GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Mosapride citrate dihydrate
CAS:Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.Formula:C27H35ClFN3O11Purity:98%Color and Shape:SolidMolecular weight:632.04[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formula:C54H71N15O14Purity:98%Color and Shape:SolidMolecular weight:1154.23APJ receptor agonist 4
CAS:Potent, orally active APJ receptor agonist 4; EC50: 0.06 nM, Ki: 0.07 nM; good pharmacokinetics in rodent HF model; safe in studies; boosts cardiac function.
Formula:C28H28ClFN6O3Color and Shape:SolidMolecular weight:551.02Adenosine 2',5'-diphosphate sodium
CAS:Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.Formula:C10H15N5NaO10P2Color and Shape:SolidMolecular weight:450.192Israpafant
CAS:Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.Formula:C28H29ClN4SColor and Shape:SolidMolecular weight:489.07CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.81%Color and Shape:SoildMolecular weight:341.49Adrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Formula:C248H381N77O75S5Purity:98%Color and Shape:SolidMolecular weight:5729.5Lintitript
CAS:Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM for CCK1 and CCK2. The Ki value is 0.2 nM for CCK1.Formula:C20H14ClN3O3SPurity:99.28%Color and Shape:SolidMolecular weight:411.86Ref: TM-T15759
1mg50.00€2mg71.00€5mg105.00€1mL*10mM (DMSO)117.00€10mg160.00€25mg344.00€50mg645.00€100mg864.00€PAMP-12 (unmodified) (TFA)
PAMP-12 (unmodified) TFA, an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine secretionFormula:C79H119F3N24O17Color and Shape:SolidMolecular weight:1733.94β-MSH, human
CAS:beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).Formula:C118H174N34O35SPurity:98%Color and Shape:SolidMolecular weight:2660.92VVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Color and Shape:Solid(D-Ala2)-GRF (1-29) amide (human)
CAS:(D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-Formula:C149H246N44O42SColor and Shape:SolidMolecular weight:3357.88G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding.Formula:C59H68N12O11SPurity:98.06%Color and Shape:SolidMolecular weight:1153.33RC-3095
CAS:RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.Formula:C56H79N15O9Purity:98%Color and Shape:SolidMolecular weight:1106.32rGHRH(1-29)NH2
RGHRH (1-29)NH2 is a synthetic peptide that stimulates the secretion of growth hormone (GH).Formula:C155H251N49O40SPurity:98%Color and Shape:SolidMolecular weight:3473.02TT-OAD2
CAS:TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.
Formula:C50H49Cl4N3O6Purity:98%Color and Shape:SolidMolecular weight:929.75Septide
CAS:Septide is an NK1 receptor agonist acting at a site distinct from substance P.Formula:C39H53N7O7SPurity:98%Color and Shape:SolidMolecular weight:763.95Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Formula:C31H44N6O9Purity:98%Color and Shape:SoildMolecular weight:644.72Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1188.38
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