GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formula:C23H31ClN4O2SPurity:99.37%Color and Shape:White SolidMolecular weight:463Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purity:99.70%Color and Shape:White To Off-White SolidMolecular weight:410.59SCH-37370
CAS:SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formula:C21H21ClN2OPurity:99.07%Color and Shape:SolidMolecular weight:352.86Ref: TM-T19686
1mg48.00€5mg89.00€10mg115.00€25mg195.00€50mg290.00€100mg393.00€200mg520.00€1mL*10mM (DMSO)90.00€Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formula:C76H103N15O28SPurity:99.35% - 99.82%Color and Shape:SolidMolecular weight:1706.78Terazosin hydrochloride dihydrate
CAS:Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92RE-640
CAS:NSC-5844 (RE-640) (RE640) is a bisquinoline compound with C-C chemokine receptor type 1 (CCR1)-agonistic activities.Formula:C20H16Cl2N4Purity:99.60% - 99.87%Color and Shape:SolidMolecular weight:383.27Serotonin
CAS:Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!
Formula:C10H12N2OPurity:97.47% - 99.92%Color and Shape:SolidMolecular weight:176.22Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formula:C17H19N3O4Color and Shape:SolidMolecular weight:329.356Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32Empagliflozin
CAS:Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with more than 300-fold selectivity for SGLT-1/4/5/6.Formula:C23H27ClO7Purity:98% - 99.98%Color and Shape:SolidMolecular weight:450.91Ref: TM-T1766
1g278.00€5mg47.00€10mg60.00€50mg79.00€100mg96.00€200mg144.00€500mg188.00€1mL*10mM (DMSO)50.00€JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Formula:C20H32N2OPurity:97.19%Color and Shape:SolidMolecular weight:316.48Melatonin
CAS:Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formula:C13H16N2O2Purity:98% - 99.89%Color and Shape:Pale Yellow Leaflets From Benzene SolidMolecular weight:232.28Ufenamate
CAS:Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseasesFormula:C18H18F3NO2Purity:99.89%Color and Shape:SolidMolecular weight:337.34Verucerfont
CAS:Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .Formula:C22H26N6O2Purity:99.90%Color and Shape:SolidMolecular weight:406.48Ref: TM-T7361
1mg60.00€2mg87.00€5mg130.00€10mg205.00€25mg376.00€50mg573.00€100mg803.00€1mL*10mM (DMSO)142.00€Pramlintide acetate(151126-32-8 free base)
CAS:Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.Formula:C173H271N51O55S2Purity:>99.99%Color and Shape:SolidMolecular weight:4009Levalbuterol tartrate
CAS:Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.Formula:C17H27NO9Purity:99.28% - 99.98%Color and Shape:SolidMolecular weight:389.39Ref: TM-T7164
2mg34.00€5mg50.00€10mg88.00€25mg100.00€50mg124.00€100mg177.00€200mg259.00€1mL*10mM (DMSO)60.00€ML-SI3
CAS:CCG-143140 is a GLP-1 receptor inverse agonists.Formula:C23H31N3O3SPurity:99.75%Color and Shape:SolidMolecular weight:429.58tcY-NH2 TFA(327177-34-4 free base)
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formula:C42H50F3N7O9Purity:>99.99%Color and Shape:SolidMolecular weight:853.9Fosaprepitant dimeglumine
CAS:Fosaprepitant dimeglumine (MK-0517) is a soluble prodrug of aprepitant, which prevents nausea by blocking NK1 receptors.
Formula:C37H56F7N6O16PPurity:98% - 99.03%Color and Shape:SolidMolecular weight:1004.83PD-168077 maleate
CAS:PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formula:C24H26N4O5Purity:99.13%Color and Shape:SolidMolecular weight:450.49Ref: TM-T5047
2mg35.00€5mg52.00€10mg80.00€25mg150.00€50mg245.00€100mg364.00€200mg517.00€1mL*10mM (DMSO)58.00€
