GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Color and Shape:SolidMolecular weight:1040.974-Butyl-α-agarofuran
CAS:4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.Formula:C18H30OColor and Shape:SolidMolecular weight:262.43Neuropeptide S(Rat)
CAS:Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formula:C95H160N34O27Purity:98%Color and Shape:SolidMolecular weight:2210.52Upidosin
CAS:Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.
Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61Sibenadet hydrochloride
CAS:Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.Formula:C22H29ClN2O5S2Color and Shape:SolidMolecular weight:501.06TT-OAD2
CAS:TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.
Formula:C50H49Cl4N3O6Purity:98%Color and Shape:SolidMolecular weight:929.75M617
CAS:Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.Formula:C112H161N29O28Purity:98%Color and Shape:SolidMolecular weight:2361.68Cortistatin-8
CAS:ghrelin receptor antagonistFormula:C47H68N12O9S2Purity:98%Color and Shape:SolidMolecular weight:1009.25LTB4-IN-2
LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with anFormula:C24H17N5S2Purity:98%Color and Shape:SolidMolecular weight:439.56RC-3095
CAS:RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.Formula:C56H79N15O9Purity:98%Color and Shape:SolidMolecular weight:1106.32WS 9326A
CAS:WS 9326A is an antagonist of tachykinin receptor from Streptomyces violaceusniger.Formula:C54H68N8O13Purity:98%Color and Shape:SolidMolecular weight:1037.181Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Formula:C77H112N20O15Purity:98.9200%Color and Shape:SolidMolecular weight:1557.84ELA-11(human)
CAS:Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.Formula:C58H90N16O13S2Purity:98%Color and Shape:SolidMolecular weight:1283.57PF-4348235 HCl
PF-4348235 HCl (β2AR/M-receptor agonist-2 HCl) is a muscarinic M3 receptor antagonist (Ki: 0.73 nM) and β2 adrenergic receptor agonist (MABA, EC50: 3.7 nM). PF-4348235 HCl is also a bronchial BM213 acetate is a bronchodilator used to study cardiovascular and respiratory diseases such as chronic obstructive pulmonary disease (COPD).
Formula:C36H50Cl2N4O7SPurity:98.81%Color and Shape:SolidMolecular weight:753.78Colulintide
CAS:Colulintide is an analog of amylin, utilized in obesity research.Color and Shape:SolidElabela(19-32)
CAS:APJ receptor agonist with Ki of 0.93 nM, derived from ELA-32, activates Gαi1, β-arrestin-2, lowers rat heart arterial pressure, effective in vivo.Formula:C75H119N25O17S2Purity:98%Color and Shape:SolidMolecular weight:1707.03P2Y14 antagonist 1
P2Y14 antagonist 1 (compound 45) is a highly selective and orally active P2Y14 receptor antagonist with an IC50 value of 0.70 nM. It demonstrates significant anti-inflammatory effects by effectively reducing pulmonary infiltration of immune cells and inflammatory responses through the inhibition of the NLRP3 signaling pathway. P2Y14 antagonist 1 is suitable for studying acute lung injury.Formula:C24H21N3O3Color and Shape:SolidMolecular weight:399.442I-BOP
CAS:I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).Formula:C23H29IO5Color and Shape:SolidMolecular weight:512.384IRL-1620 acetate
IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a Ki of 16 pM which is more selective than ETA with a Ki of 19 μM.Formula:C88H121N17O29Purity:96.64%Color and Shape:SolidMolecular weight:1881MCUF-651
CAS:MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.Formula:C17H22F2N4OSPurity:99.83%Color and Shape:SoildMolecular weight:368.44Ref: TM-T67734
1mg56.00€5mg118.00€10mg178.00€25mg344.00€50mg557.00€100mg790.00€1mL*10mM (DMSO)126.00€
