GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
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Subcategories of "GPCR/G-Protein"
5-HT Receptor
Adenosine Receptor
Adrenergic Receptor
Bombesin Receptor
Bradykinin Receptor
CXCR
CaSR
Cannabinoid Receptor
Cholecystokinin
Dopamine Receptor
Endothelin Receptor
GNRH Receptor
GPCR19
GRK
GTPase
Glucagon Receptor
Hedgehog/Smoothened
Histamine Receptor
LPA Receptor
Melatonin Receptor
OX Receptor
Opioid Receptor
PAFR
PKA
S1P Receptor
SGLT
Sigma receptor
Show 19 more subcategories
Products of "GPCR/G-Protein"
Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows …
Formula:
C80H112N18O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1693.98
Ref: TM-TP1188L
| 1mg | 106.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 340.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 979.00 € | ||
| 200mg | 1,309.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Formula:
C23H27F3N2O3
Purity:
98.10%
Color and Shape:
Soild
Molecular weight:
436.47
Ref: TM-T68023L
| 1mg | 182.00 € | ||
| 5mg | 399.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,267.00 € | ||
| 100mg | 1,710.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BAM (8-22) acetate
BAM (8-22) acetate, a proenkephalin A derivative, stimulates MrgprC11, hMrgprX1, and causes scratching in mice.
Formula:
C93H131N25O25S
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
2031.25
Ref: TM-TP1914L1
| 1mg | 292.00 € | ||
| 5mg | 547.00 € | ||
| 10mg | 730.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,464.00 € | ||
| 100mg | 1,985.00 € | ||
| 200mg | 2,681.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
PF-9184
CAS:1221971-47-6
PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 …
Formula:
C21H14Cl2N2O4S
Purity:
97.64%
Color and Shape:
Solid
Molecular weight:
461.32
Ref: TM-T21738
| 1mg | 35.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Dec 2024
2-Oleoylglycerol
CAS:3443-84-3
2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with …
Formula:
C21H40O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
356.54
Ref: TM-T37526
| 1mg (28mM*100μL in Ethanol) | 92.00 € | ||
| 25mg (28mM*2.5mL in Ethanol) | To inquire |
Estimated delivery in United States, on Monday 2 Dec 2024
![[Des-Arg9]-Bradykinin](https://static.cymitquimica.com/products/TM/thumb/T7645.jpg)
[Des-Arg9]-Bradykinin
CAS:15958-92-6
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Formula:
C44H61N11O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
904.02
Ref: TM-T7645
| 5mg | 252.00 € | ||
| 10mg | 444.00 € | ||
| 25mg | 936.00 € | ||
| 50mg | 1,470.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Mifentidine
CAS:83184-43-4
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric …
Formula:
C13H16N4
Purity:
100% - 99.20%
Color and Shape:
Liquid
Molecular weight:
228.29
Ref: TM-T68100
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
S1R agonist 2
CAS:150085-21-5
S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for …
Formula:
C21H27NO
Purity:
99.04%
Color and Shape:
Liquid
Molecular weight:
309.45
Ref: TM-T72059
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 600.00 € | ||
| 500mg | 1,268.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Senktide acetate
Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of …
Formula:
C42H59N7O13S
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
902.02
Ref: TM-T7633L
| 1mg | 89.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 930.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.
Formula:
C33H35F3N6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
620.66
Ref: TM-T11671
| 2mg | 374.00 € | ||
| 5mg | 560.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 763.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is …
Formula:
C42H61N11O19
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1024.01
Ref: TM-TP1452L1
| 1mg | 251.00 € | ||
| 5mg | 513.00 € | ||
| 10mg | 777.00 € | ||
| 25mg | 1,398.00 € | ||
| 50mg | 2,095.00 € | ||
| 100mg | 3,143.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Saterinone
CAS:102669-89-6
Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 …
Formula:
C27H30N4O4
Purity:
98.23%
Color and Shape:
Liquid
Molecular weight:
474.55
Ref: TM-T68138
| 1mg | 152.00 € | ||
| 5mg | 365.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,212.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 152.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 876.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,214.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Dalcotidine
CAS:120958-90-9
Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, …
Formula:
C18H29N3O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
319.44
Ref: TM-T31195
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,971.00 € | ||
| 1mL*10mM (DMSO) | 338.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Seganserin
CAS:87729-89-3
Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.
Formula:
C29H27F2N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
471.54
Ref: TM-T68141
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,438.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
Formula:
C22H29ClN2O2
Purity:
99.45%
Color and Shape:
Liquid
Molecular weight:
388.93
Ref: TM-T30586L
| 1mg | 183.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,415.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Fargesone B
CAS:116424-70-5
Fargesone B inhibits the vascular smooth muscle contraction by suppressing the voltage- and receptor-activated calcium …
Formula:
C21H24O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.417
Ref: TM-TN4051
| 5mg | 557.00 € | ||
| 1mL*10mM (DMSO) | 576.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Bucumolol
CAS:58409-59-9
Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and …
Formula:
C17H23NO4
Purity:
99.70%
Color and Shape:
Soild
Molecular weight:
305.37
Ref: TM-T30606L
| 1mg | 193.00 € | ||
| 5mg | 477.00 € | ||
| 10mg | 670.00 € | ||
| 25mg | 1,045.00 € | ||
| 50mg | 1,442.00 € | ||
| 100mg | 1,846.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
15(R)-15-methyl Prostaglandin D2
CAS:210978-26-0
15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor …
Formula:
C21H34O5
Color and Shape:
Liquid
Molecular weight:
366.49
Ref: TM-T37264
| 1mg | 313.00 € | ||
| 500µg | 185.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
REV 5901A
CAS:92532-23-5
REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial …
Formula:
C22H26ClNO2
Purity:
99.74%
Color and Shape:
Soild
Molecular weight:
371.90
Ref: TM-T21821L
| 1mg | 182.00 € | ||
| 5mg | 450.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,388.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
