GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .Formula:C41H57N9O10SColor and Shape:SolidMolecular weight:868.01Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Formula:C46H58F3N7O8Color and Shape:SolidMolecular weight:893.99Sauvagine TFA
Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.Formula:C204H347F3N56O65S1Color and Shape:SolidMolecular weight:4713.33LY-426965 hydrochloride
CAS:LY-426965 hydrochloride is a bioactive chemical.Formula:C28H39ClN2O2Color and Shape:SolidMolecular weight:471.07N,N′-Diferuloylputrescine
CAS:N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.Formula:C24H28N2O6Purity:98%Color and Shape:SolidMolecular weight:440.49(Phe2,Orn8)-Oxytocin
CAS:(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.Formula:C42H65N13O11S2Color and Shape:SolidMolecular weight:992.18AC 187 TFA
AC 187 TFA, a potent and orally active amylin receptor antagonist, exhibits an IC50 of 0.48 nM and a Ki of 0.275 nM.Formula:C129H206F3N37O42Color and Shape:SolidMolecular weight:3004.27hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (Formula:C37H62N10O9Purity:98%Color and Shape:SolidMolecular weight:790.95Kisspeptin-10, rat TFA
Kisspeptin-10, a rat TFA, constricts blood vessels, inhibits vessel growth, and counters Methotrexate reproductive toxicity.
Formula:C65H84F3N17O17Color and Shape:SolidMolecular weight:1432.46Guanylin(human) TFA
Guanylin (human) TFA, a 15-amino acid peptide, activates intestinal guanylate cyclase, regulating electrolyte and water transport via cGMP.Color and Shape:Liquid[Lys4] Sarafotoxin S6c
CAS:[Lys4] Sarafotoxin S6c: potent partial endothelin receptor agonist; causes pig coronary contraction, EC50=1.5 nM.Formula:C105H153N27O36S5Color and Shape:SolidMolecular weight:2529.82(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS:'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM forFormula:C107H162N30O30Color and Shape:SolidMolecular weight:2348.61Angiopeptin
CAS:Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.Formula:C54H71N11O10S2Color and Shape:SolidMolecular weight:1098.34ZL-1101
ZL-1101 is a human monoclonal antibody (mAb) targeting TNFRSF4/OX40/CD134.Color and Shape:Odour LiquidDapiglutide
CAS:Dapiglutide (ZP7570) is a long-acting GLP-1R & GLP-2R dual agonist for SBS research.Color and Shape:SolidRWJ 676070
CAS:RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.Formula:C30H26ClFN2O5Color and Shape:SolidMolecular weight:548.9915(S)-15-methyl Prostaglandin E2
CAS:15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49Obestatin(rat)
CAS:Endogenous peptide that suppresses food intake and body weight-gainFormula:C114H174N34O31Purity:98%Color and Shape:SolidMolecular weight:2516.81Human growth hormone-releasing factor TFA
Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.Formula:C217H359F3N72O68SColor and Shape:SolidMolecular weight:5153.67Ecnoglutide
CAS:Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .Formula:C194H304N48O61Color and Shape:SolidMolecular weight:4284.76
![[Lys4] Sarafotoxin S6c](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76302.webp&w=3840&q=75)
