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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5963 products of "GPCR/G-Protein"

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  • Proglumide hemicalcium

    CAS:
    Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.
    Formula:C18H28CaN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.51

    Ref: TM-T12544

    25mg
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    50mg
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    100mg
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  • Kisspeptin 234

    CAS:
    Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.
    Formula:C63H78N18O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1295.42

    Ref: TM-TP1896

    1mg
    610.00€
  • HAEGT

    CAS:

    HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.

    Formula:C20H31N7O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:513.5

    Ref: TM-TP1381

    1mg
    155.00€
    5mg
    449.00€
    10mg
    642.00€
  • FR 113680

    CAS:
    FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.
    Formula:C35H39N5O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:625.726

    Ref: TM-T27360

    25mg
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    50mg
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    100mg
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  • 5-hydroxy Propranolol

    CAS:
    5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.
    Formula:C16H21NO3
    Color and Shape:Solid
    Molecular weight:275.348

    Ref: TM-T36237

    1mg
    329.00€
    5mg
    1,539.00€
    10mg
    2,665.00€
    500µg
    210.00€
  • HL2-m5

    CAS:
    HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.
    Formula:C70H101N15O24S3
    Color and Shape:Solid
    Molecular weight:1632.83

    Ref: TM-TP3102

    10mg
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    50mg
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  • Lys-[Des-Arg9]Bradykinin TFA

    CAS:
    Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.
    Formula:C54H75F6N13O15
    Color and Shape:Solid
    Molecular weight:1260.24

    Ref: TM-T73646

    2mg
    63.00€
  • N6-Benzyl-5'-ethylcarboxamido adenosine

    CAS:
    N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.
    Formula:C19H22N6O4
    Color and Shape:Solid
    Molecular weight:398.42

    Ref: TM-T39011

    100mg
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    500mg
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  • Misoprostol acid

    CAS:
    Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.
    Formula:C21H36O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.51

    Ref: TM-T12047

    1mg
    178.00€
    5mg
    797.00€
    10mg
    1,521.00€
    50mg
    5,374.00€
  • Nesiritide

    CAS:
    Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.
    Formula:C143H244N50O42S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3464.04

    Ref: TM-TP1208

    1mg
    1,773.00€
  • Canine KP-10


    Canine KP-10 is a potent kisspeptin that induces a significant gonadotropin and estradiol response in female dogs during estrus.
    Color and Shape:Odour Solid

    Ref: TM-TP3851

    10mg
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    50mg
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  • Pal-Glu(OSu)-OH

    CAS:
    Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.
    Formula:C25H42N2O7
    Color and Shape:Solid
    Molecular weight:482.618

    Ref: TM-T40374

    100mg
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    500mg
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  • (R)-Preclamol hydrochloride

    CAS:
    (R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.
    Formula:C14H22ClNO
    Color and Shape:Solid
    Molecular weight:255.78

    Ref: TM-T73685

    2mg
    34.00€
  • ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate

    CAS:
    ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate is a platelet aggregation inhibitor.
    Formula:C22H18N4O3
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T9887

    1mg
    101.00€
    5mg
    215.00€
    10mg
    323.00€
    25mg
    545.00€
    50mg
    735.00€
    100mg
    979.00€
    200mg
    1,320.00€
    1mL*10mM (DMSO)
    To inquire
  • sGnRH-A

    CAS:
    sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.
    Formula:C64H83N17O12
    Color and Shape:Solid
    Molecular weight:1282.45

    Ref: TM-T76312

    5mg
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    50mg
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  • TAK-683 acetate


    TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.
    Formula:C66H87N17O15
    Color and Shape:Solid
    Molecular weight:1358.5

    Ref: TM-T76048

    5mg
    To inquire
    50mg
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  • MRS2500 tetraammonium

    CAS:
    Highly potent and selective antagonist of the platelet P2Y1 receptor
    Formula:C13H21IN6O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.19

    Ref: TM-T23023

    1mg
    To inquire
  • GLP-2(1-33)(human)

    CAS:
    GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.
    Formula:C165H254N44O55S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3766.19

    Ref: TM-TP1157

    1mg
    309.00€
  • Vedaprofen

    CAS:

    Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.

    Formula:C19H22O2
    Purity:99.24% - 99.70%
    Color and Shape:Solid
    Molecular weight:282.38

    Ref: TM-T36683

    1mg
    54.00€
    5mg
    73.00€
    10mg
    116.00€
    25mg
    226.00€
    50mg
    335.00€
    100mg
    470.00€
  • Vicasinabin

    CAS:
    Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.
    Formula:C15H22N10O
    Color and Shape:Solid
    Molecular weight:358.41

    Ref: TM-T38912

    5mg
    710.00€