GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5959 products of "GPCR/G-Protein"
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AF-710B
CAS:AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.Formula:C20H27N3OSPurity:98.62% - 99.89%Color and Shape:SolidMolecular weight:357.51Rotigotine
CAS:Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formula:C19H25NOSPurity:99.04% - 99.88%Color and Shape:SolidMolecular weight:315.47Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formula:(C6H14N2O2)x·xHBrColor and Shape:SolidMolecular weight:227.102KB-5492 free base
CAS:KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formula:C23H30N2O6Purity:97.10% - 97.94%Color and Shape:SolidMolecular weight:430.49Ref: TM-T62396
2mg39.00€5mg58.00€10mg82.00€25mg119.00€50mg168.00€100mg249.00€500mg613.00€1mL*10mM (DMSO)64.00€LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94UCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formula:C19H20N2O2Purity:98.88%Color and Shape:SolidMolecular weight:308.37Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37Trabodenoson
CAS:Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formula:C15H20N6O6Purity:99.94%Color and Shape:SolidMolecular weight:380.36Ref: TM-T34914
1mg40.00€5mg89.00€10mg116.00€25mg187.00€50mg285.00€100mg411.00€200mg577.00€1mL*10mM (DMSO)88.00€(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purity:99.75%Color and Shape:SolidMolecular weight:265.35Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purity:99.41% - >99.99%Color and Shape:SolidMolecular weight:517.66WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purity:99.96%Color and Shape:White SolidMolecular weight:538.645Ref: TM-T3453
2mg46.00€5mg66.00€10mg95.00€25mg159.00€50mg226.00€100mg334.00€500mg807.00€1mL*10mM (DMSO)79.00€SID 7969543
CAS:SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formula:C24H24N2O7Purity:98.94%Color and Shape:SolidMolecular weight:452.465-LOX inhibitor
CAS:5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) is an itraconazole impurity, a LOX-5 inhibitor.Formula:C22H27N5O2Purity:98.01%Color and Shape:SolidMolecular weight:393.48Ozanimod hydrochloride
CAS:Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formula:C23H25ClN4O3Purity:99.81%Color and Shape:SolidMolecular weight:440.92Ref: TM-T62552
1mg47.00€5mg92.00€10mg137.00€25mg268.00€50mg432.00€100mg620.00€200mg875.00€1mL*10mM (DMSO)101.00€Maropitant citrate
CAS:Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.Formula:C38H50N2O9Purity:98.91%Color and Shape:SolidMolecular weight:678.81Syk Inhibitor II
CAS:Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formula:C14H15F3N6OPurity:97.63%Color and Shape:SolidMolecular weight:340.3Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formula:C21H21D8Cl3N2O2Color and Shape:SolidMolecular weight:455.88(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS:(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H14D5Cl2N3SColor and Shape:SolidMolecular weight:289.28SR59230A hydrochloride
CAS:SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formula:C21H28ClNO2Purity:99.49%Color and Shape:SolidMolecular weight:361.91L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formula:C18H19ClN4Purity:98%Color and Shape:SolidMolecular weight:326.82
