN3O2Purity:98.36%Color and Shape:SolidMolecular weight:473.93Ref: TM-T7303
2mg37.00€5mg70.00€10mg104.00€25mg216.00€50mg354.00€100mg550.00€200mg785.00€1mL*10mM (DMSO)73.00€
