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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5957 products of "GPCR/G-Protein"

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  • AZD2098

    CAS:
    AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.
    Formula:C11H9Cl2N3O3S
    Purity:99.80% - >99.99%
    Color and Shape:Solid
    Molecular weight:334.18

    Ref: TM-T4300

    1mg
    34.00€
    5mg
    66.00€
    10mg
    105.00€
    25mg
    217.00€
    50mg
    334.00€
    100mg
    502.00€
    500mg
    1,063.00€
    1mL*10mM (DMSO)
    73.00€
  • C-021

    CAS:
    C 021 dihydrochloride is a potent CCR4 antagonist.
    Formula:C27H41N5O2
    Purity:99.74% - 99.90%
    Color and Shape:Solid
    Molecular weight:467.65

    Ref: TM-T21870

    1mg
    51.00€
    2mg
    71.00€
    5mg
    96.00€
    10mg
    153.00€
    25mg
    303.00€
    50mg
    469.00€
    100mg
    655.00€
    1mL*10mM (DMSO)
    96.00€
  • Nitrobenzylthioinosine

    CAS:

    Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.

    Formula:C17H17N5O6S
    Purity:99.69% - 99.74%
    Color and Shape:Off-White Solid
    Molecular weight:419.41

    Ref: TM-T8551

    5mg
    48.00€
    10mg
    66.00€
    25mg
    125.00€
    50mg
    188.00€
    100mg
    283.00€
    200mg
    434.00€
  • Chlorprothixene

    CAS:
    Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
    Formula:C18H18ClNS
    Purity:98.77% - 99.756%
    Color and Shape:Pale Yellow Crystals Solid
    Molecular weight:315.86

    Ref: TM-T0074

    1g
    133.00€
    100mg
    34.00€
    200mg
    50.00€
    500mg
    92.00€
  • CCG215022

    CAS:
    CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.
    Formula:C26H22FN7O3
    Purity:97.63% - 99.69%
    Color and Shape:Solid
    Molecular weight:499.5

    Ref: TM-T3498

    1mg
    56.00€
    5mg
    114.00€
    10mg
    178.00€
    25mg
    394.00€
    50mg
    655.00€
    100mg
    1,035.00€
    1mL*10mM (DMSO)
    127.00€
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Formula:C19H21Cl2N3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:362.3

    Ref: TM-T1822L

    5mg
    34.00€
    10mg
    50.00€
    25mg
    92.00€
    50mg
    147.00€
    100mg
    222.00€
    1mL*10mM (DMSO)
    39.00€
  • Vicriviroc maleate

    CAS:

    Vicriviroc maleate (SCH-417690 (maleate))(Sch-417690) is a piperazine-based CCR5 receptor antagonist with activity against human immunodeficiency virus.

    Formula:C32H42F3N5O6
    Purity:98.16% - 98.37%
    Color and Shape:Solid
    Molecular weight:649.7

    Ref: TM-T3435

    1mg
    42.00€
    5mg
    94.00€
    10mg
    131.00€
    25mg
    225.00€
    50mg
    339.00€
    100mg
    509.00€
  • JK184

    CAS:

    JK184 is a potent Hedgehog (Hh) pathway inhibitor.

    Formula:C19H18N4OS
    Purity:98.93% - 99.89%
    Color and Shape:Solid
    Molecular weight:350.44

    Ref: TM-T3588

    5mg
    35.00€
    10mg
    50.00€
    25mg
    93.00€
    50mg
    160.00€
    100mg
    250.00€
    200mg
    359.00€
  • AZD-4818

    CAS:
    AZD-4818 (CCR1 antagonist) is a chemokine CCR1 antagonist for the treatment of chronic obstructive pulmonary disease.
    Formula:C27H32Cl2N2O7
    Purity:99.01%
    Color and Shape:Solid
    Molecular weight:567.46

    Ref: TM-T30258

    1mg
    44.00€
    2mg
    62.00€
    5mg
    92.00€
    10mg
    147.00€
    25mg
    285.00€
    50mg
    429.00€
    100mg
    642.00€
    200mg
    865.00€
  • Maraviroc

    CAS:
    Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.
    Formula:C29H41F2N5O
    Purity:97.13% - 99.59%
    Color and Shape:Brown Solid
    Molecular weight:513.67

