GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Misoprostol acid
CAS:Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.Formula:C21H36O5Purity:98%Color and Shape:SolidMolecular weight:368.51IRL-3630
CAS:IRL 3460 is an enantiomer.Formula:C31H40N4O6SPurity:98%Color and Shape:SolidMolecular weight:596.74Lisuride maleate
CAS:Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.Formula:C24H30N4O5Purity:99.85%Color and Shape:SolidMolecular weight:454.52Ref: TM-T8775
1mg204.00€5mg627.00€10mg898.00€25mg1,346.00€50mg1,745.00€100mg2,382.00€1mL*10mM (DMSO)627.00€SB 201146
CAS:SB 201146 is a leukotriene B4 antagonist with high affinity.Formula:C30H35LiN2O5SColor and Shape:SolidMolecular weight:542.61IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formula:C33H35F3N6O3Purity:98%Color and Shape:SolidMolecular weight:620.66Kinetensin
CAS:Kinetensin is a neurotensin-like peptide.Formula:C56H85N17O11Purity:98%Color and Shape:White Lyophilised SolidMolecular weight:1172.38Amylin, amide, rat
CAS:Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.Formula:C167H272N52O53S2Purity:99.92%Color and Shape:SolidMolecular weight:3920.44Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.462Sphingosine-1-phosphate (d16:1)
CAS:C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.
Formula:C16H34NO5PColor and Shape:SolidMolecular weight:351.424Apraglutide
CAS:Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.Formula:C172H263N43O52Purity:98%Color and Shape:SolidMolecular weight:3765.25(±)-4-hydroxy Propranolol β-D-Glucuronide
CAS:(±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol , which is a metabolite of propranolol.Formula:C22H29NO9Color and Shape:SolidMolecular weight:451.47O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS:O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Formula:C11H11NO3Color and Shape:SolidMolecular weight:205.213Cannabigerorcin
CAS:Cannabigerorcin, a phytocannabinoid, serves as an analytical reference standard. It is designated for research and forensic applications.Formula:C17H24O2Color and Shape:SolidMolecular weight:260.377Dexbrompheniramine maleate
CAS:Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.Formula:C20H23BrN2O4Color and Shape:SolidMolecular weight:435.318PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C123H215N39O28SPurity:98%Color and Shape:SolidMolecular weight:2720.33N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Formula:C15H22ClNO2Purity:98.85% - 99.54%Color and Shape:SolidMolecular weight:283.79CIA-1 (Free base)
CAS:CIA-1, a COUP-TFII inhibitor, has IC50 of 1.2-7.6 μM in prostate cancer cells; inhibits tumor growth in mouse prostate cancer.Formula:C17H19N3O2SPurity:99%Color and Shape:SolidMolecular weight:329.42Vanicoside E
CAS:Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formula:C53H52O22Color and Shape:SolidMolecular weight:1040.9711β-Prostaglandin E2
CAS:11β-PGE2 is the C-11 epimer of PGE2.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47Rp-UTP-α-S tetrasodium
Rp-UTP-α-S (tetrasodium) is a nucleotide agonist of the purinergic P2Y2 and P2Y4 receptors. It can induce the accumulation of inositol phosphate in 1321N1 cells expressing P2Y2 or P2Y4, with EC50 values of 5.4 and 27 μM, respectively.Color and Shape:Odour Solid
