GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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DOPEXAMINE
CAS:Dopexamine is a dopaminergic agonistFormula:C22H32N2O2Purity:99.42%Color and Shape:SolidMolecular weight:356.5Ref: TM-T8653
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)306.00€BisfluoroModafinil
CAS:CRL-40940 is a selective dopaminergic reuptake inhibitorFormula:C15H13F2NO2SPurity:99.19%Color and Shape:SolidMolecular weight:309.33Lanreotide acetate
CAS:Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndromeFormula:C56H73N11O12S2Purity:>99.99%Color and Shape:SolidMolecular weight:1156.39RS-127445 hydrochloride
CAS:RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formula:C17H17ClFN3Purity:99.48%Color and Shape:SolidMolecular weight:317.79ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purity:99.12%Color and Shape:SolidMolecular weight:307.139Ref: TM-T21970
5mg62.00€10mg90.00€25mg133.00€50mg192.00€100mg286.00€500mg687.00€1mL*10mM (DMSO)67.00€BD 1008 Free Base
CAS:BD 1008 Free Base: Sigma-1 receptor antagonist, Kᵢ = 2 ± 1 nM, 4x more selective for sigma-1 than sigma-2.Formula:C15H22Cl2N2Color and Shape:SolidMolecular weight:301.25Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Formula:C21H28ClN3O3SColor and Shape:SolidMolecular weight:437.98Facinicline (free base)
CAS:Facinicline (free base) is a partial agonist of the nicotinic alpha-7 (α7) receptor. It is used for the oral treatment of Alzheimer's.Formula:C15H18N4OColor and Shape:SolidMolecular weight:270.33Zacopride
CAS:Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias.Formula:C15H20ClN3O2Purity:98%Color and Shape:SolidMolecular weight:309.79Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purity:98.76% - 99.79%Color and Shape:SolidMolecular weight:295.38Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43DSP 4
CAS:DSP 4: neurotoxin targeting locus coeruleus, crosses blood-brain barrier, forms aziridinium, enters nerves via noradrenaline transporter.Formula:C11H15BrClNColor and Shape:SolidMolecular weight:276.6Atipamezole hydrochloride
CAS:Atipamezole is a synthetic α2 adrenergic receptor antagonist.Formula:C14H16N2·HClPurity:99.74%Color and Shape:SolidMolecular weight:248.75Ref: TM-T6765
5mg51.00€10mg74.00€25mg133.00€50mg230.00€100mg343.00€200mg535.00€500mg843.00€1mL*10mM (DMSO)57.00€Flibanserin hydrochloride
CAS:Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formula:C20H22ClF3N4OColor and Shape:SolidMolecular weight:426.87Carazolol
CAS:Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formula:C18H22N2O2Purity:99% - 99.53%Color and Shape:Yellowish SolidMolecular weight:298.38Bindarit
CAS:Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.Formula:C19H20N2O3Purity:98.35% - 98.55%Color and Shape:SolidMolecular weight:324.37Ref: TM-T6413
1mg35.00€2mg50.00€5mg75.00€10mg110.00€25mg178.00€50mg314.00€100mg492.00€200mg710.00€1mL*10mM (DMSO)84.00€Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purity:97.97%Color and Shape:SolidMolecular weight:754.85Guanfacine hydrochloride
CAS:Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formula:C9H10Cl3N3OPurity:99.89% - 99.91%Color and Shape:SolidMolecular weight:282.55Eltoprazine hydrochloride
CAS:Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formula:C12H17ClN2O2Purity:99.35%Color and Shape:SolidMolecular weight:256.73Moxisylyte
CAS:Moxisylyte (thymoxamine) treats erectile dysfunction, Reynaud's syndrome, and reverses eye mydriasis; it's an α1-adrenergic blocker.Formula:C16H25NO3Color and Shape:SolidMolecular weight:279.37
