CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5958 products of "GPCR/G-Protein"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Antipsychotic agent-2


    Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.
    Formula:C22H26FN5O
    Color and Shape:Solid
    Molecular weight:395.47

    Ref: TM-T74798

    5mg
    To inquire
    50mg
    To inquire
  • PACAP-Related Peptide (PRP), human


    PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.
    Formula:C139H229N41O42
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3146.57

    Ref: TM-TP1850

    1mg
    122.00€
    5mg
    356.00€
  • Adrogolide HCl

    CAS:
    Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.
    Formula:C22H26ClNO4S
    Color and Shape:Solid
    Molecular weight:435.96

    Ref: TM-T29674

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • Pentagastrin meglumine

    CAS:
    Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.
    Formula:C44H66N8O14S
    Color and Shape:Solid
    Molecular weight:963.11

    Ref: TM-T33916

    100mg
    To inquire
    500mg
    To inquire
  • Lu AA33810

    CAS:
    Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and BBB permeability, anti-anxiety and antidepressant-like effects.
    Formula:C19H25N3O2S3
    Purity:97.92% - 99.61%
    Color and Shape:Solid
    Molecular weight:423.62

    Ref: TM-T22935

    1mg
    164.00€
    5mg
    398.00€
    10mg
    681.00€
    25mg
    1,036.00€
    50mg
    1,420.00€
    100mg
    1,821.00€
  • YM 09538

    CAS:
    YM 09538 is a biochemical.
    Formula:C18H25ClN2O5S
    Color and Shape:Solid
    Molecular weight:416.92

    Ref: TM-T35252

    25mg
    1,369.00€
  • MMC(TMZ)-TOC TFA


    MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.
    Formula:C74H99F3N20O21S2
    Color and Shape:Solid
    Molecular weight:1725.82

    Ref: TM-T204151

    10mg
    To inquire
    50mg
    To inquire
  • Pancreatic Polypeptide, rat

    CAS:
    Rat Pancreatic Polypeptide: 36-amino acid peptide, NPYR4 agonist, secreted by islet PP cells.
    Formula:C195H298N58O57S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4398.87

    Ref: TM-TP1044

    1mg
    324.00€
    5mg
    973.00€
  • Adrenomedullin (AM) (22-52), human

    CAS:
    Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.
    Formula:C159H252N46O48
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3576.04

    Ref: TM-TP1257

    1mg
    178.00€
    5mg
    712.00€
  • Bremelanotide

    CAS:
    Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.
    Formula:C50H68N14O10
    Purity:98%
    Color and Shape:White Powder
    Molecular weight:1025.16

    Ref: TM-T20467

    100mg
    To inquire
    500mg
    To inquire
  • GR 64349

    CAS:
    Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.
    Formula:C42H68N10O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:921.12

    Ref: TM-TP2023

    1mg
    1,575.00€
  • Propranolol hydrochloride

    CAS:
    Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse
    Formula:C16H22ClNO2
    Purity:99.94% - >99.99%
    Color and Shape:White Or Almost White Powder White Powder
    Molecular weight:295.80

    Ref: TM-T0812

    1g
    117.00€
    25mg
    38.00€
    50mg
    50.00€
    100mg
    67.00€
    200mg
    82.00€
    500mg
    97.00€
    1mL*10mM (DMSO)
    55.00€
  • Synephrine hemitartrate

    CAS:
    Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.
    Formula:C9H13NO2C4H6O6
    Color and Shape:Solid
    Molecular weight:242.26

    Ref: TM-T75425

    5mg
    To inquire
    50mg
    To inquire
  • Antisauvagine-30 TFA


    aSvg-30 TFA: potent CRF2 receptor antagonist, Kd 1.4 nM (mCRFR2β), 150 nM (CRFR1).
    Formula:C163H275N48F3O49S
    Color and Shape:Solid
    Molecular weight:3764.28

    Ref: TM-T75805

    5mg
    To inquire
    50mg
    To inquire
  • ACTH (11-24)

    CAS:
    ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.
    Formula:C77H134N24O16
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1652.04

    Ref: TM-TP1248

    1mg
    56.00€
    5mg
    104.00€
    10mg
    142.00€
  • 11-deoxy Prostaglandin E1

    CAS:
    11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause
    Formula:C20H34O4
    Color and Shape:Solid
    Molecular weight:338.48

    Ref: TM-T36770

    1mg
    212.00€
    5mg
    874.00€
    10mg
    1,510.00€
    500µg
    118.00€
  • D[LEU4,LYS8]-VP TFA


    D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.

    Formula:C49H68F3N11O13S2
    Color and Shape:Solid
    Molecular weight:1140.25

    Ref: TM-T75826

    5mg
    To inquire
    50mg
    To inquire
  • Adrenomedullin (16-31), human

    CAS:
    Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).
    Formula:C82H129N25O21S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1865.19

    Ref: TM-TP1486

    100mg
    To inquire
    500mg
    To inquire
  • BQ-123 TFA


    BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.
    Formula:C33H43F3N6O9
    Color and Shape:Solid
    Molecular weight:724.72

    Ref: TM-T73877

    5mg
    To inquire
    50mg
    To inquire
  • BAY-6672 hydrochloride

    CAS:
    BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.
    Formula:C26H28BrCl2N3O3
    Color and Shape:Solid
    Molecular weight:581.33

    Ref: TM-T74213

    5mg
    To inquire
    50mg
    To inquire