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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5984 products of "GPCR/G-Protein"

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  • Naratriptan

    CAS:
    Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.
    Formula:C17H25N3O2S
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:335.47

    Ref: TM-T8666

    1mg
    42.00€
    2mg
    52.00€
    5mg
    77.00€
    10mg
    97.00€
    25mg
    170.00€
    50mg
    254.00€
    100mg
    380.00€
    1mL*10mM (DMSO)
    93.00€
  • Taminadenant mesylate

    CAS:
    Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.
    Formula:C11H12BrN7O3S
    Color and Shape:Solid
    Molecular weight:402.227

    Ref: TM-T69723

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Valbenazine dihydrochloride

    CAS:
    Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.
    Formula:C24H40Cl2N2O4
    Color and Shape:Solid
    Molecular weight:491.49

    Ref: TM-T70322

    25mg
    2,727.00€
    50mg
    3,591.00€
    100mg
    4,940.00€
  • Selexipag

    CAS:
    Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.
    Formula:C26H32N4O4S
    Purity:99.98% - >99.99%
    Color and Shape:Solid
    Molecular weight:496.62

    Ref: TM-T3216

    5mg
    49.00€
    10mg
    64.00€
    25mg
    92.00€
    50mg
    96.00€
    1mL*10mM (DMSO)
    50.00€
  • CID 1375606

    CAS:
    CID 1375606: Surrogate agonist for GPR27, conserved in vertebrates, mainly in CNS.
    Formula:C20H14Cl2N2O2
    Purity:99.41%
    Color and Shape:Solid
    Molecular weight:385.24

    Ref: TM-T5422

    2mg
    35.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    144.00€
    50mg
    235.00€
    100mg
    349.00€
    1mL*10mM (DMSO)
    52.00€
  • Substance P (7-11)

    CAS:
    Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
    Formula:C31H44N6O5S
    Purity:98.39%
    Color and Shape:Solid
    Molecular weight:612.78

    Ref: TM-T7554

    2mg
    47.00€
    5mg
    70.00€
    10mg
    111.00€
    25mg
    178.00€
    50mg
    269.00€
    100mg
    370.00€
  • Ataciguat

    CAS:
    Ataciguat (HMR-1766) (HMR-1766) is a potent and specific soluble guanylate cyclase (sGC) activator.
    Formula:C21H19Cl2N3O6S3
    Purity:99.09%
    Color and Shape:Solid
    Molecular weight:576.49

    Ref: TM-T21607

    1mg
    52.00€
    5mg
    88.00€
    10mg
    144.00€
    25mg
    283.00€
    50mg
    406.00€
    100mg
    562.00€
    1mL*10mM (DMSO)
    117.00€
  • Dimethocaine

    CAS:
    Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.
    Formula:C16H26N2O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:278.39

    Ref: TM-T7118

    1g
    123.00€
    100mg
    48.00€
    500mg
    93.00€
    1mL*10mM (DMSO)
    34.00€
  • GSK2018682 HCl

    CAS:
    GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.
    Formula:C22H22Cl2N4O4
    Color and Shape:Solid
    Molecular weight:477.34

    Ref: TM-T71564

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Arformoterol Tartrate

    CAS:
    Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.
    Formula:C23H30N2O10
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:494.49

    Ref: TM-T22245

    5mg
    60.00€
    10mg
    87.00€
    25mg
    150.00€
    50mg
    221.00€
    100mg
    329.00€
    200mg
    487.00€
    1mL*10mM (DMSO)
    85.00€
  • Landiolol hydrochloride

    CAS:
    Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
    Formula:C25H40ClN3O8
    Purity:99.91%
    Color and Shape:White Crystalline Powder
    Molecular weight:546.05

    Ref: TM-T5028

    5mg
    35.00€
    10mg
    48.00€
    25mg
    80.00€
    50mg
    104.00€
    100mg
    144.00€
    200mg
    207.00€
    1mL*10mM (DMSO)
    52.00€
  • WAY-100635 Monomaleate

