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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • 1,8-Cineole

    CAS:
    Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.
    Formula:C10H18O
    Purity:97.44% - 97.44%
    Color and Shape:Solid
    Molecular weight:154.25

    Ref: TM-T1714

    50mg
    39.00€
    100mg
    50.00€
    500mg
    109.00€
    1g
    160.00€
  • PEN (human)

    CAS:
    PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
    Formula:C97H159N27O32
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2215.49

    Ref: TM-TP1949

    1mg
    138.00€
  • Urocortin, rat

    CAS:
    Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.
    Formula:C206H338N62O64
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4707.26

    Ref: TM-TP1020

    1mg
    1,161.00€
  • Urocortin II, human acetate


    Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.
    Color and Shape:Odour Solid

    Ref: TM-TP3688

    10mg
    To inquire
    50mg
    To inquire
  • Kisspeptin 234

    CAS:
    Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.
    Formula:C63H78N18O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1295.42

    Ref: TM-TP1896

    1mg
    610.00€
  • Sarafotoxin S6c

    CAS:
    Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).
    Formula:C103H147N27O37S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2516

    Ref: TM-TP2120

    100µg
    842.00€
  • Methimepip dihydrobromide

    CAS:
    Methimepip dihydrobromide is a selective H3R agonist.
    Formula:C10H19Br2N3
    Color and Shape:Solid
    Molecular weight:341.091

    Ref: TM-T37727

    200mg
    1,304.00€
  • Bradykinin (1-3)

    CAS:

    Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.

    Formula:C16H28N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.43

    Ref: TM-TP1780

    5mg
    79.00€
    10mg
    97.00€
    25mg
    188.00€
  • Cannabinol methyl ether

    CAS:
    Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.
    Formula:C22H28O2
    Color and Shape:Solid
    Molecular weight:324.5

    Ref: TM-TN7267

    10mg
    To inquire
    50mg
    To inquire
  • Prostaglandin F2α methyl ester

    CAS:
    Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.
    Formula:C21H36O5
    Color and Shape:Solid
    Molecular weight:368.51

    Ref: TM-T38198

    500µg
    105.00€
    1mg
    197.00€
    5mg
    775.00€
    10mg
    1,378.00€
  • Parstatin(human)

    CAS:
    Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.
    Formula:C191H330N64O53S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4467.29

    Ref: TM-TP1965

    1mg
    328.00€
  • Sphingosine-1-phosphate (d16:1)

    CAS:

    C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.

    Formula:C16H34NO5P
    Color and Shape:Solid
    Molecular weight:351.424

    Ref: TM-T37955

    500µg
    677.00€
    1mg
    1,216.00€
    5mg
    3,990.00€
  • allo-Yohimbine

    CAS:
    allo-Yohimbine is a biochemical.
    Formula:C21H26N2O3
    Color and Shape:Solid
    Molecular weight:354.44

    Ref: TM-T29884

    25mg
    1,369.00€
  • Ilatreotide

    CAS:
    Ilatreotide is a Amadori compound of octreotide.
    Formula:C61H86N10O20S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1343.53

    Ref: TM-TP2387

    100mg
    To inquire
    500mg
    To inquire
  • (+)-OSU 6162

    CAS:
    (+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.
    Formula:C15H23NO2S
    Purity:98.19%
    Color and Shape:Soild
    Molecular weight:281.41

    Ref: TM-T60027

    1mg
    73.00€
    5mg
    146.00€
    1mL*10mM (DMSO)
    155.00€
    10mg
    208.00€
    25mg
    319.00€
    50mg
    447.00€
    100mg
    600.00€
    200mg
    808.00€
  • RF9

    CAS:
    RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).
    Formula:C26H38N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:482.62

    Ref: TM-T16738

    1mg
    304.00€
    5mg
    1,108.00€
    10mg
    1,918.00€
  • Obestatin(rat)

    CAS:
    Endogenous peptide that suppresses food intake and body weight-gain
    Formula:C114H174N34O31
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2516.81

    Ref: TM-TP2279

    50mg
    To inquire
    100mg
    To inquire
  • Pasireotide ditrifluoroacetate


    Pasireotide is a stable cyclohexapeptide somatostatin mimic.
    Formula:C62H68F6N10O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1275.25

    Ref: TM-T13811

    50mg
    To inquire
    100mg
    To inquire
    1mg
    162.00€
    5mg
    515.00€
    10mg
    822.00€
  • Etelcalcetide

    CAS:
    Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.
    Formula:C38H73N21O10S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1048.26

    Ref: TM-TP1235

    1mg
    52.00€
    5mg
    104.00€
    10mg
    190.00€
    25mg
    384.00€
  • 16,16-dimethyl Prostaglandin E1

    CAS:
    16,16-dimethyl Prostaglandin E1 is a PGE1 (T1626) analog that induces bronchoconstriction and vascular smooth muscle contraction and inhibits indomethacin-
    Formula:C22H38O5
    Color and Shape:Solid
    Molecular weight:382.541

    Ref: TM-T36214

    1mg
    239.00€
    5mg
    1,018.00€
    10mg
    1,783.00€