
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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11-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48α-CGRP (mouse, rat) (TFA)
α-CGRP (mouse, rat) TFA is a neuropeptide (calcitonin gene-related peptide) predominantly found at neuromuscular junctions and acts as a potent vasodilator. This compound is useful in research concerning cardiovascular, pro-inflammatory, migraine, and metabolic processes.Color and Shape:Odour SolidQuinazosin hydrochloride
CAS:Quinazosin hydrochloride is an antihypertensive agent.Formula:C17H25Cl2N5O2Color and Shape:SolidMolecular weight:402.32TT 232
CAS:sst1/sst4 somatostatin receptors agonistFormula:C45H58N10O9S2Purity:98%Color and Shape:SolidMolecular weight:947.13Hemopressin(rat)
CAS:Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formula:C53H77N13O12Purity:98%Color and Shape:SolidMolecular weight:1088.27Sch 202596
CAS:Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formula:C25H22Cl2O12Color and Shape:SolidMolecular weight:585.34Glucagon-like peptide 1 (1-37), human
CAS:Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.Formula:C186H275N51O59Purity:98%Color and Shape:SolidMolecular weight:4169.48GPR61 Inverse agonist 1
Compound 1, identified as a GPR61 inverse agonist, exhibits an IC50 of 11 nM, rendering it suitable for metabolism and body weight disorder research, includingColor and Shape:Odour SolidGLP-1 receptor agonist 13
Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1].Formula:C25H23ClF2N6OColor and Shape:SolidMolecular weight:496.94Clozapine N-oxide dihydrochloride
CAS:Clozapine N-oxide dihydrochloride is a derivative of Clozapine and an agonist of DREADDs.Formula:C18H21Cl3N4OPurity:98.11%Color and Shape:SolidMolecular weight:415.74Zovaglutide
CAS:Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Color and Shape:SolidK-(D-1-Nal)-FwLL-NH2
CAS:Potent ghrelin receptor inverse agonist with Ki of 4.9/31 nM in COS7/HEK293T; blocks Gq/G13 signaling.Formula:C51H67N9O6Purity:98%Color and Shape:SolidMolecular weight:902.13Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.Formula:C212H316F3N57O59SPurity:98%Color and Shape:SolidMolecular weight:4696.18Bromchlorbuterol hydrochloride
CAS:Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.Formula:C12H19BrCl2N2OColor and Shape:SolidMolecular weight:358.1Cholecystokinin Octapeptide, desulfated TFA
CAS:Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.Formula:C51H63F3N10O15S2Color and Shape:SolidMolecular weight:1177.24Cetamolol hydrochloride
CAS:Cetamolol hydrochloride is a biochemical.Formula:C16H27ClN2O4Color and Shape:SolidMolecular weight:346.85GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Formula:C140H214N36O43Purity:97%Color and Shape:SolidMolecular weight:3089.41Osanetant
CAS:Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.Formula:C35H41Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:606.62Lu AA33810
CAS:Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and BBB permeability, anti-anxiety and antidepressant-like effects.Formula:C19H25N3O2S3Purity:97.92% - 99.61%Color and Shape:SolidMolecular weight:423.62Amylin (8-37), rat
CAS:Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.Formula:C140H227N43O43Purity:98%Color and Shape:SolidMolecular weight:3200.61

