
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Jmv 390-1
CAS:Jmv 390-1 is an inhibitor of metallopeptidase.Formula:C23H35N3O6Purity:98%Color and Shape:SolidMolecular weight:449.54UCM-05194
CAS:UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD 19.6 nM, inactive at LPA2-6/autotaxin).
Formula:C19H30BrO6PPurity:90% - 91.22%Color and Shape:SolidMolecular weight:465.32SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.86TIK-301
CAS:TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nMFormula:C14H17ClN2O2Purity:98%Color and Shape:SolidMolecular weight:280.75Levomoprolol
CAS:Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.Formula:C13H21NO3Purity:98%Color and Shape:SolidMolecular weight:239.312-Methylthioadenosine diphosphate trisodium
CAS:2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.Formula:C11H14N5Na3O10P2SColor and Shape:SolidMolecular weight:539.24Way 100289
CAS:Way 100289 is a selective 5-HT3 receptor antagonist.Formula:C20H27N3O3Color and Shape:SolidMolecular weight:357.45MK-2894
CAS:MK-2894 is a highly potent and selective antagonist of second generation EP4 .Formula:C25H22F3NO3SPurity:99.22%Color and Shape:SolidMolecular weight:473.51Ref: TM-T12061
1mg57.00€5mg120.00€1mL*10mM (DMSO)128.00€10mg205.00€25mg497.00€50mg879.00€100mg1,161.00€500mg2,367.00€RP5063 Hydrochloride
CAS:RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.Formula:C22H26Cl3N3O3Purity:98%Color and Shape:SolidMolecular weight:486.82Isamoltane hemifumarate
CAS:5-HT1B antagonistFormula:C16H22N202C4H404Purity:98%Color and Shape:SolidMolecular weight:332.4Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Formula:C16H17ClN2OSPurity:98%Color and Shape:SolidMolecular weight:320.84Cinalukast
CAS:CysLT1 leukotriene receptor antagonistFormula:C23H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:412.55L-771688 dihydrochloride
CAS:L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.Formula:C28H35Cl2F2N5O5Purity:98%Color and Shape:SolidMolecular weight:630.51Levoprotiline
CAS:Levoprotiline, a fast-acting antidepressant, is the R-enantiomer of Oxaprotiline and successor to maprotiline.Formula:C20H23NOPurity:98%Color and Shape:SolidMolecular weight:293.4Azintamide
CAS:Azintamide is a choleretic. It has shown effective and safe for dyspepsia symptoms when Domperidone therapy is not satisfactory.Formula:C10H14ClN3OSPurity:98%Color and Shape:SolidMolecular weight:259.76AUY954 HCl
CAS:AUY-954 is a potent and selective S1P(1) modulator. AUY-954 prevents experimental autoimmune neuritis in rats.Formula:C25H21ClF3NO2SColor and Shape:SolidMolecular weight:491.95SNAP 5089
CAS:α1A-adrenoceptor antagonistFormula:C36H40N4O5Purity:98%Color and Shape:SolidMolecular weight:608.73Dilevalol
CAS:Dilevalol ((+)-Labetalol) is a selective β2-adrenergic receptor agonist and non-selective β-adrenergic receptor blocker, hypertension and angina pectoris.Formula:C19H24N2O3Purity:98.05%Color and Shape:SolidMolecular weight:328.41TC-G1003
CAS:TC-G1003 is an effective agonist of the somatostatin sst2 receptor.Formula:C26H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:432.94Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Formula:C12H11N3OSColor and Shape:SolidMolecular weight:245.3
