GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5981 products of "GPCR/G-Protein"
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Talnetant hydrochloride
CAS:Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.Formula:C25H23ClN2O2Color and Shape:SolidMolecular weight:418.92Norfluoxetine Hydrochloride
CAS:Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.Formula:C16H17ClF3NOPurity:99.71%Color and Shape:SolidMolecular weight:331.76PGS-IN-1
CAS:PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formula:C19H26O3Purity:99.39%Color and Shape:SolidMolecular weight:302.41Ref: TM-T10098
1mg52.00€5mg97.00€10mg170.00€25mg369.00€50mg540.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)110.00€N-Cbz-DL-tryptophan
CAS:N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.Formula:C19H18N2O4Purity:99.97%Color and Shape:SolidMolecular weight:338.36BMS-986020
CAS:BMS-986020 (AM152) is a selective antagonist of LPA1.Formula:C29H26N2O5Purity:98.82% - >99.99%Color and Shape:SolidMolecular weight:482.53Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.Formula:C91H143N27O26S4Purity:99.41%Color and Shape:SolidMolecular weight:2157Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purity:97.84% - 99.90%Color and Shape:SolidMolecular weight:575.61Samelisant dihydrochloride
CAS:SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.Formula:C21H33Cl2N3O3Color and Shape:SolidMolecular weight:446.41OS-3-106
CAS:OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.Formula:C25H30N4O2SPurity:99.4% - 99.57%Color and Shape:SolidMolecular weight:450.6Aprocitentan
CAS:Aprocitentan (ACT-132577) is ETA and ETB antagonist .Formula:C16H14Br2N6O4SPurity:99.17%Color and Shape:SolidMolecular weight:546.19Ref: TM-T7817
1mg58.00€5mg116.00€10mg170.00€25mg311.00€50mg439.00€100mg655.00€200mg887.00€1mL*10mM (DMSO)142.00€Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formula:C13H13ClN2OPurity:99.61% - >99.99%Color and Shape:Yellow To Slightly Green Crystalline PowderMolecular weight:248.71HJC0350
CAS:HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of Epac1.Formula:C15H19NO2SPurity:99.27% - 99.65%Color and Shape:SolidMolecular weight:277.38Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Formula:C14H16N2OPurity:97.38%Color and Shape:SolidMolecular weight:228.29Cinaciguat
CAS:<p>Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.</p>Formula:C36H39NO5Purity:98% - 99.18%Color and Shape:SolidMolecular weight:565.7Neuropeptide FF acetate(99566-27-5 free base)
<p>Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family.</p>Formula:C56H80N14O12Purity:98.03%Color and Shape:SolidMolecular weight:1141.32PF-4136309
CAS:PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formula:C29H31F3N6O3Purity:98.85% - 99.47%Color and Shape:SolidMolecular weight:568.59Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Formula:C5H11Cl2N3Purity:99.12%Color and Shape:SolidMolecular weight:184.067Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4Formula:C59H69F3N12O12Purity:99.22%Color and Shape:SolidMolecular weight:1195.25Donitriptan Mesylate
CAS:Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formula:C24H29N5O5SColor and Shape:SolidMolecular weight:499.58
