
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(444 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47Ref: TM-T8666
1mg42.00€2mg52.00€5mg77.00€10mg97.00€25mg170.00€50mg254.00€100mg380.00€1mL*10mM (DMSO)93.00€Taminadenant mesylate
CAS:Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formula:C11H12BrN7O3SColor and Shape:SolidMolecular weight:402.227Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Color and Shape:SolidMolecular weight:491.49Selexipag
CAS:Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.Formula:C26H32N4O4SPurity:99.98% - >99.99%Color and Shape:SolidMolecular weight:496.62CID 1375606
CAS:CID 1375606: Surrogate agonist for GPR27, conserved in vertebrates, mainly in CNS.Formula:C20H14Cl2N2O2Purity:99.41%Color and Shape:SolidMolecular weight:385.24Substance P (7-11)
CAS:Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .Formula:C31H44N6O5SPurity:98.39%Color and Shape:SolidMolecular weight:612.78Ataciguat
CAS:Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.Formula:C21H19Cl2N3O6S3Purity:99.09%Color and Shape:SolidMolecular weight:576.49Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Formula:C16H26N2O2Purity:99.52%Color and Shape:SolidMolecular weight:278.39GSK2018682 HCl
CAS:GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formula:C22H22Cl2N4O4Color and Shape:SolidMolecular weight:477.34Arformoterol Tartrate
CAS:Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49Ref: TM-T22245
5mg60.00€10mg87.00€25mg150.00€50mg221.00€100mg329.00€200mg487.00€1mL*10mM (DMSO)85.00€Landiolol hydrochloride
CAS:Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formula:C25H34N4O2·C4H4O4Purity:98.44% - 99.46%Color and Shape:SolidMolecular weight:538.64Ref: TM-T2631
2mg46.00€5mg66.00€10mg95.00€25mg180.00€50mg334.00€100mg495.00€200mg717.00€500mg1,111.00€1mL*10mM (DMSO)79.00€MCL0020
CAS:MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.Formula:C34H39N7O4Purity:99.18%Color and Shape:SolidMolecular weight:609.72BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg88.00€5mg170.00€10mg248.00€25mg444.00€50mg638.00€100mg889.00€200mg1,198.00€1mL*10mM (DMSO)182.00€Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purity:98% - 99.9%Color and Shape:SolidMolecular weight:5218.88Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurity:94.61%Color and Shape:SolidMolecular weight:2996.45Capadenoson
CAS:Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.Formula:C25H18ClN5O2S2Purity:98.85% - 99.57%Color and Shape:SolidMolecular weight:520.03SCH 58261
CAS:SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formula:C18H15N7OPurity:99.07% - 99.75%Color and Shape:SolidMolecular weight:345.36Ref: TM-T6979
1mg40.00€2mg51.00€5mg85.00€10mg125.00€25mg225.00€50mg364.00€100mg582.00€1mL*10mM (DMSO)86.00€Piboserod
CAS:Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formula:C22H31N3O2Purity:97.21% - 99.49%Color and Shape:SolidMolecular weight:369.5Ref: TM-T2278
1mg40.00€2mg52.00€5mg88.00€10mg125.00€25mg233.00€50mg424.00€100mg613.00€500mg1,264.00€1mL*10mM (DMSO)127.00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57
