
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5958 products of "GPCR/G-Protein"
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Antipsychotic agent-2
Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.Formula:C22H26FN5OColor and Shape:SolidMolecular weight:395.47PACAP-Related Peptide (PRP), human
PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.Formula:C139H229N41O42Purity:98%Color and Shape:SolidMolecular weight:3146.57Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColor and Shape:SolidMolecular weight:435.96Pentagastrin meglumine
CAS:Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.Formula:C44H66N8O14SColor and Shape:SolidMolecular weight:963.11Lu AA33810
CAS:Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and BBB permeability, anti-anxiety and antidepressant-like effects.Formula:C19H25N3O2S3Purity:97.92% - 99.61%Color and Shape:SolidMolecular weight:423.62YM 09538
CAS:YM 09538 is a biochemical.Formula:C18H25ClN2O5SColor and Shape:SolidMolecular weight:416.92MMC(TMZ)-TOC TFA
MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.Formula:C74H99F3N20O21S2Color and Shape:SolidMolecular weight:1725.82Pancreatic Polypeptide, rat
CAS:Rat Pancreatic Polypeptide: 36-amino acid peptide, NPYR4 agonist, secreted by islet PP cells.Formula:C195H298N58O57SPurity:98%Color and Shape:SolidMolecular weight:4398.87Adrenomedullin (AM) (22-52), human
CAS:Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.Formula:C159H252N46O48Purity:98%Color and Shape:SolidMolecular weight:3576.04Bremelanotide
CAS:Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.Formula:C50H68N14O10Purity:98%Color and Shape:White PowderMolecular weight:1025.16GR 64349
CAS:Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.Formula:C42H68N10O11SPurity:98%Color and Shape:SolidMolecular weight:921.12Propranolol hydrochloride
CAS:Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverseFormula:C16H22ClNO2Purity:99.94% - >99.99%Color and Shape:White Or Almost White Powder White PowderMolecular weight:295.80Synephrine hemitartrate
CAS:Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.Formula:C9H13NO2C4H6O6Color and Shape:SolidMolecular weight:242.26Antisauvagine-30 TFA
aSvg-30 TFA: potent CRF2 receptor antagonist, Kd 1.4 nM (mCRFR2β), 150 nM (CRFR1).Formula:C163H275N48F3O49SColor and Shape:SolidMolecular weight:3764.28ACTH (11-24)
CAS:ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.Formula:C77H134N24O16Purity:98%Color and Shape:SolidMolecular weight:1652.0411-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48D[LEU4,LYS8]-VP TFA
D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.
Formula:C49H68F3N11O13S2Color and Shape:SolidMolecular weight:1140.25Adrenomedullin (16-31), human
CAS:Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Formula:C82H129N25O21S2Purity:98%Color and Shape:SolidMolecular weight:1865.19BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formula:C33H43F3N6O9Color and Shape:SolidMolecular weight:724.72BAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Formula:C26H28BrCl2N3O3Color and Shape:SolidMolecular weight:581.33