    CAS:
    WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.
    Formula:C25H34N4O2·C4H4O4
    Purity:98.44% - 99.46%
    Color and Shape:Solid
    Molecular weight:538.64

    Ref: TM-T2631

    2mg
    46.00€
    5mg
    66.00€
    10mg
    95.00€
    25mg
    180.00€
    50mg
    334.00€
    100mg
    495.00€
    200mg
    717.00€
    500mg
    1,111.00€
    1mL*10mM (DMSO)
    79.00€
  • MCL0020

    CAS:
    MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.
    Formula:C34H39N7O4
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:609.72

    Ref: TM-TP1889

    1mg
    110.00€
    5mg
    269.00€
    10mg
    371.00€
    25mg
    572.00€
    50mg
    783.00€
    100mg
    1,035.00€
    200mg
    1,404.00€
  • BAY-545

    CAS:
    BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).
    Formula:C18H22F3N3O4S
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:433.45

    Ref: TM-T8512

    1mg
    88.00€
    5mg
    170.00€
    10mg
    248.00€
    25mg
    444.00€
    50mg
    638.00€
    100mg
    889.00€
    200mg
    1,198.00€
    1mL*10mM (DMSO)
    182.00€
  • Lixisenatide acetate (320367-13-3 free base)

    CAS:
    <p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>
    Formula:C215H347N61O65S·6C2H4O2
    Purity:98% - 99.9%
    Color and Shape:Solid
    Molecular weight:5218.88

    Ref: TM-TP1469

    1mg
    64.00€
    5mg
    116.00€
    10mg
    183.00€
    25mg
    306.00€
    50mg
    439.00€
    100mg
    598.00€
    200mg
    805.00€
  • Orexin B, rat, mouse Acetate


    Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.
    Formula:C128H219N45O36S
    Purity:94.61%
    Color and Shape:Solid
    Molecular weight:2996.45

    Ref: TM-TP1045L

    1mg
    128.00€
    5mg
    300.00€
    10mg
    423.00€
    25mg
    627.00€
    50mg
    845.00€
    100mg
    1,130.00€
    200mg
    1,520.00€
  • Capadenoson

    CAS:
    Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
    Formula:C25H18ClN5O2S2
    Purity:98.85% - 99.57%
    Color and Shape:Solid
    Molecular weight:520.03

    Ref: TM-TQ0125

    5mg
    34.00€
    10mg
    44.00€
    50mg
    107.00€
    1mL*10mM (DMSO)
    34.00€
  • SCH 58261

    CAS:
    SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.
    Formula:C18H15N7O
    Purity:99.07% - 99.75%
    Color and Shape:Solid
    Molecular weight:345.36

    Ref: TM-T6979

    1mg
    40.00€
    2mg
    51.00€
    5mg
    85.00€
    10mg
    125.00€
    25mg
    225.00€
    50mg
    364.00€
    100mg
    582.00€
    1mL*10mM (DMSO)
    86.00€
  • Piboserod

    CAS:
    Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.
    Formula:C22H31N3O2
    Purity:97.21% - 99.49%
    Color and Shape:Solid
    Molecular weight:369.5

    Ref: TM-T2278

    1mg
    40.00€
    2mg
    52.00€
    5mg
    88.00€
    10mg
    125.00€
    25mg
    233.00€
    50mg
    424.00€
    100mg
    613.00€
    500mg
    1,264.00€
    1mL*10mM (DMSO)
    127.00€
  • Perospirone

    CAS:
    Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
    Formula:C23H30N4O2S
    Purity:99.23%
    Color and Shape:White Powder
    Molecular weight:426.57

    Ref: TM-T4576

    10mg
    48.00€
    25mg
    82.00€
    50mg
    133.00€
    100mg
    221.00€
    200mg
    309.00€
    1mL*10mM (DMSO)
    34.00€