GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,003 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formula:C17H25N3O2SPurity:99.08%Color and Shape:SolidMolecular weight:335.47Ref: TM-T8666
1mg39.00€2mg50.00€5mg73.00€10mg92.00€25mg166.00€50mg240.00€100mg360.00€1mL*10mM (DMSO)88.00€α-MSH
CAS:α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of adenylyl cyclase.Formula:C77H109N21O19SPurity:99.10% - 99.67%Color and Shape:White PowderMolecular weight:1664.89Brimonidine Tartrate
CAS:Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).Formula:C15H16BrN5O6Purity:99.95%Color and Shape:Off-White Crystalline SolidMolecular weight:442.22ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.Formula:C60H94N16O15S2Purity:99.53%Color and Shape:SolidMolecular weight:1343.61Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Purity:98.27%Color and Shape:LiquidMolecular weight:N/AAntazoline
CAS:Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Tolazoline
CAS:Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formula:C10H12N2Purity:99.52%Color and Shape:SolidMolecular weight:160.22Naluzotan
CAS:Naluzotan（PRX 00023） is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+Formula:C23H38N4O3SPurity:>99.99%Color and Shape:SolidMolecular weight:450.64Secretin (33-59), rat
CAS:Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35Maropitant
CAS:Maropitant is a selective neurokinin (NK1) receptor antagonist.Formula:C32H40N2OPurity:97.35% - 99.75%Color and Shape:SolidMolecular weight:468.67Ref: TM-T7209
5mg50.00€10mg80.00€25mg116.00€50mg212.00€100mg316.00€200mg454.00€1mL*10mM (DMSO)To inquireOlcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purity:>99.99%Color and Shape:SolidMolecular weight:1024.18BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formula:C34H51N5NaO7Color and Shape:SolidMolecular weight:664.8Moxilubant
CAS:Moxilubant, a small molecule, blocks LTB4R to treat immune, skin, and joint disorders, may help in psoriasis and rheumatoid arthritis research.Formula:C26H37N3O4Purity:98%Color and Shape:SolidMolecular weight:455.59Cutamesine dihydrochloride
CAS:Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.Formula:C23H32N2O2·2HClPurity:99.96%Color and Shape:SolidMolecular weight:441.43Ref: TM-T3597
2mg34.00€5mg50.00€10mg86.00€25mg167.00€50mg260.00€100mg401.00€200mg580.00€1mL*10mM (DMSO)55.00€Cinaciguat
CAS:Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:C36H39NO5Purity:98% - 99.18%Color and Shape:SolidMolecular weight:565.7Ki16425
CAS:Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formula:C23H23ClN2O5SPurity:97.6% - 97.78%Color and Shape:SolidMolecular weight:474.96JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Formula:C27H27Cl2N5O3SPurity:99.54% - 99.84%Color and Shape:SolidMolecular weight:572.51Ref: TM-T4453
1mg42.00€2mg55.00€5mg90.00€10mg133.00€25mg234.00€50mg350.00€100mg522.00€1mL*10mM (DMSO)101.00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55Relenopride hydrochloride
CAS:Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.Formula:C24H31Cl2FN4O4Color and Shape:SolidMolecular weight:529.43
