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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Jmv 390-1

    CAS:
    Jmv 390-1 is an inhibitor of metallopeptidase.
    Formula:C23H35N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.54

    Ref: TM-T25554

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UCM-05194

    CAS:

    UCM-05194: potent LPA1 agonist, best for neuropathic pain relief (Emax 118%, EC50 0.24 μM, KD 19.6 nM, inactive at LPA2-6/autotaxin).

    Formula:C19H30BrO6P
    Purity:90% - 91.22%
    Color and Shape:Solid
    Molecular weight:465.32

    Ref: TM-T69647

    1mg
    316.00€
    5mg
    750.00€
    10mg
    1,064.00€
    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,783.00€
  • SCH-23390 maleate

    CAS:
    SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,
    Formula:C21H22ClNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.86

    Ref: TM-T12865

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TIK-301

    CAS:
    TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM
    Formula:C14H17ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.75

    Ref: TM-T17095

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Levomoprolol

    CAS:
    Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.
    Formula:C13H21NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.31

    Ref: TM-T25694

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-Methylthioadenosine diphosphate trisodium

    CAS:
    2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.
    Formula:C11H14N5Na3O10P2S
    Color and Shape:Solid
    Molecular weight:539.24

    Ref: TM-T23581

    1mg
    133.00€
    5mg
    570.00€
    10mg
    875.00€
  • Way 100289

    CAS:
    Way 100289 is a selective 5-HT3 receptor antagonist.
    Formula:C20H27N3O3
    Color and Shape:Solid
    Molecular weight:357.45

    Ref: TM-T35106

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MK-2894

    CAS:
    MK-2894 is a highly potent and selective antagonist of second generation EP4 .
    Formula:C25H22F3NO3S
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:473.51

    Ref: TM-T12061

    1mg
    57.00€
    5mg
    120.00€
    1mL*10mM (DMSO)
    128.00€
    10mg
    205.00€
    25mg
    497.00€
    50mg
    879.00€
    100mg
    1,161.00€
    500mg
    2,367.00€
  • RP5063 Hydrochloride

    CAS:
    RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.
    Formula:C22H26Cl3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.82

    Ref: TM-T24736

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Isamoltane hemifumarate

    CAS:
    5-HT1B antagonist
    Formula:C16H22N202C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.4

    Ref: TM-T22872

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dacemazine hydrochloride

    CAS:
    Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.
    Formula:C16H17ClN2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.84

    Ref: TM-T23949

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cinalukast

    CAS:
    CysLT1 leukotriene receptor antagonist
    Formula:C23H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.55

    Ref: TM-T22668

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-771688 dihydrochloride

    CAS:
    L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.
    Formula:C28H35Cl2F2N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:630.51

    Ref: TM-T24378

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • Levoprotiline

    CAS:
    Levoprotiline, a fast-acting antidepressant, is the R-enantiomer of Oxaprotiline and successor to maprotiline.
    Formula:C20H23NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.4

    Ref: TM-T25698

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Azintamide

    CAS:
    Azintamide is a choleretic. It has shown effective and safe for dyspepsia symptoms when Domperidone therapy is not satisfactory.
    Formula:C10H14ClN3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:259.76

    Ref: TM-T19851

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AUY954 HCl

    CAS:
    AUY-954 is a potent and selective S1P(1) modulator. AUY-954 prevents experimental autoimmune neuritis in rats.
    Formula:C25H21ClF3NO2S
    Color and Shape:Solid
    Molecular weight:491.95

    Ref: TM-T26685

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SNAP 5089

    CAS:
    α1A-adrenoceptor antagonist
    Formula:C36H40N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:608.73

    Ref: TM-T23374

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dilevalol

    CAS:
    Dilevalol ((+)-Labetalol) is a selective β2-adrenergic receptor agonist and non-selective β-adrenergic receptor blocker, hypertension and angina pectoris.
    Formula:C19H24N2O3
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:328.41

    Ref: TM-T25333

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
  • TC-G1003

    CAS:
    TC-G1003 is an effective agonist of the somatostatin sst2 receptor.
    Formula:C26H25ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.94

    Ref: TM-T24860

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Dacopafant

    CAS:
    Dacopafant is an antagonist of platlet activationg factor receptor.
    Formula:C12H11N3OS
    Color and Shape:Solid
    Molecular weight:245.3

    Ref: TM-T23951

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€