
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formula:C32H51F3N8O9Purity:99.88%Color and Shape:SolidMolecular weight:748.79PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.88Gadolinium chloride
CAS:Gadolinium chloride is a calcium-sensing receptor (CaSR) agonistFormula:Cl3GdPurity:98%Color and Shape:White Crystalline SolidMolecular weight:263.61Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formula:C27H22F2N4OPurity:99.91%Color and Shape:SolidMolecular weight:456.49Ozanimod
CAS:Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.Formula:C23H24N4O3Purity:98.68% - 99.58%Color and Shape:SolidMolecular weight:404.46Ref: TM-T6923
1mg46.00€5mg90.00€10mg137.00€25mg268.00€50mg430.00€100mg622.00€200mg879.00€500mg1,305.00€1mL*10mM (DMSO)90.00€Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Formula:C20H33NO7Purity:99.26%Color and Shape:White Crystalline PowdeMolecular weight:399.48Adenosine receptor antagonist 4
CAS:Adenosine receptor antagonist 4 is an adenosine receptor antagonist.Formula:C10H13N3Purity:99.63% - 99.65%Color and Shape:Off-White PowderMolecular weight:175.23Ablukast
CAS:Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formula:C28H34O8Purity:98.58%Color and Shape:SolidMolecular weight:498.56Serotonin hydrochloride
CAS:Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (Formula:C10H13ClN2OPurity:98.05% - 99.93%Color and Shape:White To Cream PowderMolecular weight:212.676ONO-AE3-208
CAS:ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of prostate cancer.
Formula:C24H21FN2O3Purity:98.04% - 99.55%Color and Shape:SolidMolecular weight:404.43Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Formula:C16H21N5O2·HClPurity:99.35% - 99.48%Color and Shape:CoaMolecular weight:351.83CYM2503
CAS:CYM2503 is a GAL2 receptor PAM enhancing galanin-induced IP1 without binding the galanin site.
Formula:C45H55N5O7Purity:97.04%Color and Shape:SolidMolecular weight:777.95SB399885
CAS:SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formula:C18H21Cl2N3O4SPurity:98.94%Color and Shape:SolidMolecular weight:446.35Ref: TM-T19669
1mg67.00€5mg123.00€10mg177.00€25mg291.00€50mg393.00€100mg553.00€200mg743.00€1mL*10mM (DMSO)150.00€HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formula:C27H33F3N4O9Purity:99.51%Color and Shape:SolidMolecular weight:614.57Etrasimod
CAS:Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).Formula:C26H26F3NO3Purity:98.52% - 99.73%Color and Shape:SolidMolecular weight:457.48Ref: TM-TQ0227
1mg50.00€5mg105.00€10mg170.00€25mg230.00€50mg289.00€100mg401.00€1mL*10mM (DMSO)107.00€JNJ-10229570
CAS:JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), which inhibits sebaceous glandFormula:C22H19N3O2SPurity:98.41%Color and Shape:SolidMolecular weight:389.47Ref: TM-T5464
1mg104.00€5mg178.00€10mg281.00€25mg447.00€50mg620.00€100mg802.00€1mL*10mM (DMSO)203.00€ENMD-1068 HBr
CAS:ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.Formula:C15H30BrN3O2Color and Shape:SolidMolecular weight:364.32NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formula:C28H29Cl2N3OPurity:98.79%Color and Shape:SolidMolecular weight:494.46Ref: TM-T28167
2mg38.00€5mg55.00€10mg86.00€25mg155.00€50mg264.00€100mg374.00€500mgTo inquire1mL*10mM (DMSO)72.00€Hemokinin 1 (mouse) acetate(208041-90-1 free base)
Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.Formula:C63H104N22O17SPurity:98.33%Color and Shape:SolidMolecular weight:1473.72MHP
CAS:MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.Formula:C16H23NO4Purity:98.58%Color and Shape:SolidMolecular weight:293.36Ref: TM-T4658
1mg34.00€2mg46.00€5mg66.00€10mg101.00€25mg207.00€50mg334.00€100mg537.00€200mg762.00€1mL*10mM (DMSO)73.00€
