GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Ecraprost
CAS:Ecraprost is used as a prodrug of prostaglandin E1.Formula:C28H48O6Color and Shape:SolidMolecular weight:480.68Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS:Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .Formula:C44H59N13O10SPurity:98%Color and Shape:SolidMolecular weight:962.09Neurokinin B acetate(86933-75-7 free base)
Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological effects.Formula:C57H83N13O16S2Purity:98.53%Color and Shape:SolidMolecular weight:1270.48Cortistatin-14
CAS:Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Formula:C81H114N20O18S2Purity:98.06% - 98.23%Color and Shape:SolidMolecular weight:1720.03Oxaprotiline hydrochloride
CAS:Oxaprotiline hydrochloride is an antidepressant.Formula:C20H24ClNOPurity:98%Color and Shape:SolidMolecular weight:329.86MLN-3897 TFA
MLN-3897 TFA is a potent CCR1 antagonist that inhibits the binding of 125I-MIP-1α to THP-1 cell membranes.Formula:C32H32ClF3N2O6Purity:98.62%Color and Shape:SolidMolecular weight:633.05Ref: TM-T28072L
1mg115.00€5mg245.00€10mg363.00€25mg562.00€50mg775.00€100mg1,035.00€200mg1,406.00€1mL*10mM (DMSO)To inquireCenicriviroc Mesylate
CAS:Cenicriviroc Mesylate (TBR-652 Mesylate) is an oral dual CCR2/CCR5 antagonist exhibiting anti-inflammatory and anti-fibrotic effects for liver fibrosis.Formula:C42H56N4O7S2Purity:98.819%Color and Shape:SolidMolecular weight:793.05Ref: TM-T10756
1mg80.00€5mg127.00€10mg202.00€25mg406.00€50mg692.00€100mg924.00€1mL*10mM (DMSO)177.00€U92016A
CAS:U92016A is a highly potent and selective agonist of 5-HT1A receptor.Formula:C19H25N3Purity:98%Color and Shape:SolidMolecular weight:295.42GHRF, mouse
CAS:GHRF (mouse), a mouse growth hormone-releasing factor, is a 44-amino acid peptide that promotes the synthesis and release of growth hormone [1].Benzquinamide
CAS:Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancerFormula:C22H32N2O5Purity:94.86%Color and Shape:SolidMolecular weight:404.5Prostaglandin F2α Alcohol
CAS:Prostaglandin F2α Alcohol is a PGF2α (T15133) analogue. Prostaglandin F2α Alcohol is an orally active prostaglandin F receptor (FP receptor) agonist.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.5Acmopatide
CAS:Acmopatide (Compound E-153) is a dual agonist of GIP and GLP-1 receptors and can be utilized in diabetes research.Color and Shape:SolidMibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].Purity:98%Color and Shape:Odour SolidGastrin-Releasing Peptide, human
CAS:Gastrin-releasing peptide, released by vagal fibers, stimulates stomach G cells to secrete gastrin, affecting acid secretion and gut motility.Formula:C130H204N38O31S2Purity:98%Color and Shape:SolidMolecular weight:2859.38Bimatoprost cyclohexyl amide
Bimatoprostcyclohexyl amide (N-Cyclohexyl-desamethyl bimatoprost; 17-Phenyl trinor prostaglandin F2α cyclohexyl amide) is an analogue of Bimatoprost. This compound acts as an agonist of the prostaglandin F2α receptor (FP receptor) and can be utilized for research in lowering intraocular pressure and in studies of glaucoma.Color and Shape:Odour SolidMethimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Color and Shape:SolidMolecular weight:341.091Prostaglandin F2α methyl ester
CAS:Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.Formula:C21H36O5Color and Shape:SolidMolecular weight:368.51Prostaglandin E3
CAS:Prostaglandin E3 (PGE3) is an eicosapentaenoic acid (EPA) derivative with anti-inflammatory and anti-tumor activity, and shows anti-proliferative effects.Formula:C20H30O5Purity:98%Color and Shape:SolidMolecular weight:350.45[D-Trp11]-Neurotensin
CAS:[D-Trp11]-Neurotensin, selective NT antagonist in rat hearts, agonist in guinea pig atria/rat stomach, blocks NT-induced hypotension.Formula:C80H122N22O19Molecular weight:1695.991HGS101
HGS101 is a fully humanized CCR5 monoclonal antibody that exhibits high affinity for CCR5. It binds to the second extracellular loop (ECL-2) and functions as a signaling antagonist. HGS101 restores the inhibitory effect of Maraviroc in Maraviroc-resistant HIV-1 infected PBMCs. In an uninfected simian immunodeficiency virus model of rhesus monkeys, HGS101 shows anti-HIV activity by inhibiting CCR5 signaling.Color and Shape:Odour Liquid
