GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purity:98% - 99.82%Color and Shape:SolidMolecular weight:425.91GR 103691
CAS:GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).Formula:C30H35N3O3Purity:98.94% - 99.29%Color and Shape:SolidMolecular weight:485.62Ref: TM-T11463
2mg42.00€5mg62.00€10mg97.00€25mg187.00€50mg305.00€100mg487.00€200mg692.00€1mL*10mM (DMSO)66.00€Desvenlafaxine
CAS:Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formula:C16H25NO2Purity:99.46% - 99.81%Color and Shape:White Crystalline PowderMolecular weight:263.38Sarizotan 2HCl
CAS:Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.Formula:C22H23Cl2FN2OPurity:98.83%Color and Shape:SoildMolecular weight:421.34Retatrutide
CAS:<p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>Formula:C221H342N46O68Purity:98.31%Color and Shape:SolidMolecular weight:4732.09Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormula:C21H21ClN4OS·HCl·H2OPurity:98% - 99.83%Color and Shape:Off-White PowderMolecular weight:467.12JNJ-39758979
CAS:JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).Formula:C11H19N5Purity:98.33% - 99.62%Color and Shape:SolidMolecular weight:221.3Ref: TM-T11723L
1mg48.00€5mg97.00€10mg156.00€25mg255.00€50mg369.00€100mg543.00€200mg738.00€1mL*10mM (DMSO)105.00€Isothiuronium
CAS:Isothiouronium, a functional group, is the acid salt of isothiourea.Formula:C12H25IN2SPurity:>99.99%Color and Shape:SolidMolecular weight:356.31CGS 15943
CAS:CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formula:C13H8ClN5OPurity:97.4%Color and Shape:SolidMolecular weight:285.69Ref: TM-T14944
2mg35.00€5mg52.00€10mg87.00€25mg156.00€50mg235.00€100mg354.00€200mg520.00€1mL*10mM (DMSO)58.00€Vabicaserin hydrochloride
CAS:Vabicaserin hydrochloride (SCA 136) is a selective agonist of 5-hydroxytryptamine 2C (5-HT2C) receptor (EC50: 8 nM).Formula:C15H21ClN2Purity:98.32%Color and Shape:SolidMolecular weight:264.79Ref: TM-T13275
1mg84.00€5mg178.00€10mg264.00€25mg424.00€50mg562.00€100mg775.00€200mg1,026.00€1mL*10mM (DMSO)188.00€Isoxsuprine hydrochloride
CAS:Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formula:C18H24ClNO3Purity:99.38%Color and Shape:Crystals From Water SolidMolecular weight:337.84PF-04995274
CAS:PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formula:C23H32N2O6Purity:99.52%Color and Shape:SolidMolecular weight:432.51PF-4348235 2HCl
PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.Formula:C36H51Cl3N4O7SPurity:99.85%Color and Shape:SolidMolecular weight:790.24Ogerin
CAS:Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).Formula:C17H17N5OPurity:99.5% - 99.75%Color and Shape:SolidMolecular weight:307.35Naftidrofuryl oxalate
CAS:<p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>Formula:C26H35NO7Purity:97.12% - 98.38%Color and Shape:SolidMolecular weight:473.56Cimetidine
CAS:Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.Formula:C10H16N6SPurity:99.82%Color and Shape:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Molecular weight:252.34Abarelix
CAS:Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.Formula:C72H95ClN14O14Purity:>99.99%Color and Shape:SolidMolecular weight:1416.06Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24EMPA
CAS:EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nMFormula:C23H26N4O4SPurity:99.11%Color and Shape:SolidMolecular weight:454.54Ref: TM-T11186
1mg51.00€2mgTo inquire5mg97.00€10mg150.00€25mg264.00€50mg396.00€100mg595.00€200mg838.00€1mL*10mM (DMSO)110.00€Ticagrelor
CAS:Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.Formula:C23H28F2N6O4SPurity:98.08% - 99.77%Color and Shape:SolidMolecular weight:522.57
