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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • SB269652

    CAS:
    SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.
    Formula:C27H30N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.55

    Ref: TM-T16857

    25mg
    1,288.00€
    50mg
    1,674.00€
    100mg
    2,250.00€
  • A1/A3 AR antagonist 2

    CAS:
    The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.
    Formula:C22H16N2O3S
    Color and Shape:Solid
    Molecular weight:388.44

    Ref: TM-T61744

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AB-MECA

    CAS:
    AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.
    Formula:C18H21N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.4

    Ref: TM-T14082

    1mg
    239.00€
    5mg
    1,018.00€
    10mg
    1,783.00€
  • B 4148

    CAS:
    B 4148 is a bradykinin inhibitor.
    Formula:C62H95N19O14S2
    Color and Shape:Solid
    Molecular weight:1394.67

    Ref: TM-T71571

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB-221284

    CAS:
    5-HT2C/2B receptor antagonist
    Formula:C16H14F3N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.36

    Ref: TM-T23317

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MS47134


    MS47134: potent MRGPRX4 agonist, EC50 = 149 nM, for pain/itch/hypersensitivity research.
    Formula:C22H29NO3
    Color and Shape:Solid
    Molecular weight:355.47

    Ref: TM-T73433

    25mg
    812.00€
    50mg
    1,054.00€
    100mg
    1,691.00€
  • ASP1126

    CAS:
    ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).
    Formula:C26H26ClF6NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:581.93

    Ref: TM-T10387

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • AS604872

    CAS:
    AS604872: Selective FP receptor antagonist, expedites cerebral/aorta degeneration, aids vascular disease models, inhibits uterine contraction.
    Formula:C28H25N3O3S2
    Color and Shape:Solid
    Molecular weight:515.65

    Ref: TM-T26665

    25mg
    1,369.00€
  • RP101988


    RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.
    Formula:C23H22N4O4
    Color and Shape:Solid
    Molecular weight:418.45

    Ref: TM-T73361

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • (R)-V-0219


    (R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.
    Formula:C20H25F3N4O2
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T73080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VUF-10497

    CAS:
    VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).
    Formula:C18H20ClN5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.9

    Ref: TM-T24951

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Acreozast

    CAS:
    Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.
    Formula:C15H14ClN3O6
    Color and Shape:Solid
    Molecular weight:367.74

    Ref: TM-T26555

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CB1 inverse agonist 2

    CAS:
    CB1 inverse agonist 2, an oral drug, counters CB1 effects, reducing CP55940-induced hypothermia and anorexia in mice.
    Formula:C24H20ClFN2OS
    Color and Shape:Solid
    Molecular weight:438.94

    Ref: TM-T72395

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RS 23597-190 hydrochloride

    CAS:
    RS 23597-190 hydrochloride is a 5-HT4 receptor antagonist.
    Formula:C16H24Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.28

    Ref: TM-T23255

    10mg
    388.00€
  • Hedgehog IN-3

    CAS:
    Hedgehog IN-3 (compound 3), with an IC50 value of 0.01 µM, serves as a hedgehog pathway inhibitor, proving beneficial for cancer research applications [1].
    Formula:C18H13ClF3N5O
    Color and Shape:Solid
    Molecular weight:407.78

    Ref: TM-T75148

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Flestolol sulfate

    CAS:
    Flestolol sulfate is an anti-adrenergic beta-receptor.
    Formula:C15H24FN3O8S
    Color and Shape:Solid
    Molecular weight:425.43

    Ref: TM-T27332

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Phenindamine Tartrate

    CAS:
    Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.
    Formula:C23H25NO6
    Color and Shape:Solid
    Molecular weight:411.454

    Ref: TM-T33978

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 163443

    CAS:
    LY 163443 is an dual receptor antagonist of LTD4 and LTE4.
    Formula:C20H22N4O3
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T27877

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Mabuterol hydrochloride

    CAS:
    Mabuterol hydrochloride is a selective β2 adrenoreceptor agonist. Mabuterol has a specific effect on beta 2-adrenoceptors with no beta 1-stimulation.
    Formula:C13H19Cl2F3N2O
    Color and Shape:Solid
    Molecular weight:347.20

    Ref: TM-T71803

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Quininib

    CAS:
    Quininib inhibits ocular angiogenesis, blocks HMEC-1 tubules, aortic sprouts, and retinal revascularization in OIR mice.
    Formula:C17H13NO
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:247.29

    Ref: TM-T28487

    500µg
    62.00€
    1mg
    89.00€
    5mg
    187.00€
    10mg
    281.00€
    25mg
    475.00€
    50mg
    675.00€
    100mg
    888.00€