GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
[Ala2] Endothelin-3, human
CAS:[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.Formula:C120H166N26O32S4Color and Shape:SolidMolecular weight:2613.02Dotanoc
CAS:Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Formula:C69H94N14O17S2Color and Shape:SolidMolecular weight:1455.71Gastrin I, rat
CAS:Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.Formula:C94H128N22O31S2Color and Shape:SolidMolecular weight:2126.3Neuropeptide Y (3-36) (porcine)
CAS:Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.Formula:C176H271N53O54Color and Shape:SolidMolecular weight:3993.36Kisspeptin-54(human) TFA
Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.Formula:C258H401N79O78·C2HF3O2Color and Shape:SolidMolecular weight:5971.45Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Formula:C53H71N11O14S2Color and Shape:SolidMolecular weight:1150.33[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Color and Shape:SolidMolecular weight:1033.14(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formula:C52H77N15O14Purity:99.46%Color and Shape:SolidMolecular weight:1136.26Alsactide
CAS:Alsactide, an adrenocorticotropic hormone (ACTH) agonist and a heptadecapeptide analogue, is utilized in the study of the central nervous system [1].Formula:C99H155N29O21SColor and Shape:SolidMolecular weight:2119.53GLP-1(9-36)amide TFA
GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.Formula:C142H215F3N36O45Color and Shape:SolidMolecular weight:3203.43AC-264613
CAS:AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5.Formula:C19H18BrN3O2Purity:98%Color and Shape:SolidMolecular weight:400.28Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Color and Shape:SolidMolecular weight:1979.21Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formula:C58H73F6N11O14S2Color and Shape:SolidMolecular weight:1326.39Amylin (8-37), human
CAS:Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formula:C138H216N42O45Color and Shape:SolidMolecular weight:3183.495Orexin B, rat, mouse TFA
Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.Formula:C128H216F3N45O36SColor and Shape:SolidMolecular weight:3050.42PAMP-12 (unmodified)
CAS:PAMP-12 (unmodified), an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine release fromFormula:C77H118N24O15Color and Shape:SolidMolecular weight:1619.91Adrenotensin (human)
CAS:Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.Formula:C143H224N42O43Color and Shape:SolidMolecular weight:3219.56Zebrafish Kisspeptin-1
CAS:Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Formula:C58H84N16O15Color and Shape:SolidMolecular weight:1245.39Biotin-NeurokininA
Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.Formula:C60H94N16O16S2Color and Shape:SolidMolecular weight:1359.61(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.Formula:C54H76N14O11Color and Shape:SolidMolecular weight:1097.27
![[Ala2] Endothelin-3, human](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76305.webp&w=3840&q=75)
![[Asu1,6-Arg8]Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76510.webp&w=3840&q=75)
