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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • PF-9184

    CAS:
    PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.
    Formula:C21H14Cl2N2O4S
    Purity:97.43%
    Color and Shape:Solid
    Molecular weight:461.32

    Ref: TM-T21738

    25mg
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    50mg
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    1mg
    34.00€
    5mg
    72.00€
    10mg
    98.00€
  • Sarafotoxin S6b

    CAS:
    non-selective endothelin receptor agonist
    Formula:C110H163N27O34S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2567.96

    Ref: TM-TP2290

    1mg
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    100mg
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    500mg
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  • Neuropeptide S(Mouse)

    CAS:
    Endogenous NPSR agonist, EC50 = 3 nM. Boosts Ca2+ levels, activity, wakefulness, reduces anxiety in mice.
    Formula:C93H156N34O27
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2182.47

    Ref: TM-TP1981

    1mg
    867.00€
  • Atilmotin

    CAS:
    Atilmotin is a gastrointestinal agent for treating motility disorders.
    Formula:C86H135N20O19
    Color and Shape:Solid
    Molecular weight:1753.146

    Ref: TM-T30199

    25mg
    1,369.00€
  • Adrenomedullin (AM) (22-52), human

    CAS:
    Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.
    Formula:C159H252N46O48
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3576.04

    Ref: TM-TP1257

    1mg
    178.00€
    5mg
    712.00€
  • Albenatide

    CAS:

    Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.

    Formula:C26H47N7O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:633.76

    Ref: TM-TP2368

    100mg
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    500mg
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  • Cholecystokinin (27-32)-amide

    CAS:
    Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
    Formula:C36H48N8O12S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:881.01

    Ref: TM-T23886

    100mg
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    500mg
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  • Urocortin II, human acetate


    Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.
    Color and Shape:Odour Solid

    Ref: TM-TP3688

    10mg
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    50mg
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  • T-10430


    T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.
    Formula:C17H22N6O
    Color and Shape:Solid
    Molecular weight:326.396

    Ref: TM-T204318

    10mg
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    50mg
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  • K-(D-1-Nal)-FwLL-NH2 TFA


    K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.
    Formula:C53H68F3N9O8
    Color and Shape:Solid
    Molecular weight:1016.16

    Ref: TM-T75948

    5mg
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    50mg
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  • Ecnoglutide

    CAS:
    Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .
    Formula:C194H304N48O61
    Color and Shape:Solid
    Molecular weight:4284.76

    Ref: TM-T76234

    5mg
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    50mg
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  • BQ-123 TFA


    BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.
    Formula:C33H43F3N6O9
    Color and Shape:Solid
    Molecular weight:724.72

    Ref: TM-T73877

    5mg
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    50mg
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  • Neurokinin Receptor (393-407), rat

    CAS:
    Rat NK1R fragment (393-407) binds SP, enabling endocytosis and plasma membrane recycling; key in neurogenic inflammation research.
    Formula:C72H113N17O26S2
    Color and Shape:Solid
    Molecular weight:1696.9

    Ref: TM-T76429

    5mg
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    50mg
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  • Neuropeptide Y (18-36) (porcine)

    CAS:
    "Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."
    Formula:C112H174N36O27
    Color and Shape:Solid
    Molecular weight:2456.8

    Ref: TM-T76357

    5mg
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    50mg
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  • Icatibant

    CAS:
    Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).
    Formula:C59H89N19O13S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:1304.52

    Ref: TM-T15547

    500µg
    883.00€
  • P2Y6R antagonist 1


    P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.
    Color and Shape:Odour Solid

    Ref: TM-T200515

    10mg
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    50mg
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  • Dulaglutide

    CAS:
    Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).
    Color and Shape:Solid

    Ref: TM-T75718

    1mg
    216.00€
    5mg
    635.00€
    10mg
    1,075.00€
    25mg
    1,839.00€
    50mg
    3,055.00€
  • Dotanoc

    CAS:
    Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.
    Formula:C69H94N14O17S2
    Color and Shape:Solid
    Molecular weight:1455.71

    Ref: TM-T24014

    25mg
    1,369.00€
  • BA 1

    CAS:
    Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.
    Formula:C57H76N14O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1133.32

    Ref: TM-TP1913

    1mg
    200.00€
  • RFRP-1(human)

    CAS:
    Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.
    Formula:C67H101N19O14S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1428.72

    Ref: TM-TP1937

    50mg
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    100mg
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