GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide
CAS:Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which hasFormula:C25H35NO4Color and Shape:SolidMolecular weight:413.558(Phe2,Orn8)-Oxytocin
CAS:(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.Formula:C42H65N13O11S2Color and Shape:SolidMolecular weight:992.18Bosentan-d4
CAS:Bosentan-d4: deuterium version of Bosentan, competitive ET A/B antagonist, Ki: 4.7nM (ET A), 95nM (ET B) in human SMC.Formula:C27H25D4N5O6SColor and Shape:SolidMolecular weight:555.64[8-L-arginine] deaminovasopressin
CAS:[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .Formula:C46H64N14O13S2Color and Shape:SolidMolecular weight:1085.22Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Color and Shape:SolidMolecular weight:461.81CIA-1 (Free base)
CAS:CIA-1, a COUP-TFII inhibitor, has IC50 of 1.2-7.6 μM in prostate cancer cells; inhibits tumor growth in mouse prostate cancer.Formula:C17H19N3O2SPurity:99%Color and Shape:SolidMolecular weight:329.42[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Formula:C58H82N16O12Color and Shape:SolidMolecular weight:1195.37Tecastemizole
CAS:Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formula:C19H21FN4Purity:99.70%Color and Shape:SolidMolecular weight:324.4Ref: TM-T26253
1mg54.00€5mg118.00€1mL*10mM (DMSO)131.00€10mg168.00€25mg288.00€50mg414.00€100mg583.00€500mg1,161.00€(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS:(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formula:C53H62N12O11Molecular weight:1043.13TT 232
CAS:sst1/sst4 somatostatin receptors agonistFormula:C45H58N10O9S2Purity:98%Color and Shape:SolidMolecular weight:947.13Corticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.Purity:98.30%Color and Shape:LiquidOxopurpureine
CAS:Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.Formula:C21H19NO6Color and Shape:SolidMolecular weight:381.38[Leu13]-Motilin
CAS:[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinalFormula:C121H190N34O35Purity:98%Color and Shape:SolidMolecular weight:2681.01tetranor-PGDM
CAS:PGD2, made by H-PGDS in mast cells and lipocalin-PGD-synthase in the brain, aids sleep, cools the body, and inhibits platelet aggregation.Formula:C16H24O7Color and Shape:SolidMolecular weight:328.361PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purity:98%Color and Shape:SolidMolecular weight:2215.492,3-dinor Thromboxane B1
CAS:TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formula:C18H32O6Color and Shape:SolidMolecular weight:344.448(Leu31,Pro34)-Peptide YY (human)
CAS:(Leu31,Pro34)-Peptide YY (human) is a derivative of Peptide YY, acting as a potent and selective Y1 receptor agonist with a dissociation constant (KD) of 1.0 nMFormula:C195H296N54O56Color and Shape:SolidMolecular weight:4292.75tcY-NH2
CAS:Selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formula:C40H49N7O7Purity:98%Color and Shape:SolidMolecular weight:739.87PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09Pasireotide pamoate
CAS:Pasireotide pamoate is a stable cyclohexapeptide somatostatin mimic. Pasireotide pamoate exhibits antisecretory, antiproliferative, and proapoptotic activity.Formula:C81H82N10O15Purity:98%Color and Shape:SolidMolecular weight:1435.58
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