
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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SB269652
CAS:SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.Formula:C27H30N4OPurity:98%Color and Shape:SolidMolecular weight:426.55A1/A3 AR antagonist 2
CAS:The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.Formula:C22H16N2O3SColor and Shape:SolidMolecular weight:388.44AB-MECA
CAS:AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.Formula:C18H21N7O4Purity:98%Color and Shape:SolidMolecular weight:399.4B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Color and Shape:SolidMolecular weight:1394.67SB-221284
CAS:5-HT2C/2B receptor antagonistFormula:C16H14F3N3OSPurity:98%Color and Shape:SolidMolecular weight:353.36MS47134
MS47134: potent MRGPRX4 agonist, EC50 = 149 nM, for pain/itch/hypersensitivity research.Formula:C22H29NO3Color and Shape:SolidMolecular weight:355.47ASP1126
CAS:ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).Formula:C26H26ClF6NO5Purity:98%Color and Shape:SolidMolecular weight:581.93AS604872
CAS:AS604872: Selective FP receptor antagonist, expedites cerebral/aorta degeneration, aids vascular disease models, inhibits uterine contraction.Formula:C28H25N3O3S2Color and Shape:SolidMolecular weight:515.65RP101988
RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.Formula:C23H22N4O4Color and Shape:SolidMolecular weight:418.45(R)-V-0219
(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.Formula:C20H25F3N4O2Color and Shape:SolidMolecular weight:410.43VUF-10497
CAS:VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).Formula:C18H20ClN5SPurity:98%Color and Shape:SolidMolecular weight:373.9Acreozast
CAS:Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.Formula:C15H14ClN3O6Color and Shape:SolidMolecular weight:367.74CB1 inverse agonist 2
CAS:CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.Formula:C24H20ClFN2OSColor and Shape:SolidMolecular weight:438.94RS 23597-190 hydrochloride
CAS:RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.Formula:C16H24Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:363.28Hedgehog IN-3
CAS:Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].Formula:C18H13ClF3N5OColor and Shape:SolidMolecular weight:407.78Flestolol sulfate
CAS:Flestolol sulfate is an anti-adrenergic beta-receptor.Formula:C15H24FN3O8SColor and Shape:SolidMolecular weight:425.43Phenindamine Tartrate
CAS:Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.Formula:C23H25NO6Color and Shape:SolidMolecular weight:411.454LY 163443
CAS:LY 163443 is an dual receptor antagonist of LTD4 and LTE4.Formula:C20H22N4O3Color and Shape:SolidMolecular weight:366.41Mabuterol hydrochloride
CAS:Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.Formula:C13H19Cl2F3N2OColor and Shape:SolidMolecular weight:347.20Quininib
CAS:Quininib inhibits ocular angiogenesis, blocks HMEC-1 tubules, aortic sprouts, and retinal revascularization in OIR mice.Formula:C17H13NOPurity:99.81%Color and Shape:SolidMolecular weight:247.29