    Ref: TM-T6016

    5mg
    51.00€
    10mg
    95.00€
    25mg
    160.00€
    50mg
    273.00€
    100mg
    492.00€
    200mg
    633.00€
    500mg
    998.00€
    1mL*10mM (DMSO)
    59.00€
  • Cenicriviroc

    CAS:
    Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.
    Formula:C41H52N4O4S
    Purity:97.87%
    Color and Shape:Solid
    Molecular weight:696.94

    Ref: TM-TQ0297

    1mg
    63.00€
    2mg
    90.00€
    5mg
    133.00€
    10mg
    212.00€
    25mg
    423.00€
    50mg
    550.00€
    100mg
    715.00€
    200mg
    964.00€
    1mL*10mM (DMSO)
    200.00€
  • SAG hydrochloride (912545-86-9(free base))

    CAS:
    SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.
    Formula:C28H29Cl2N3OS
    Purity:99.19% - 99.97%
    Color and Shape:Solid
    Molecular weight:526.52

    Ref: TM-T4211

    1mg
    49.00€
    2mg
    65.00€
    5mg
    90.00€
    10mg
    114.00€
    25mg
    222.00€
    50mg
    334.00€
    100mg
    502.00€
    200mg
    717.00€
    1mL*10mM (DMSO)
    105.00€
  • R243

    CAS:
    R243 is CCR8 signaling and chemotaxis inhibitor.
    Formula:C21H27NO4
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:357.44

    Ref: TM-T24700

    1mg
    40.00€
    2mg
    52.00€
    5mg
    80.00€
    10mg
    117.00€
    25mg
    207.00€
    50mg
    333.00€
    100mg
    495.00€
    1mL*10mM (DMSO)
    90.00€
  • Sonidegib

    CAS:
    Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.
    Formula:C26H26F3N3O3
    Purity:98% - 99.97%
    Color and Shape:Solid
    Molecular weight:485.5

    Ref: TM-T1926

    5mg
    59.00€
    10mg
    84.00€
    25mg
    116.00€
    50mg
    161.00€
    100mg
    260.00€
    1mL*10mM (DMSO)
    64.00€
  • Salmeterol Xinafoate

    CAS:
    Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.
    Formula:C36H45NO7
    Purity:98% - 98.24%
    Color and Shape:White Solid
    Molecular weight:603.75

    Ref: TM-T6653

    5mg
    48.00€
    10mg
    74.00€
    25mg
    133.00€
    50mg
    215.00€
    100mg
    356.00€
    1mL*10mM (DMSO)
    60.00€
  • MRT-81

    CAS:
    MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.
    Formula:C31H29N3O5S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:555.64

    Ref: TM-T9532

    1mg
    48.00€
    5mg
    97.00€
    10mg
    145.00€
    25mg
    255.00€
    50mg
    368.00€
    100mg
    505.00€
    200mg
    692.00€
    1mL*10mM (DMSO)
    116.00€
  • BA 1 acetate(183241-31-8 free base)


    BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.
    Formula:C59H80N14O13
    Purity:95.3%
    Color and Shape:Solid
    Molecular weight:1193.35

    Ref: TM-TP1913L1

    1mg
    60.00€
    5mg
    110.00€
    10mg
    164.00€
    25mg
    286.00€
    50mg
    414.00€
    100mg
    577.00€
  • Binodenoson

    CAS:
    Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.
    Formula:C17H25N7O4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T9516

    1mg
    94.00€
    5mg
    222.00€
    10mg
    334.00€
    25mg
    557.00€
    50mg
    745.00€
    100mg
    1,044.00€
    1mL*10mM (DMSO)
    245.00€
  • Lecirelin acetate(61012-19-9 free base)


    Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts
    Formula:C61H88N16O14
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:1269.45

    Ref: TM-TP1434L

    1mg
    71.00€
    5mg
    124.00€
    10mg
    170.00€
    25mg
    255.00€
    50mg
    305.00€
    100mg
    462.00€
  • AR-M 1896 Acetate


    AR-M 1896 Acetate is the selective agonist of GalR2.
    Formula:C56H85N13O16
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:1196.35

    Ref: TM-T21646L

    1mg
    305.00€
    5mg
    605.00€
    10mg
    827.00€
    25mg
    1,215.00€
    50mg
    1,603.00€
    100mg
    2,142.00€
    1mL*10mM (DMSO)
    1,251.00€