GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Clomipramine hydrochloride
CAS:Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.Formula:C19H23ClN2·HClPurity:99.04% - 99.47%Color and Shape:White To Slightly Yellow Crystalline PowderMolecular weight:351.31RS102895 hydrochloride
CAS:RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).Formula:C21H22ClF3N2O2Purity:98.95%Color and Shape:SolidMolecular weight:426.86Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Formula:C30H32ClN3O8SPurity:98.46% - 99.89%Color and Shape:SolidMolecular weight:630.11Avexitide acetate
CAS:Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.Formula:C155H246N40O53SPurity:96.64% - 98.65%Color and Shape:SolidMolecular weight:3549.91CCR2-RA-[R]
CAS:CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).Formula:C18H19ClFNO3Purity:99.7%Color and Shape:SolidMolecular weight:351.8Isoxsuprine hydrochloride
CAS:Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formula:C18H24ClNO3Purity:99.38%Color and Shape:Crystals From Water SolidMolecular weight:337.84Traxanox
CAS:Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.Formula:C13H6ClN5O2Purity:98.37%Color and Shape:SolidMolecular weight:299.67(Rac)-MGV354
CAS:<p>(Rac)-MGV354: a racemic sGC activator; EC50s <0.5 nM (CHO cells), 5 nM (GTM-3 E cells).</p>Formula:C35H37N5O3Purity:99.26%Color and Shape:SolidMolecular weight:575.7Leronlimab
CAS:Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.Purity:SDS-PAGE:95.0%;SEC-HPLC:99.6%Color and Shape:LiquidMolecular weight:146.66 kDaCloroperone
CAS:<p>Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.</p>Formula:C22H23ClFNO2Purity:98.40%Color and Shape:SoildMolecular weight:387.88Promethazine
CAS:Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .Formula:C17H20N2SPurity:99.76%Color and Shape:CrystalsMolecular weight:284.42Pimethixene
CAS:Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.Formula:C19H19NSPurity:97.50%Color and Shape:SolidMolecular weight:293.43Ref: TM-T12489
2mg34.00€5mg50.00€10mg65.00€25mg106.00€50mg158.00€100mg226.00€200mg339.00€1mL*10mM (DMSO)52.00€Clopidogrel hydrogen sulfate
CAS:Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.Formula:C16H16ClNO2S·H2SO4Purity:99.57% - 99.79%Color and Shape:SolidMolecular weight:419.9Ziprasidone hydrochloride monohydrate
CAS:Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormula:C21H21ClN4OS·HCl·H2OPurity:98% - 99.83%Color and Shape:Off-White PowderMolecular weight:467.12Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurity:99.85%Color and Shape:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Molecular weight:320.88Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formula:C24H29ClF3N5O5SPurity:96.56%Color and Shape:SoildMolecular weight:592.03Aripiprazole Lauroxil
CAS:Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Formula:C36H51Cl2N3O4Purity:99.64%Color and Shape:SolidMolecular weight:660.71Ref: TM-T14319
10mg48.00€25mg72.00€50mg96.00€100mg130.00€200mg188.00€500mg318.00€1mL*10mM (DMSO)49.00€J-113863
CAS:J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).Formula:C30H37Cl2IN2O2Purity:95.11%Color and Shape:SolidMolecular weight:655.44Ref: TM-T11699
1mg59.00€2mg87.00€5mg126.00€10mg169.00€25mg304.00€50mg527.00€100mg758.00€1mL*10mM (DMSO)180.00€Isoprenaline hydrochloride
CAS:Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.Formula:C11H18ClNO3Purity:98% - 99.65%Color and Shape:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Molecular weight:247.719CCX140
CAS:CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.Formula:C20H13ClF3N5O3SPurity:99.66% - 99.95%Color and Shape:SolidMolecular weight:495.86
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