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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5963 products of "GPCR/G-Protein"

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  • Thrombin Receptor Activator for Peptide


    Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.
    Formula:C32H51F3N8O9
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:748.79

    Ref: TM-T7674

    1mg
    47.00€
    5mg
    90.00€
    10mg
    145.00€
    25mg
    258.00€
    50mg
    373.00€
    100mg
    535.00€
    200mg
    728.00€
  • PAR-2 Activating Peptide acetate


    PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
    Formula:C31H60N10O9
    Purity:98.5% - 99.92%
    Color and Shape:Solid
    Molecular weight:716.88

    Ref: TM-TP1046L

    1mg
    81.00€
    5mg
    185.00€
    10mg
    330.00€
    25mg
    557.00€
    50mg
    792.00€
    100mg
    1,071.00€
    200mg
    1,431.00€
  • Gadolinium chloride

    CAS:
    Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
    Formula:Cl3Gd
    Purity:98%
    Color and Shape:White Crystalline Solid
    Molecular weight:263.61

    Ref: TM-T22795

    25mg
    48.00€
    50mg
    58.00€
    100mg
    89.00€
    200mg
    126.00€
  • Paltusotine

    CAS:
    Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.
    Formula:C27H22F2N4O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:456.49

    Ref: TM-T9692

    1mg
    166.00€
    5mg
    401.00€
    10mg
    580.00€
    25mg
    879.00€
    50mg
    1,189.00€
    100mg
    1,603.00€
  • Ozanimod

    CAS:
    Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.
    Formula:C23H24N4O3
    Purity:98.68% - 99.58%
    Color and Shape:Solid
    Molecular weight:404.46

    Ref: TM-T6923

    1mg
    46.00€
    5mg
    90.00€
    10mg
    137.00€
    25mg
    268.00€
    50mg
    430.00€
    100mg
    622.00€
    200mg
    879.00€
    500mg
    1,305.00€
    1mL*10mM (DMSO)
    90.00€
  • Desvenlafaxine succinate hydrate

    CAS:
    Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
    Formula:C20H33NO7
    Purity:99.26%
    Color and Shape:White Crystalline Powde
    Molecular weight:399.48

    Ref: TM-T6188

    1g
    99.00€
    2g
    146.00€
    50mg
    34.00€
    100mg
    46.00€
    500mg
    80.00€
    1mL*10mM (DMSO)
    34.00€
  • Adenosine receptor antagonist 4

    CAS:
    Adenosine receptor antagonist 4 is an adenosine receptor antagonist.
    Formula:C10H13N3
    Purity:99.63% - 99.65%
    Color and Shape:Off-White Powder
    Molecular weight:175.23

    Ref: TM-T21620

    1g
    213.00€
    50mg
    46.00€
    100mg
    71.00€
    500mg
    147.00€
    1mL*10mM (DMSO)
    33.00€
  • Ablukast

    CAS:
    Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.
    Formula:C28H34O8
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:498.56

    Ref: TM-T26519

    2mg
    43.00€
    5mg
    73.00€
    10mg
    105.00€
    25mg
    200.00€
    50mg
    281.00€
    100mg
    383.00€
    1mL*10mM (DMSO)
    80.00€
  • Serotonin hydrochloride

    CAS:
    Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (
    Formula:C10H13ClN2O
    Purity:98.05% - 99.93%
    Color and Shape:White To Cream Powder
    Molecular weight:212.676

    Ref: TM-T2209

    25mg
    35.00€
    50mg
    49.00€
    100mg
    57.00€
    200mg
    79.00€
    1mL*10mM (DMSO)
    51.00€
  • ONO-AE3-208

    CAS:

    ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.

    Formula:C24H21FN2O3
    Purity:98.04% - 99.55%
    Color and Shape:Solid
    Molecular weight:404.43

    Ref: TM-TQ0290

    2mg
    42.00€
    5mg
    64.00€
    10mg
    92.00€
    25mg
    157.00€
    50mg
    224.00€
    100mg
    To inquire
  • Alizapride hydrochloride

    CAS:
    Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.
    Formula:C16H21N5O2·HCl
    Purity:99.35% - 99.48%
    Color and Shape:Coa
    Molecular weight:351.83

    Ref: TM-T2574

    25mg
    34.00€
    50mg
    46.00€
    100mg
    66.00€
    500mg
    144.00€
    1mL*10mM (DMSO)
    44.00€
  • CYM2503

    CAS:

    CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.

    Formula:C45H55N5O7
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:777.95

    Ref: TM-T8963

    1mg
    37.00€
    5mg
    80.00€
    10mg
    116.00€
    25mg
    226.00€
    50mg
    363.00€
    100mg
    512.00€
    200mg
    697.00€
  • SB399885

    CAS:
    SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.
    Formula:C18H21Cl2N3O4S
    Purity:98.94%
    Color and Shape:Solid
    Molecular weight:446.35

    Ref: TM-T19669

    1mg
    67.00€
    5mg
    123.00€
    10mg
    177.00€
    25mg
    291.00€
    50mg
    393.00€
    100mg
    553.00€
    200mg
    743.00€
    1mL*10mM (DMSO)
    150.00€
  • HTMT dimaleate

    CAS:
    HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
    Formula:C27H33F3N4O9
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:614.57

    Ref: TM-T22842

    1mg
    35.00€
    5mg
    87.00€
    10mg
    133.00€
    25mg
    216.00€
  • Etrasimod

    CAS:
    Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).
    Formula:C26H26F3NO3
    Purity:98.52% - 99.73%
    Color and Shape:Solid
    Molecular weight:457.48

    Ref: TM-TQ0227

    1mg
    50.00€
    5mg
    105.00€
    10mg
    170.00€
    25mg
    230.00€
    50mg
    289.00€
    100mg
    401.00€
    1mL*10mM (DMSO)
    107.00€
  • JNJ-10229570

    CAS:
    JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous gland
    Formula:C22H19N3O2S
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:389.47

    Ref: TM-T5464

    1mg
    104.00€
    5mg
    178.00€
    10mg
    281.00€
    25mg
    447.00€
    50mg
    620.00€
    100mg
    802.00€
    1mL*10mM (DMSO)
    203.00€
  • ENMD-1068 HBr

    CAS:
    ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.
    Formula:C15H30BrN3O2
    Color and Shape:Solid
    Molecular weight:364.32

    Ref: TM-T24028

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NGB 2904

    CAS:
    NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).
    Formula:C28H29Cl2N3O
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:494.46

    Ref: TM-T28167

    2mg
    38.00€
    5mg
    55.00€
    10mg
    86.00€
    25mg
    155.00€
    50mg
    264.00€
    100mg
    374.00€
    500mg
    To inquire
    1mL*10mM (DMSO)
    72.00€
  • Hemokinin 1 (mouse) acetate(208041-90-1 free base)


    Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.
    Formula:C63H104N22O17S
    Purity:98.33%
    Color and Shape:Solid
    Molecular weight:1473.72

    Ref: TM-TP1772L

    1mg
    89.00€
    5mg
    222.00€
    10mg
    331.00€
    25mg
    527.00€
    50mg
    712.00€
    100mg
    954.00€
  • MHP

    CAS:
    MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.
    Formula:C16H23NO4
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:293.36

    Ref: TM-T4658

    1mg
    34.00€
    2mg
    46.00€
    5mg
    66.00€
    10mg
    101.00€
    25mg
    207.00€
    50mg
    334.00€
    100mg
    537.00€
    200mg
    762.00€
    1mL*10mM (DMSO)
    73.00€