GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Adenosine receptor antagonist 1
CAS:A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Formula:C22H15ClFN7OColor and Shape:SolidMolecular weight:447.86MR 409
CAS:MR 409, a selective growth hormone-releasing hormone (GHRH) agonist, exhibits notable neuroprotective properties by augmenting endogenous neurogenesis inFormula:C153H252N44O43Color and Shape:SolidMolecular weight:3395.91[Tyr1]-Somatostatin-14
CAS:[Tyr1]-Somatostatin-14 could binds to SSTR2.Formula:C82H108N18O20S2Molecular weight:1729.9915(S)-15-methyl Prostaglandin F2α methyl ester
CAS:15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.53Amylin (IAPP), feline
Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.Formula:C165H270N52O54S2Purity:98%Color and Shape:SolidMolecular weight:3910.45PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C123H215N39O28SPurity:98%Color and Shape:SolidMolecular weight:2720.33[D-p-Cl-Phe6,Leu17]-VIP TFA
[D-p-Cl-Phe6,Leu17]-VIP TFA acts as a competitive and selective antagonist of the vasoactive intestinal peptide (VIP) receptor, exhibiting an IC50 of 125.8 nM.Formula:C150H240F3ClN44O44Color and Shape:SolidMolecular weight:3456.22HHS-0701
CAS:HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.Formula:C20H20N4O3SPurity:97.24%Color and Shape:SoildMolecular weight:396.46Dexbrompheniramine maleate
CAS:Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.Formula:C20H23BrN2O4Color and Shape:SolidMolecular weight:435.318IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formula:C33H35F3N6O3Purity:98%Color and Shape:SolidMolecular weight:620.66Y4R agonist-1
CAS:Y4R Agonist-1 is a potent agonist of the Y4 receptor, exhibiting a K_i (inhibition constant) value of 0.048 nM.Formula:C51H80N18O11Molecular weight:1121.29Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formula:C58H79N15O15Color and Shape:SolidMolecular weight:1226.34Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Formula:C16H28N6O4Purity:98%Color and Shape:SolidMolecular weight:368.43Parstatin(mouse)
CAS:Peptide inhibits endothelial migration/proliferation (IC50 ~20μM), induces cell cycle arrest, triggers apoptosis, and has cardioprotective effects.Formula:C189H326N58O57S3Purity:98%Color and Shape:SolidMolecular weight:4419.19[Lys8, Lys9]-Neurotensin (8-13)
CAS:[JMV438] is a Neurotensin analog, analgesic via NTS1/NTS2 activation, with K i of 0.33 nM (hNTS1) and 0.95 nM (hNTS2).Formula:C38H64N8O8Molecular weight:760.978Olanzapine Lactam Impurity
CAS:Olanzapine lactam impurity, found in olanzapine, forms under heat or oxidative stress.Formula:C17H20N4O2Color and Shape:SolidMolecular weight:312.373FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formula:C30H28BrCl2N5O4Purity:98%Color and Shape:SolidMolecular weight:673.38GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19Kinetensin
CAS:Kinetensin is a neurotensin-like peptide.Formula:C56H85N17O11Purity:98%Color and Shape:White Lyophilised SolidMolecular weight:1172.38(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formula:C15H23NO2SPurity:98.19%Color and Shape:SoildMolecular weight:281.41Ref: TM-T60027
1mg73.00€5mg146.00€1mL*10mM (DMSO)155.00€10mg208.00€25mg319.00€50mg447.00€100mg600.00€200mg808.00€
