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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5962 products of "GPCR/G-Protein"

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  • LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:480.39
  • SB-423562

    CAS:
    SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
    Formula:C26H32N2O4
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:436.54
  • Vofopitant

    CAS:
    Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).
    Formula:C21H23F3N6O
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:432.44
  • Vofopitant dihydrochloride

    CAS:
    Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.
    Formula:C21H25Cl2F3N6O
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:505.36
  • AZD5462

    CAS:
    AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.
    Formula:C30H41FN2O6
    Purity:98.32% - 99.63%
    Color and Shape:Solid
    Molecular weight:544.65
  • PF-07258669

    CAS:
    PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
    Formula:C25H27FN6O2
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:462.52
  • Treprostinil diethanolamine

    CAS:
    <p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>
    Formula:C27H45NO7
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:495.65
  • BQ-788

    CAS:
    BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.
    Formula:C34H51N5O7
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:641.8
  • Rolapitant hydrochloride

    CAS:
    Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.
    Formula:C25H27ClF6N2O2
    Purity:98.35% - 99.79%
    Color and Shape:Solid
    Molecular weight:536.94
  • 7-Desmethyl-agomelatine

    CAS:
    7-Desmethyl-agomelatine, a metabolite of Agomelatine, exhibits lower activity than Agomelatine, which functions as a melatonergic (MT1 and MT2) agonist and 5-HT2C antagonist.
    Formula:C14H15NO2
    Color and Shape:Solid
    Molecular weight:229.27

    Ref: TM-T10193

    1mg
    Discontinued
    Discontinued product
  • Arotinolol

    CAS:
    Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand [125I-ICYP] to [5HT1B-serotonergic] receptor sites. It is an antihypertensive agent.
    Formula:C15H21N3O2S3
    Color and Shape:White Solid
    Molecular weight:371.54

    Ref: TM-T10371

    1mg
    Discontinued
    Discontinued product
  • SHA 68

    CAS:
    SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with IC50 values of 22.0 nM for NPSR Asn107 and 23.8 nM for NPSR Ile107.
    Formula:C26H24FN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.49

    Ref: TM-T12895

    1mg
    Discontinued
    Discontinued product
  • SB-399885 hydrochloride

    CAS:
    SB-399885 hydrochloride is an antagonist of 5-HT6 receptor.
    Formula:C18H22Cl3N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.81

    Ref: TM-T12843

    1mg
    Discontinued
    Discontinued product
  • JMV 2959

    CAS:
    JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).
    Formula:C30H32N6O2
    Color and Shape:Solid
    Molecular weight:508.61

    Ref: TM-T11719L

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product
  • Protease-Activated Receptor-4

    CAS:
    Protease-Activated Receptor-4 (PAR4) is a proteinase-activated receptor-4 agonist used in antiplatelet therapy.
    Formula:C33H46N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:666.77

    Ref: TM-T7380

    1mg
    Discontinued
    Discontinued product
  • BIBP3226 TFA

    CAS:
    BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).
    Formula:C29H32F3N5O5
    Color and Shape:Solid
    Molecular weight:587.59

    Ref: TM-T10540

    1mg
    Discontinued
    Discontinued product
  • HOKU-81

    CAS:
    HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.
    Formula:C12H18ClNO2
    Color and Shape:Solid
    Molecular weight:243.73

    Ref: TM-T15498

    1mg
    Discontinued
    Discontinued product
  • SR 146131

    CAS:
    SR 146131 is a potent and selective agonist of the nonpeptide receptor.
    Formula:C32H36ClN3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:610.16

    Ref: TM-T16935

    1mg
    Discontinued
    Discontinued product
  • ML-290

    CAS:
    ML-290 is an effective relaxin/insulin-like family peptide receptor (RXFP1) agonist and activator of anti-fibrotic genes. It shows an EC50 of 94 nM.
    Formula:C24H21F3N2O5S
    Color and Shape:Solid
    Molecular weight:506.49

    Ref: TM-T16101

    1mg
    Discontinued
    Discontinued product
  • CYM 9484

    CAS:
    CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with an IC50 value of 19 nM.
    Formula:C27H31N3O3S2
    Color and Shape:Solid
    Molecular weight:509.68

    Ref: TM-T10921

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product