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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5984 products of "GPCR/G-Protein"

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  • RS102895

    CAS:
    RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.
    Formula:C21H21F3N2O2
    Purity:97.64% - 99.80%
    Color and Shape:Solid
    Molecular weight:390.4

    Ref: TM-TQ0283

    2mg
    42.00€
    5mg
    62.00€
    10mg
    90.00€
    25mg
    166.00€
    50mg
    241.00€
    100mg
    359.00€
    1mL*10mM (DMSO)
    69.00€
  • AR-M 1896 Acetate


    AR-M 1896 Acetate is the selective agonist of GalR2.
    Formula:C56H85N13O16
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:1196.35

    Ref: TM-T21646L

    1mg
    537.00€
    2mg
    727.00€
    5mg
    1,064.00€
    10mg
    1,454.00€
    25mg
    2,147.00€
    50mg
    2,822.00€
    1mL*10mM (DMSO)
    2,213.00€
  • ICI 89406

    CAS:
    ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.
    Formula:C19H22N4O3
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:354.4

    Ref: TM-T22852

    1mg
    69.00€
    5mg
    138.00€
    10mg
    190.00€
    25mg
    359.00€
    50mg
    525.00€
    1mL*10mM (DMSO)
    145.00€
  • GLP-1(7-36), amide

    CAS:
    GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.
    Formula:C149H226N40O45
    Purity:99.85%
    Color and Shape:White Powder
    Molecular weight:3297.63

    Ref: TM-T3984

    1mg
    172.00€
    2mg
    294.00€
    5mg
    497.00€
    10mg
    713.00€
    25mg
    1,099.00€
    50mg
    1,468.00€
    100mg
    1,998.00€
  • Melperone

    CAS:
    Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.
    Formula:C16H22FNO
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:263.35

    Ref: TM-T7421

    25mg
    48.00€
    50mg
    64.00€
    100mg
    111.00€
    200mg
    164.00€
    1mL*10mM (DMSO)
    34.00€
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Formula:C19H26ClNOS
    Purity:99.53% - 99.56%
    Color and Shape:Almost White To White Crystalline Powder
    Molecular weight:351.93

    Ref: TM-T21446

    5mg
    44.00€
    10mg
    59.00€
    25mg
    96.00€
    50mg
    116.00€
    100mg
    159.00€
    200mg
    227.00€
  • Xamoterol

    CAS:
    Xamoterol is a cardiac stimulant.
    Formula:C16H25N3O5
    Color and Shape:Solid
    Molecular weight:339.39

    Ref: TM-T35153

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Cinitapride

    CAS:
    Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.
    Formula:C21H30N4O4
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:402.49

    Ref: TM-T21385

    1mg
    73.00€
    5mg
    155.00€
    10mg
    240.00€
    25mg
    479.00€
    50mg
    692.00€
    100mg
    973.00€
    1mL*10mM (DMSO)
    177.00€
  • Syk Inhibitor II dihydrochloride dihydrate

    CAS:
    Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.
    Formula:C14H21Cl2F3N6O3
    Color and Shape:Solid
    Molecular weight:449.26

    Ref: TM-T62691

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Formula:C24H40NaO4
    Purity:99.66% - 99.96%
    Color and Shape:Solid
    Molecular weight:415.56

    Ref: TM-T29078

    100mg
    34.00€
  • Bilastine

    CAS:
    Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of
    Formula:C28H37N3O3
    Purity:99.86% - >99.99%
    Color and Shape:Solid
    Molecular weight:463.61

    Ref: TM-T4250

    25mg
    44.00€
    50mg
    66.00€
    100mg
    98.00€
    500mg
    219.00€
    1mL*10mM (DMSO)
    44.00€
  • Atrasentan sodium

    CAS:
    Atrasentan (ABT-627) is an oral ETA receptor blocker with potential cancer-fighting properties, inhibiting angiogenesis and tumor growth.
    Formula:C29H37N2NaO6
    Color and Shape:Solid
    Molecular weight:532.61

    Ref: TM-T70198

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • LY2828360

    CAS:
    LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.
    Formula:C22H27ClN6O
    Purity:98.45% - 99.51%
    Color and Shape:Solid
    Molecular weight:426.94

    Ref: TM-T7316

    2mg
    35.00€
    5mg
    49.00€
    10mg
    80.00€
    25mg
    137.00€
    50mg
    192.00€
    100mg
    281.00€
    200mg
    419.00€
  • carfenazine

    CAS:
    <p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>
    Formula:C24H31N3O2S
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:425.59

    Ref: TM-T9827

    1mg
    92.00€
    5mg
    183.00€
    10mg
    274.00€
    25mg
    472.00€
    50mg
    To inquire
  • GW842166X

    CAS:
    GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.
    Formula:C18H17Cl2F3N4O2
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:449.25

    Ref: TM-T6527

    5mg
    49.00€
    10mg
    82.00€
    25mg
    138.00€
    50mg
    197.00€
    100mg
    278.00€
    200mg
    396.00€
    1mL*10mM (DMSO)
    48.00€
  • GLP-1(7-37) acetate(106612-94-6 free base)

    CAS:
    Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
    Formula:C151H228N40O47
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:3355.67

    Ref: TM-TP1376

    1mg
    97.00€
    5mg
    216.00€
    10mg
    329.00€
    25mg
    560.00€
    50mg
    800.00€
    100mg
    1,103.00€
    200mg
    1,483.00€
  • Lidamidine Hydrochloride

    CAS:
    Lidamidine HCl: α2-adrenergic agonist; lowers gut secretion, slows transit, stops muscle contractions.
    Formula:C11H17ClN4O
    Color and Shape:Solid
    Molecular weight:256.73

    Ref: TM-T27829

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Dobutamine hydrochloride

    CAS:
    <p>Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.</p>
    Formula:C18H24ClNO3
    Purity:97.15% - 99.94%
    Color and Shape:Solid
    Molecular weight:337.84

    Ref: TM-T8149

    25mg
    52.00€
    50mg
    74.00€
    100mg
    96.00€
    500mg
    221.00€
  • NNC-0640

    CAS:
    NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
    Formula:C29H31N7O4S
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:573.67

    Ref: TM-T7364

    1mg
    48.00€
    2mg
    65.00€
    5mg
    96.00€
    10mg
    169.00€
    25mg
    298.00€
    50mg
    454.00€
    100mg
    655.00€
    1mL*10mM (DMSO)
    96.00€
  • PF-06882961 Tris

    CAS:
    PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C35H41FN6O7
    Purity:98.74% - 99.79%
    Color and Shape:Solid
    Molecular weight:676.7

    Ref: TM-T8876

    1mg
    131.00€
    5mg
    286.00€
    10mg
    430.00€
    25mg
    710.00€
    50mg
    998.00€
    100mg
    1,349.00€
    500mg
    2,688.00€