GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Niaprazine
CAS:Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.Formula:C20H25FN4OPurity:99.56%Color and Shape:SolidMolecular weight:356.44SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formula:C17H18BrNOPurity:95.00% - 99.82%Color and Shape:SolidMolecular weight:332.23Bexagliflozin
CAS:Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values of 2 nM for human SGLT2.Formula:C24H29ClO7Purity:98.99% - 99.89%Color and Shape:SolidMolecular weight:464.94Ref: TM-T7217
1mg67.00€2mg95.00€5mg129.00€10mg187.00€25mg371.00€50mg552.00€100mg785.00€1mL*10mM (DMSO)137.00€Bosentan (hydrate)
CAS:Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A (ET-A) and endothelin-B (ET-B) receptors.Formula:C27H29N5O6S·H2OPurity:99.31% - 99.86%Color and Shape:White PowderMolecular weight:569.63Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Purity:98.42%Color and Shape:LiquidMolecular weight:N/ADobutamine tartrate
CAS:Dobutamine tartrate is a cardiotonic.Formula:C22H29NO9Color and Shape:SolidMolecular weight:451.472Enprofylline
CAS:Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Ref: TM-T21389
2mg42.00€5mg62.00€10mg88.00€25mg141.00€50mg215.00€100mg318.00€200mg442.00€1mL*10mM (DMSO)59.00€Fluorogestone acetate
CAS:FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.Formula:C23H31FO5Purity:99.47%Color and Shape:CoaMolecular weight:406.49Ref: TM-T21335
2mg44.00€5mg67.00€10mg96.00€25mg178.00€50mg261.00€100mg374.00€200mg494.00€1mL*10mM (DMSO)80.00€Scyliorhinin II acetate
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.Formula:C79H123N21O28S3Purity:99.06%Color and Shape:SolidMolecular weight:1911.14Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formula:C52H83N13O14Purity:99.86%Color and Shape:SolidMolecular weight:1114.29PAR-2-IN-1
CAS:PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
Formula:C12H14ClN3O2Purity:99.75%Color and Shape:SolidMolecular weight:267.71Vercirnon sodium
CAS:Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formula:C22H21ClN2NaO4SColor and Shape:SolidMolecular weight:467.92TNCA
CAS:TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.Formula:C12H12N2O2Purity:97.33% - 97.73%Color and Shape:SolidMolecular weight:216.24OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formula:C18H22N2O2SPurity:99.58%Color and Shape:SolidMolecular weight:330.44Pancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.Purity:97.53%Color and Shape:SolidMolecular weight:N/ARef: TM-TP1044L
1mg215.00€5mg510.00€10mg692.00€25mg1,009.00€50mg1,378.00€100mg1,863.00€200mg2,520.00€Valbenazine dihydrochloride
CAS:Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.Formula:C24H40Cl2N2O4Color and Shape:SolidMolecular weight:491.49[D-Trp8]-γ-MSH acetate(321351-81-9 free base)
[D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 andFormula:C76H103N21O18SPurity:99.75%Color and Shape:SolidMolecular weight:1630.82Phentolamine hydrochloride
CAS:Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].Formula:C17H20ClN3OColor and Shape:SolidMolecular weight:317.82Alcaftadine
CAS:Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.Formula:C19H21N3OPurity:98% - 98.65%Color and Shape:SolidMolecular weight:307.39Albiglutide TFA (782500-75-8 free base)
Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
Formula:C150H225F3N40O47Purity:>99.99%Color and Shape:SolidMolecular weight:3397.63
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