
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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1,8-Cineole
CAS:Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.Formula:C10H18OPurity:97.44% - 97.44%Color and Shape:SolidMolecular weight:154.25PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purity:98%Color and Shape:SolidMolecular weight:2215.49Urocortin, rat
CAS:Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.26Urocortin II, human acetate
Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.Color and Shape:Odour SolidKisspeptin 234
CAS:Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.Formula:C63H78N18O13Purity:98%Color and Shape:SolidMolecular weight:1295.42Sarafotoxin S6c
CAS:Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).Formula:C103H147N27O37S5Purity:98%Color and Shape:SolidMolecular weight:2516Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Color and Shape:SolidMolecular weight:341.091Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Formula:C16H28N6O4Purity:98%Color and Shape:SolidMolecular weight:368.43Cannabinol methyl ether
CAS:Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formula:C22H28O2Color and Shape:SolidMolecular weight:324.5Prostaglandin F2α methyl ester
CAS:Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.Formula:C21H36O5Color and Shape:SolidMolecular weight:368.51Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Formula:C191H330N64O53S3Purity:98%Color and Shape:SolidMolecular weight:4467.29Sphingosine-1-phosphate (d16:1)
CAS:C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.
Formula:C16H34NO5PColor and Shape:SolidMolecular weight:351.424allo-Yohimbine
CAS:allo-Yohimbine is a biochemical.Formula:C21H26N2O3Color and Shape:SolidMolecular weight:354.44Ilatreotide
CAS:Ilatreotide is a Amadori compound of octreotide.Formula:C61H86N10O20S2Purity:98%Color and Shape:SolidMolecular weight:1343.53(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formula:C15H23NO2SPurity:98.19%Color and Shape:SoildMolecular weight:281.41Ref: TM-T60027
1mg73.00€5mg146.00€1mL*10mM (DMSO)155.00€10mg208.00€25mg319.00€50mg447.00€100mg600.00€200mg808.00€RF9
CAS:RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).Formula:C26H38N6O3Purity:98%Color and Shape:SolidMolecular weight:482.62Obestatin(rat)
CAS:Endogenous peptide that suppresses food intake and body weight-gainFormula:C114H174N34O31Purity:98%Color and Shape:SolidMolecular weight:2516.81Pasireotide ditrifluoroacetate
Pasireotide is a stable cyclohexapeptide somatostatin mimic.Formula:C62H68F6N10O13Purity:98%Color and Shape:SolidMolecular weight:1275.25Etelcalcetide
CAS:Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.Formula:C38H73N21O10S2Purity:98%Color and Shape:SolidMolecular weight:1048.2616,16-dimethyl Prostaglandin E1
CAS:16,16-dimethyl Prostaglandin E1 is a PGE1 (T1626) analog that induces bronchoconstriction and vascular smooth muscle contraction and inhibits indomethacin-Formula:C22H38O5Color and Shape:SolidMolecular weight:382.541

