GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Phenylethanolamine A
CAS:Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formula:C19H24N2O4Color and Shape:SolidMolecular weight:344.40CGRP antagonist 6
CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.Color and Shape:Odour Solid[D-Phe12,Leu14]-Bombesin
CAS:Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.Formula:C77H113F3N22O20Purity:98%Color and Shape:SolidMolecular weight:1724.95-MeO-pyr-T
CAS:5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.Formula:C15H20N2OColor and Shape:SolidMolecular weight:244.33Exendin-3/4 (59-86)
Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.Formula:NAPurity:98%Color and Shape:SolidMolecular weight:3055.49γ-2-MSH (41-58), amide
CAS:Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.Formula:C74H100N22O15SPurity:98%Color and Shape:SolidMolecular weight:1569.79U-46619 serinol amide
U-46619 serinol amide is a derivative of U-46619, acting as a stable analog of Thromboxane A2 (TXA2). It effectively functions as a TXA2 agonist, capable of inducing platelet shape change and aggregation.Formula:C24H41NO5Color and Shape:SolidMolecular weight:423.298475-HT7R antagonist 1 free base
CAS:5-HT7R antagonist 1 (free base) is a G protein-biased antagonist for the 5-HT 7 R receptor, with a dissociation constant (K i) of 6.5 nM.Formula:C14H17ClN4Color and Shape:SolidMolecular weight:276.77FXR/TGR5 agonist 1
CAS:FXR/TGR5 agonist 1 acts as an agonist on both FXR and TGR5 receptors and is utilized for treating fatty liver disease.Formula:C31H32ClN3O3Color and Shape:SolidMolecular weight:530.07HAEGT
CAS:HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.Formula:C20H31N7O9Purity:98%Color and Shape:SolidMolecular weight:513.5N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42PG 931 acetate
PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.
Formula:C61H89N15O13Purity:98.74%Color and Shape:SolidMolecular weight:1240.45Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Formula:C22H26O4Color and Shape:SolidMolecular weight:354.446MAO-B-IN-3
MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a KiFormula:C24H25N3O2Purity:98%Color and Shape:SolidMolecular weight:387.47Formoterol O-β-D-Glucuronide
CAS:Formoterol O-β-D-glucuronide is a metabolite of formoterol .Formula:C25H32N2O10Color and Shape:SolidMolecular weight:520.535Prepro VIP (81-122), human
CAS:Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Formula:C202H325N53O64SPurity:98%Color and Shape:SolidMolecular weight:4552.13SGLT1/2-IN-2
CAS:SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).Formula:C23H26F2O7Color and Shape:SolidMolecular weight:452.451α-Helical CRF(9-41)
CAS:Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).Formula:C166H274N46O53S2Purity:98%Color and Shape:SolidMolecular weight:3827PACAP (1-27), human, ovine, rat TFA
PACAP (1-27) TFA is a pacap-38 fragment and PACAP receptor antagonist with IC50s: 3nm (rat PAC1), 2nm (rat VPAC1), 5nm (human VPAC2).Formula:C144H225F3N40O41SPurity:98%Color and Shape:SolidMolecular weight:3261.68(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Formula:C14H22ClNOColor and Shape:SolidMolecular weight:255.78
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