
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Proglumide hemicalcium
CAS:Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.Formula:C18H28CaN2O4Purity:98%Color and Shape:SolidMolecular weight:376.51Kisspeptin 234
CAS:Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.Formula:C63H78N18O13Purity:98%Color and Shape:SolidMolecular weight:1295.42HAEGT
CAS:HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.
Formula:C20H31N7O9Purity:98%Color and Shape:SolidMolecular weight:513.5FR 113680
CAS:FR 113680 is a tripeptide substance P antagonist with NK1 receptor selectivity.Formula:C35H39N5O6Purity:98%Color and Shape:SolidMolecular weight:625.7265-hydroxy Propranolol
CAS:5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Formula:C16H21NO3Color and Shape:SolidMolecular weight:275.348HL2-m5
CAS:HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formula:C70H101N15O24S3Color and Shape:SolidMolecular weight:1632.83Lys-[Des-Arg9]Bradykinin TFA
CAS:Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Formula:C54H75F6N13O15Color and Shape:SolidMolecular weight:1260.24N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42Misoprostol acid
CAS:Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.Formula:C21H36O5Purity:98%Color and Shape:SolidMolecular weight:368.51Nesiritide
CAS:Nesiritide, recombinant human B-type natriuretic peptide, binds NPR-A/C with Kd 7.3/13 pM.Formula:C143H244N50O42S4Purity:98%Color and Shape:SolidMolecular weight:3464.04Canine KP-10
Canine KP-10 is a potent kisspeptin that induces a significant gonadotropin and estradiol response in female dogs during estrus.Color and Shape:Odour SolidPal-Glu(OSu)-OH
CAS:Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.Formula:C25H42N2O7Color and Shape:SolidMolecular weight:482.618(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Formula:C14H22ClNOColor and Shape:SolidMolecular weight:255.78ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate
CAS:ethyl 1-[(4-cyanobenzyl)oxy]-2-(3-cyanophenyl)-4-methyl-1H-imidazole-5-carboxylate is a platelet aggregation inhibitor.Formula:C22H18N4O3Purity:99.86%Color and Shape:SolidMolecular weight:386.4Ref: TM-T9887
1mg101.00€5mg215.00€10mg323.00€25mg545.00€50mg735.00€100mg979.00€200mg1,320.00€1mL*10mM (DMSO)To inquiresGnRH-A
CAS:sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formula:C64H83N17O12Color and Shape:SolidMolecular weight:1282.45TAK-683 acetate
TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.Formula:C66H87N17O15Color and Shape:SolidMolecular weight:1358.5MRS2500 tetraammonium
CAS:Highly potent and selective antagonist of the platelet P2Y1 receptorFormula:C13H21IN6O8P2Purity:98%Color and Shape:SolidMolecular weight:578.19GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19Vedaprofen
CAS:Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.
Formula:C19H22O2Purity:99.24% - 99.70%Color and Shape:SolidMolecular weight:282.38Vicasinabin
CAS:Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.Formula:C15H22N10OColor and Shape:SolidMolecular weight:358.41

