GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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GRA Ex-25
CAS:GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61RS102895
CAS:RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.Formula:C21H21F3N2O2Purity:97.64% - 99.80%Color and Shape:SolidMolecular weight:390.4Vercirnon
CAS:Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formula:C22H21ClN2O4SPurity:99.23%Color and Shape:SolidMolecular weight:444.93Ref: TM-T17225
1mg105.00€5mg259.00€10mg406.00€25mg680.00€50mg938.00€100mg1,301.00€500mg2,593.00€1mL*10mM (DMSO)363.00€Alprenolol hydrochloride
CAS:Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.Formula:C15H24ClNO2Purity:99.79%Color and Shape:SolidMolecular weight:285.81PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7Eprazinone
CAS:Erazinone is a mucus dissolver and bronchospasm reliever.Formula:C24H32N2O2Color and Shape:SolidMolecular weight:380.52BPTU
CAS:BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).Formula:C23H22F3N3O3Purity:99.37% - 99.89%Color and Shape:SolidMolecular weight:445.43Ref: TM-T4132
1mg35.00€2mg50.00€5mg69.00€10mg110.00€25mg225.00€50mg389.00€100mg577.00€1mL*10mM (DMSO)69.00€VUF10460
CAS:VUF10460 is a non-imidazole histamine H4 receptor agonist.Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.Formula:C59H80N14O13Purity:95.3%Color and Shape:SolidMolecular weight:1193.35BAY-545
CAS:BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).Formula:C18H22F3N3O4SPurity:98.05%Color and Shape:SolidMolecular weight:433.45Ref: TM-T8512
1mg84.00€5mg161.00€10mg235.00€25mg420.00€50mg605.00€100mg842.00€200mg1,134.00€1mL*10mM (DMSO)172.00€Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48NAV-2729
CAS:NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formula:C25H17ClN4O3Purity:98.83% - 98.91%Color and Shape:SolidMolecular weight:456.88Ref: TM-T5142
2mg43.00€5mg63.00€10mg90.00€25mg193.00€50mg286.00€100mg429.00€500mg888.00€1mL*10mM (DMSO)71.00€CAY10526
CAS:CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formula:C12H7BrO3SPurity:98.75%Color and Shape:SolidMolecular weight:311.15CHEMBL241987
CAS:CHEMBL241987 targets the Adenosine receptor A3 (human)Formula:C16H11N3OPurity:99.81%Color and Shape:SolidMolecular weight:261.28SB-203186 hydrochloride
CAS:SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFormula:C16H20N2O2·HClPurity:99.64%Color and Shape:SolidMolecular weight:308.81Human growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) onPurity:99.26%Color and Shape:LiquidMolecular weight:N/AVilazodone Hydrochloride
CAS:Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormula:C26H27N5O2·HClPurity:99.56% - >99.99%Color and Shape:SolidMolecular weight:477.99DORA-22
CAS:DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormula:C23H22F2N4O2Purity:97.67%Color and Shape:SolidMolecular weight:424.44Ref: TM-T5500
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)331.00€2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.Formula:C38H64F3N11O10Purity:>99.99%Color and Shape:SolidMolecular weight:891.98
