GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5959 products of "GPCR/G-Protein"
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L-745870
CAS:L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formula:C18H19ClN4Purity:98%Color and Shape:SolidMolecular weight:326.82R 59-022
CAS:R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formula:C27H26FN3OSPurity:98.55%Color and Shape:SolidMolecular weight:459.58Ref: TM-T16709
1mg35.00€5mg74.00€10mg119.00€25mg269.00€50mg447.00€100mg733.00€200mg973.00€1mL*10mM (DMSO)75.00€Travoprost
CAS:Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formula:C26H35F3O6Purity:97.39% - 99.58%Color and Shape:Colorless OilMolecular weight:500.55Ref: TM-T5841
1mg46.00€5mg88.00€10mg120.00€25mg175.00€50mg255.00€100mg371.00€200mg507.00€1mL*10mM (DMSO)96.00€PACAP (1-38), human, ovine, rat
CAS:PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formula:C203H331N63O53SPurity:96.93% - 98.16%Color and Shape:SolidMolecular weight:4534.26Cyproheptadine hydrochloride
CAS:Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formula:C21H21N·HClPurity:99.88% - 99.97%Color and Shape:SolidMolecular weight:323.86Triflupromazine
CAS:Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formula:C18H19F3N2SColor and Shape:SolidMolecular weight:352.42Metoxibutropate
CAS:Metoxibutropate is a biochemical.Formula:C20H24O3Color and Shape:SolidMolecular weight:312.4PF-610355
CAS:PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.
Formula:C34H39N3O6SPurity:99.73%Color and Shape:SolidMolecular weight:617.76Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formula:C15H21ClN2SPurity:99.84%Color and Shape:SolidMolecular weight:296.8617-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the AllerganFormula:C26H38O5Color and Shape:SolidMolecular weight:430.58P2Y14R antagonist 1
CAS:P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.Formula:C15H12BrN3O2Purity:98.88%Color and Shape:SolidMolecular weight:346.18GPR183-IN-1
CAS:GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.Formula:C16H19BrN2O2Color and Shape:SolidMolecular weight:351.24GLP-1 Receptor modulator 1
CAS:GLP-1 Receptormodulator 1 (Compound 7) is an effective positive allosteric modulator of the GLP-1 receptor. It is utilized in the research of obesity and type 2 diabetes.Formula:C18H21NOSMolecular weight:299.43Meticillin
CAS:Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.Formula:C17H20N2O6SColor and Shape:SolidMolecular weight:380.42Eptinezumab
CAS:Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Purity:95% - 95%Color and Shape:LiquidEscitalopram
CAS:Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formula:C20H21FN2OPurity:99.82%Color and Shape:White Or White Crystalline PowderMolecular weight:324.39N-Methyl amisulpride
CAS:N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formula:C18H29N3O4SColor and Shape:SolidMolecular weight:383.51Olopatadine
CAS:Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.Formula:C21H23NO3Purity:98%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:337.41Risperidone Mesylate
CAS:Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formula:C24H31FN4O5SPurity:98%Color and Shape:SolidMolecular weight:506.59Arazasetron HCl
CAS:Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formula:C17H20ClN3O3Purity:98%Color and Shape:SolidMolecular weight:349.81
